ECSP056162A - Cristal derivado de benzimidazol y procedimiento para producirlo - Google Patents

Cristal derivado de benzimidazol y procedimiento para producirlo

Info

Publication number
ECSP056162A
ECSP056162A EC2005006162A ECSP056162A ECSP056162A EC SP056162 A ECSP056162 A EC SP056162A EC 2005006162 A EC2005006162 A EC 2005006162A EC SP056162 A ECSP056162 A EC SP056162A EC SP056162 A ECSP056162 A EC SP056162A
Authority
EC
Ecuador
Prior art keywords
benzimidazol
procedure
produce
crystal derived
derived
Prior art date
Application number
EC2005006162A
Other languages
English (en)
Inventor
Mitsuru Teramoto
Naoki Tsuchiya
Hiroshi Saitoh
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33447189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP056162(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of ECSP056162A publication Critical patent/ECSP056162A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se proveen varias formas cristalinas de ácido 4-(1-((4-metilbenzotiofen-3-il)metil)benzimidazol-2-iltio)butanoico a partir de un solvente, y un proceso para la preparación de las mismas.
EC2005006162A 2003-05-14 2005-11-14 Cristal derivado de benzimidazol y procedimiento para producirlo ECSP056162A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2003135567 2003-05-14

Publications (1)

Publication Number Publication Date
ECSP056162A true ECSP056162A (es) 2006-04-19

Family

ID=33447189

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2005006162A ECSP056162A (es) 2003-05-14 2005-11-14 Cristal derivado de benzimidazol y procedimiento para producirlo

Country Status (25)

Country Link
US (1) US7649008B2 (es)
EP (1) EP1626048A4 (es)
JP (1) JPWO2004101551A1 (es)
KR (1) KR20060011997A (es)
CN (1) CN1788007A (es)
AR (1) AR044340A1 (es)
AU (1) AU2004238708A1 (es)
BR (1) BRPI0410266A (es)
CA (1) CA2523978A1 (es)
CL (1) CL2004001034A1 (es)
CO (1) CO5660259A2 (es)
EC (1) ECSP056162A (es)
IS (1) IS8177A (es)
MA (1) MA27805A1 (es)
MX (1) MXPA05011851A (es)
NO (1) NO20055181L (es)
NZ (1) NZ542978A (es)
PE (1) PE20050203A1 (es)
RU (1) RU2332417C2 (es)
SA (1) SA04250117B1 (es)
TN (1) TNSN05288A1 (es)
TW (1) TW200505911A (es)
UA (1) UA81493C2 (es)
WO (1) WO2004101551A1 (es)
ZA (1) ZA200508640B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CL2004001034A1 (es) 2003-05-14 2005-03-28 Teijin Pharma Ltd Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r
KR20060120601A (ko) * 2003-08-22 2006-11-27 데이진 화-마 가부시키가이샤 키마제 저해제를 유효 성분으로서 함유하는 약제
JPWO2006052026A1 (ja) * 2004-11-12 2008-05-29 帝人ファーマ株式会社 ベンズイミダゾール誘導体の酸性塩及びその結晶
JP2016150917A (ja) * 2015-02-17 2016-08-22 株式会社トクヤマ バルサルタンの結晶の製造方法
WO2022257845A1 (zh) * 2021-06-11 2022-12-15 苏州科睿思制药有限公司 Tolebrutinib的晶型及其制备方法和用途

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0237608B1 (de) 1986-03-21 1992-01-29 HEUMANN PHARMA GMBH & CO Kristalline, wasserfreie Sigma -Form von 2-[4-(2-Furoyl-(2-piperazin)-1-yl]-4-amino-6,7-dimethoxychinazolinhydrochlorid und Verfahren zu ihrer Herstellung
US5015646A (en) 1987-08-28 1991-05-14 Bristol-Myers Squibb Co. Pharmaceutically useful polymorphic modification of buspirone
KR100287579B1 (ko) 1994-05-31 2001-05-02 야스이 쇼사꾸 나프탈렌유도체
ES2150353B1 (es) 1998-04-15 2001-07-01 Esteve Labor Dr Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos.
US20040010004A1 (en) * 2000-01-17 2004-01-15 Naoki Tsuchiya Benzimidazole derivatives
HUP0103256A3 (en) 1998-07-15 2002-05-28 Teijin Ltd Thiobenzimidazole derivatives and pharmaceutical compositions containing the compounds
ES2295128T3 (es) 2000-01-17 2008-04-16 Teijin Pharma Limited Derivados de bencimidazol como inhibidores de quimasa humana.
EP1362854B1 (en) 2001-02-22 2007-10-31 Teijin Pharma Limited Benzo[b[thiophene derivatives and process for producing the same
US6774245B2 (en) 2001-05-07 2004-08-10 Teijin Limited 3-Hydroxymethylbenzo[b]thiophene derivatives and process for their preparation
JP4173098B2 (ja) * 2001-08-24 2008-10-29 帝人株式会社 キマーゼ阻害剤及びａｃｅ阻害剤を有効成分として含有する薬剤
CL2004001034A1 (es) 2003-05-14 2005-03-28 Teijin Pharma Ltd Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r

Also Published As

Publication number Publication date
CL2004001034A1 (es) 2005-03-28
TW200505911A (en) 2005-02-16
PE20050203A1 (es) 2005-03-26
US7649008B2 (en) 2010-01-19
CN1788007A (zh) 2006-06-14
BRPI0410266A (pt) 2006-05-16
SA04250117B1 (ar) 2009-09-02
CA2523978A1 (en) 2004-11-25
TNSN05288A1 (en) 2007-07-10
US20060293375A1 (en) 2006-12-28
ZA200508640B (en) 2007-02-28
RU2332417C2 (ru) 2008-08-27
MXPA05011851A (es) 2006-02-17
MA27805A1 (fr) 2006-03-01
EP1626048A4 (en) 2008-11-12
JPWO2004101551A1 (ja) 2006-07-13
IS8177A (is) 2005-12-13
UA81493C2 (en) 2008-01-10
NZ542978A (en) 2009-04-30
NO20055181D0 (no) 2005-11-03
AR044340A1 (es) 2005-09-07
AU2004238708A1 (en) 2004-11-25
CO5660259A2 (es) 2006-07-31
RU2005138868A (ru) 2006-07-10
KR20060011997A (ko) 2006-02-06
WO2004101551A1 (ja) 2004-11-25
NO20055181L (no) 2006-01-24
EP1626048A1 (en) 2006-02-15

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