ECSP088805A - 2-(piridin-2-il)-pirimidinas como fungicidas - Google Patents
2-(piridin-2-il)-pirimidinas como fungicidasInfo
- Publication number
- ECSP088805A ECSP088805A EC2008008805A ECSP088805A ECSP088805A EC SP088805 A ECSP088805 A EC SP088805A EC 2008008805 A EC2008008805 A EC 2008008805A EC SP088805 A ECSP088805 A EC SP088805A EC SP088805 A ECSP088805 A EC SP088805A
- Authority
- EC
- Ecuador
- Prior art keywords
- alkyl
- membered
- halogenalkoxy
- halogenalkyl
- alkoxy
- Prior art date
Links
- 239000000417 fungicide Substances 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 3
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 3
- 125000001188 haloalkyl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 150000002431 hydrogen Chemical group 0.000 abstract 3
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 3
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 2
- JCXJVPUVTGWSNB-UHFFFAOYSA-N Nitrogen dioxide Chemical group O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 229910052717 sulfur Chemical group 0.000 abstract 2
- 239000011593 sulfur Chemical group 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- YJVKLLJCUMQBHN-UHFFFAOYSA-N 2-pyridin-2-ylpyrimidine Chemical class N1=CC=CC=C1C1=NC=CC=N1 YJVKLLJCUMQBHN-UHFFFAOYSA-N 0.000 abstract 1
- 125000001054 5 membered carbocyclic group Chemical group 0.000 abstract 1
- 125000006163 5-membered heteroaryl group Chemical group 0.000 abstract 1
- 125000004008 6 membered carbocyclic group Chemical group 0.000 abstract 1
- 125000001960 7 membered carbocyclic group Chemical group 0.000 abstract 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- 241000233866 Fungi Species 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000006413 ring segment Chemical group 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se refiere a 2-(piridin-2-il)-pirimidinas y su uso para el combate de hongos dañinos, así como a agentes fitoprotectores, que contienen estos compuestos como componente eficaz. en donde: Q es un carbociclo condensado, saturado, de 5, 6 ó 7 miembros o un heterociclo de 5, 6 ó 7 miembros que presenta, además de los miembros del anillo de carbono, uno o dos heteroátomos seleccionados entre oxígeno y azufre como miembros del anillo, en donde el carbociclo y el heterociclo no están sustituidos o presentan 1, 2, 3 ó 4 grupos alquilo C1-C4 como sustituyentes; R1 es hidrógeno, OH, alquilo C1-C4, alcoxi C1-C4, halogenalquilo C1-C4, halogenalcoxi C1-C4 o halógeno; R2 es hidrógeno, NO2, halógeno, alquilo C1-C6, cicloalquilo C3-C6, alcoxi C1-C6, halogenalquilo C1-C6 o halogenalcoxi C1-C6; R3 es hidrógeno, halógeno, alquilo C1-C4, alcoxi C1-C4, halogenalquilo C1-C4 o halogenalcoxi C1-C4; R4 es fenilo, heteroarilo de 5 miembros que presenta 1, 2, 3 ó 4 átomos de nitrógeno o 1 heteroátomo seleccionado entre oxígeno y azufre y eventualmente 1, 2 ó 3 átomos de nitrógeno como átomos del anillo, o hetarilo de 6 miembros, que presenta 1, 2, 3 ó 4 átomos de nitrógeno como miembros del anillo, en donde el fenilo, el hetarilo de 5 y 6 miembros pueden presentar 1, 2, 3 ó 4 sustituyentes Ra..
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06007744 | 2006-04-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP088805A true ECSP088805A (es) | 2008-11-27 |
Family
ID=38261469
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2008008805A ECSP088805A (es) | 2006-04-12 | 2008-10-08 | 2-(piridin-2-il)-pirimidinas como fungicidas |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20090105072A1 (es) |
| EP (1) | EP2010515A1 (es) |
| JP (1) | JP2009534318A (es) |
| KR (1) | KR20090006191A (es) |
| CN (1) | CN101460475A (es) |
| AR (1) | AR060438A1 (es) |
| AU (1) | AU2007235863A1 (es) |
| BR (1) | BRPI0710010A2 (es) |
| CA (1) | CA2647945A1 (es) |
| CR (1) | CR10344A (es) |
| EA (1) | EA200802052A1 (es) |
| EC (1) | ECSP088805A (es) |
| IL (1) | IL194549A0 (es) |
| MA (1) | MA30397B1 (es) |
| ME (1) | MEP27208A (es) |
| MX (1) | MX2008012513A (es) |
| NZ (1) | NZ571611A (es) |
| TW (1) | TW200808760A (es) |
| UA (1) | UA89000C2 (es) |
| WO (1) | WO2007116079A1 (es) |
| ZA (1) | ZA200809557B (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ596546A (en) * | 2009-05-29 | 2012-12-21 | Syngenta Participations Ag | Substituted quinazolines as fungicides |
| CN102770433A (zh) * | 2010-02-24 | 2012-11-07 | 先正达参股股份有限公司 | 新颖的杀微生物剂 |
| EP2632913A1 (en) | 2010-10-28 | 2013-09-04 | Syngenta Participations AG | Novel microbicides |
| WO2012066122A1 (en) | 2010-11-18 | 2012-05-24 | Syngenta Participations Ag | 2 - (pyridin- 2 -yl) -quinazoline derivatives and their use as microbicides |
| WO2013026900A1 (en) * | 2011-08-23 | 2013-02-28 | Syngenta Participations Ag | Pyridine derivatives as microbiocides |
| AR087609A1 (es) | 2011-08-23 | 2014-04-03 | Syngenta Participations Ag | Microbiocidas |
| CN104583215B (zh) | 2012-08-30 | 2016-12-07 | 霍夫曼-拉罗奇有限公司 | 二噁烯并-和噁嗪-[2,3-d]嘧啶pi3k抑制剂化合物及使用方法 |
| JP2021008403A (ja) * | 2017-09-26 | 2021-01-28 | 日本曹達株式会社 | １，３，５，６−テトラ置換チエノ［２，３−ｄ］ピリミジン−２，４（１Ｈ，３Ｈ）ジオン化合物および農園芸用殺菌剤 |
| EP4155299A4 (en) * | 2020-05-19 | 2024-07-10 | Unimatec Co., Ltd. | Fluoropyrimidine compound and fluoropyrimidinone compound |
| CN112939939B (zh) * | 2021-03-11 | 2023-12-26 | 西华大学 | 2-(4-氯苯基)吡啶类化合物及其在农药中的应用 |
| CN112979620B (zh) * | 2021-03-11 | 2023-11-10 | 湖南道仕医药科技有限公司 | 6-甲氧基吡啶衍生物及其在农药中的应用 |
| WO2023004138A1 (en) * | 2021-07-22 | 2023-01-26 | Bhaskar Das | Agonists of tyro3 as protection against podocyte injury in kidney glomerular disease |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH23565A (en) * | 1986-09-05 | 1989-08-25 | Sumitomo Chemical Co | Novel pyrimidinylpyrimidine derivatives and a plant disease protectant containing them as the active ingredient |
| JP2517981B2 (ja) * | 1986-09-05 | 1996-07-24 | 住友化学工業株式会社 | ピリジルピリミジン誘導体およびそれを有効成分とする植物病害防除剤 |
| JPH04224580A (ja) * | 1990-12-25 | 1992-08-13 | Nippon Soda Co Ltd | ピリミジン誘導体、その製造方法及び農園芸用殺菌剤 |
| PE20060115A1 (es) * | 2004-07-23 | 2006-03-23 | Basf Ag | 2-(piridin-2-il)-pirimidinas como agentes fungicidas |
-
2007
- 2007-04-11 TW TW096112734A patent/TW200808760A/zh unknown
- 2007-04-11 EA EA200802052A patent/EA200802052A1/ru unknown
- 2007-04-11 BR BRPI0710010-8A patent/BRPI0710010A2/pt not_active IP Right Cessation
- 2007-04-11 NZ NZ571611A patent/NZ571611A/en unknown
- 2007-04-11 EP EP07727984A patent/EP2010515A1/de not_active Withdrawn
- 2007-04-11 CA CA002647945A patent/CA2647945A1/en not_active Abandoned
- 2007-04-11 UA UAA200812906A patent/UA89000C2/ru unknown
- 2007-04-11 MX MX2008012513A patent/MX2008012513A/es not_active Application Discontinuation
- 2007-04-11 CN CNA2007800204007A patent/CN101460475A/zh active Pending
- 2007-04-11 KR KR1020087027565A patent/KR20090006191A/ko not_active Withdrawn
- 2007-04-11 ME MEP-272/08A patent/MEP27208A/xx unknown
- 2007-04-11 AU AU2007235863A patent/AU2007235863A1/en not_active Abandoned
- 2007-04-11 JP JP2009504737A patent/JP2009534318A/ja active Pending
- 2007-04-11 WO PCT/EP2007/053516 patent/WO2007116079A1/de not_active Ceased
- 2007-04-11 US US12/225,862 patent/US20090105072A1/en not_active Abandoned
- 2007-04-12 AR ARP070101568A patent/AR060438A1/es not_active Application Discontinuation
-
2008
- 2008-10-06 IL IL194549A patent/IL194549A0/en unknown
- 2008-10-06 CR CR10344A patent/CR10344A/es not_active Application Discontinuation
- 2008-10-08 EC EC2008008805A patent/ECSP088805A/es unknown
- 2008-11-04 MA MA31354A patent/MA30397B1/fr unknown
- 2008-11-10 ZA ZA200809557A patent/ZA200809557B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20090105072A1 (en) | 2009-04-23 |
| JP2009534318A (ja) | 2009-09-24 |
| MEP27208A (en) | 2010-06-10 |
| KR20090006191A (ko) | 2009-01-14 |
| IL194549A0 (en) | 2009-08-03 |
| CN101460475A (zh) | 2009-06-17 |
| TW200808760A (en) | 2008-02-16 |
| ZA200809557B (en) | 2010-01-27 |
| CR10344A (es) | 2008-10-29 |
| CA2647945A1 (en) | 2007-10-18 |
| AR060438A1 (es) | 2008-06-18 |
| MA30397B1 (fr) | 2009-05-04 |
| AU2007235863A1 (en) | 2007-10-18 |
| NZ571611A (en) | 2011-06-30 |
| EP2010515A1 (de) | 2009-01-07 |
| UA89000C2 (ru) | 2009-12-10 |
| EA200802052A1 (ru) | 2009-04-28 |
| MX2008012513A (es) | 2008-10-10 |
| WO2007116079A1 (de) | 2007-10-18 |
| BRPI0710010A2 (pt) | 2011-08-02 |
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