ECSP088762A - Tratamiento del dolor - Google Patents

Tratamiento del dolor

Info

Publication number
ECSP088762A
ECSP088762A EC2008008762A ECSP088762A ECSP088762A EC SP088762 A ECSP088762 A EC SP088762A EC 2008008762 A EC2008008762 A EC 2008008762A EC SP088762 A ECSP088762 A EC SP088762A EC SP088762 A ECSP088762 A EC SP088762A
Authority
EC
Ecuador
Prior art keywords
pain
pain treatment
mammal
compound
formula
Prior art date
Application number
EC2008008762A
Other languages
English (en)
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ECSP088762A publication Critical patent/ECSP088762A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Esta invención proporciona un método para tratar el dolor en un mamífero que incluye administrar a un mamífero que necesita dicho tratamiento una cantidad efectiva para tratar el dolor de un compuesto de la Fórmula I: Io una sal farmacéuticamente aceptable del mismo, donde cada uno de R1, R2, R3, R4, R5, R6, n, y m es como se definió y describió en la presente. La presente invención también proporciona composiciones farmacéuticas para tratar el dolor que contienen una cantidad efectiva para tratar el dolor de un compuesto de Fórmula I.
EC2008008762A 2006-03-24 2008-09-23 Tratamiento del dolor ECSP088762A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78563306P 2006-03-24 2006-03-24

Publications (1)

Publication Number Publication Date
ECSP088762A true ECSP088762A (es) 2008-10-31

Family

ID=38332439

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008762A ECSP088762A (es) 2006-03-24 2008-09-23 Tratamiento del dolor

Country Status (16)

Country Link
US (1) US20070225277A1 (es)
EP (1) EP1998781A2 (es)
JP (1) JP2009531434A (es)
KR (1) KR20080110759A (es)
CN (1) CN101410118A (es)
AR (1) AR060089A1 (es)
AU (1) AU2007230997A1 (es)
BR (1) BRPI0709163A2 (es)
CA (1) CA2644656A1 (es)
EC (1) ECSP088762A (es)
IL (1) IL193748A0 (es)
MX (1) MX2008012092A (es)
PA (1) PA8720901A1 (es)
PE (1) PE20081192A1 (es)
TW (1) TW200806299A (es)
WO (1) WO2007112000A2 (es)

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RU2015140748A (ru) * 2010-05-21 2018-12-26 Эббви Инк. Модуляторы 5-нт рецепторов и способы их применения
US20140080813A1 (en) 2012-09-14 2014-03-20 AbbVie Deutschland GmbH & Co. KG Tricyclic quinoline and quinoxaline derivatives
KR20150056608A (ko) * 2012-09-14 2015-05-26 아비에 도이치란트 게엠베하 운트 콤파니 카게 트리사이클릭 퀴놀린 및 퀴녹살린 유도체
EP3116873B1 (en) 2014-03-14 2018-02-28 AbbVie Deutschland GmbH & Co. KG Hexahydrodiazepinoquinolines carrying a cyclic radical
US9540376B2 (en) 2014-03-14 2017-01-10 AbbVie Deutschland GmbH & Co. KG Hexahydrodiazepinoquinolines carrying a substituted alkyl radical
WO2016210431A1 (en) * 2015-06-26 2016-12-29 Wright State University Method of treating sepsis-induced myopathy
US20180339996A1 (en) 2015-11-25 2018-11-29 AbbVie Deutschland GmbH & Co. KG Hexahydropyrazinobenz- or -pyrido-oxazepines carrying an oxygen-containing substituent and use thereof in the treatment of 5-ht2c-dependent disorders
US20200039930A1 (en) 2017-03-21 2020-02-06 AbbVie Deutschland GmbH & Co. KG Proline amide compounds and their azetidine analogues carrying a specifically substituted benzyl radical

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Also Published As

Publication number Publication date
AR060089A1 (es) 2008-05-21
MX2008012092A (es) 2008-10-03
CA2644656A1 (en) 2007-10-04
CN101410118A (zh) 2009-04-15
PE20081192A1 (es) 2008-10-07
IL193748A0 (en) 2009-08-03
WO2007112000A2 (en) 2007-10-04
US20070225277A1 (en) 2007-09-27
PA8720901A1 (es) 2008-11-19
WO2007112000A3 (en) 2008-01-17
TW200806299A (en) 2008-02-01
EP1998781A2 (en) 2008-12-10
BRPI0709163A2 (pt) 2011-06-28
JP2009531434A (ja) 2009-09-03
AU2007230997A1 (en) 2007-10-04
KR20080110759A (ko) 2008-12-19

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