ECSP089024A - Camsilato de (s)-(-)-amlodipino o hidrato del mismo y composición farmacéutica que comprende el mismo - Google Patents
Camsilato de (s)-(-)-amlodipino o hidrato del mismo y composición farmacéutica que comprende el mismoInfo
- Publication number
- ECSP089024A ECSP089024A EC2008009024A ECSP089024A ECSP089024A EC SP089024 A ECSP089024 A EC SP089024A EC 2008009024 A EC2008009024 A EC 2008009024A EC SP089024 A ECSP089024 A EC SP089024A EC SP089024 A ECSP089024 A EC SP089024A
- Authority
- EC
- Ecuador
- Prior art keywords
- same
- pharmaceutical composition
- camsilato
- amlodipino
- hydration
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 230000036571 hydration Effects 0.000 title 1
- 238000006703 hydration reaction Methods 0.000 title 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicinal Preparation (AREA)
Abstract
La invención se relaciona con un camsilato de (S)-(-)-amlodipino o un hidrato del mismo que tiene buena fotoestabilidad y alta solubilidad, y una composición farmacéutica que comprende el mismo, la cual puede utilizarse eficientemente en el tratamiento de enfermedades cardiovasculares.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020060068401A KR100913791B1 (ko) | 2006-07-21 | 2006-07-21 | (s)-(-)-암로디핀 캠실레이트 또는 이의 수화물 및 이를함유하는 약학적 조성물 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP089024A true ECSP089024A (es) | 2009-01-30 |
Family
ID=38956963
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2008009024A ECSP089024A (es) | 2006-07-21 | 2008-12-31 | Camsilato de (s)-(-)-amlodipino o hidrato del mismo y composición farmacéutica que comprende el mismo |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20090326234A1 (es) |
| EP (1) | EP2044022A1 (es) |
| JP (1) | JP2009544695A (es) |
| KR (1) | KR100913791B1 (es) |
| CN (1) | CN101495451B (es) |
| AR (1) | AR062009A1 (es) |
| AU (1) | AU2007276038B2 (es) |
| BR (1) | BRPI0714313A2 (es) |
| CA (1) | CA2658384C (es) |
| EC (1) | ECSP089024A (es) |
| IL (1) | IL196318A0 (es) |
| MX (1) | MX2009000454A (es) |
| MY (1) | MY152884A (es) |
| NO (1) | NO20090819L (es) |
| NZ (1) | NZ574006A (es) |
| RU (1) | RU2403241C1 (es) |
| UA (1) | UA93724C2 (es) |
| WO (1) | WO2008010659A1 (es) |
| ZA (1) | ZA200900231B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA33056B1 (fr) | 2009-01-23 | 2012-02-01 | Hanmi Holding Co Ltd | Composition pharmaceutique solide comprenant de l'amlodipine et du losartan et son procede de fabrication |
| ES2363964B1 (es) | 2009-11-20 | 2012-08-22 | Gp Pharm, S.A. | Cápsulas de principios activos farmacéuticos y ésteres de ácidos grasos poliinsaturados. |
| KR102521227B1 (ko) * | 2018-09-12 | 2023-04-13 | 후지필름 가부시키가이샤 | 약액, 기판의 처리 방법 |
| CN113041244B (zh) | 2019-11-08 | 2022-06-21 | 施慧达药业集团(吉林)有限公司 | 含苯磺酸左氨氯地平水合物的组合物及其制备方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9405833D0 (en) * | 1994-03-24 | 1994-05-11 | Pfizer Ltd | Separation of the enantiomers of amlodipine |
| PL189666B1 (pl) * | 1998-04-09 | 2005-09-30 | Adamed Sp Z Oo | Sposób otrzymywania benzenosulfonianu amlodypiny |
| WO2002079518A1 (en) | 2001-03-29 | 2002-10-10 | Chugai Seiyaku Kabushiki Kaisha | A method for genotyping individuals for multiple snps |
| KR100452491B1 (ko) * | 2001-03-29 | 2004-10-12 | 한미약품 주식회사 | 신규한 결정형 암로디핀 캠실레이트 염 및 그의 제조방법 |
| CN1152013C (zh) * | 2001-11-22 | 2004-06-02 | 张喜田 | 一类左旋氨氯地平盐的水合物及其制剂 |
| KR20040011751A (ko) * | 2002-07-30 | 2004-02-11 | 씨제이 주식회사 | 암로디핀의 유기산염 |
| EP1587792B1 (en) * | 2003-01-27 | 2014-08-27 | Hanmi Science Co., Ltd. | Stable amorphous amlodipine camsylate, process for preparing same and composition for oral administration thereof |
| KR100841409B1 (ko) * | 2003-12-16 | 2008-06-25 | 에스케이케미칼주식회사 | 암로디핀 겐티세이트 염과 이의 제조방법 |
| ES2307209T3 (es) * | 2004-10-20 | 2008-11-16 | Emcure Pharmaceuticals Limited | Procedimiento de produccion de un enantiomero de amlodipina con una pureza optica alta. |
| GB0502509D0 (en) * | 2005-02-07 | 2005-03-16 | Pfizer Ltd | Novel salt form of a dopamine agonist |
-
2006
- 2006-07-21 KR KR1020060068401A patent/KR100913791B1/ko not_active Expired - Fee Related
-
2007
- 2007-07-16 BR BRPI0714313-3A patent/BRPI0714313A2/pt not_active IP Right Cessation
- 2007-07-16 EP EP07768773A patent/EP2044022A1/en active Pending
- 2007-07-16 CA CA2658384A patent/CA2658384C/en not_active Expired - Fee Related
- 2007-07-16 WO PCT/KR2007/003444 patent/WO2008010659A1/en not_active Ceased
- 2007-07-16 MY MYPI20090230 patent/MY152884A/en unknown
- 2007-07-16 AU AU2007276038A patent/AU2007276038B2/en not_active Ceased
- 2007-07-16 MX MX2009000454A patent/MX2009000454A/es not_active Application Discontinuation
- 2007-07-16 US US12/374,087 patent/US20090326234A1/en not_active Abandoned
- 2007-07-16 ZA ZA200900231A patent/ZA200900231B/xx unknown
- 2007-07-16 UA UAA200901416A patent/UA93724C2/ru unknown
- 2007-07-16 NZ NZ574006A patent/NZ574006A/en not_active IP Right Cessation
- 2007-07-16 CN CN2007800277402A patent/CN101495451B/zh not_active Expired - Fee Related
- 2007-07-16 JP JP2009521693A patent/JP2009544695A/ja active Pending
- 2007-07-16 RU RU2009106073/04A patent/RU2403241C1/ru not_active IP Right Cessation
- 2007-07-20 AR ARP070103244A patent/AR062009A1/es not_active Application Discontinuation
-
2008
- 2008-12-31 EC EC2008009024A patent/ECSP089024A/es unknown
-
2009
- 2009-01-01 IL IL196318A patent/IL196318A0/en unknown
- 2009-02-20 NO NO20090819A patent/NO20090819L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2403241C1 (ru) | 2010-11-10 |
| AU2007276038B2 (en) | 2011-06-16 |
| JP2009544695A (ja) | 2009-12-17 |
| MY152884A (en) | 2014-11-28 |
| ZA200900231B (en) | 2010-04-28 |
| KR20080008752A (ko) | 2008-01-24 |
| MX2009000454A (es) | 2009-01-28 |
| KR100913791B1 (ko) | 2009-08-26 |
| AU2007276038A1 (en) | 2008-01-24 |
| WO2008010659A1 (en) | 2008-01-24 |
| IL196318A0 (en) | 2009-09-22 |
| AR062009A1 (es) | 2008-08-10 |
| CA2658384C (en) | 2012-01-17 |
| NZ574006A (en) | 2010-09-30 |
| RU2009106073A (ru) | 2010-08-27 |
| CN101495451A (zh) | 2009-07-29 |
| EP2044022A1 (en) | 2009-04-08 |
| CA2658384A1 (en) | 2008-01-24 |
| NO20090819L (no) | 2009-02-20 |
| UA93724C2 (ru) | 2011-03-10 |
| US20090326234A1 (en) | 2009-12-31 |
| BRPI0714313A2 (pt) | 2013-04-02 |
| CN101495451B (zh) | 2012-07-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CL2016002589A1 (es) | Uso del compuesto genz-112638 (eliglustat), inhibidor de glucosilceramida sintasa, en el tratamiento de la enfermedad de gaucher y enfermedad de fabry (divisional de solicitud 201201348). | |
| CL2011002787A1 (es) | Compuestos derivados de 1-cianoetilheterociclilcarboxamida sustituidos, inhibidores de dipeptidilpeptidasa i (dppi) o catepsina c; composicion farmaceutica; combinacion faramceutica; y su uso en el tratamiento del asma, la enfermedad obstructiva cronica o la rinitis alergica. | |
| CL2008002369A1 (es) | Compuestos derivados de piridin-3-il-oxipiridin-2-il-amino, inhibidores de alk5; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento del cancer. | |
| UY33397A (es) | Forma sólida de un naftaleno carboxamida | |
| EA200900091A1 (ru) | Новые показания к применению прямых ингибиторов тромбина в лечении сердечно-сосудистых заболеваний | |
| CL2008001855A1 (es) | Compuestos ciclicos condensados derivados del boro; composicion farmaceutica; y uso en el tratamiento y/o prevencion de una enfermedad infecciosa. | |
| BR112014012524A2 (pt) | composições compreendendo um componente de estabilidade do prazo de validade | |
| CL2007001992A1 (es) | Compuestos derivados de pirimidilciclopentanos; procedimiento de preparacion; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de una enfermedad inflamatoria, hiperproliferante, cardiovascular, neurodege | |
| CL2007002866A1 (es) | Compuestos derivados de 6-sustituidos-2-(bencimidazolil) purina y purinona; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de enfermedades autoinmunes, enfermedad inflamatoria, enfermedad mediada por m | |
| EA201300242A1 (ru) | Фармацевтические композиции, содержащие замещенные ациланилиды | |
| CL2010001483A1 (es) | Compuestos derivados de 5-fenil-1h-piridin-2-ona y 6-fenil-2h-piridazin-3-ona, inhibidores de tirosina-quinasa (btk); composicion farmaceutica que comprende a dichos compuestos y su uso para el tratamiento de un estado patologico inflamatorio y/o autoinmune. | |
| NO20081636L (no) | FAP - inhibitorer | |
| CL2007002167A1 (es) | Compuestos derivados de indol, antagonistas iap; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de cancer. | |
| CL2010001361A1 (es) | Compuestos derivados de piperidin-carboxamida, inhibidores de renina; composicion farmaceutica que los comprende; y uso en el tratamiento o prevencion de una enfermedad circulatoria, hipertension y/o diversos daños organicos atribuibles a la hipertension. | |
| EA201071315A1 (ru) | Ингибиторы протеазы вируса гепатита с | |
| EA200970916A1 (ru) | Соединения 5,6-дигидро-1н-пиридин-2-она | |
| CL2011000979A1 (es) | Compuestos derivados ftalazina 1,4-disustituida; composicion farmaceutica; y su uso en el tratamiento del cancer. | |
| DOP2010000075A (es) | Compuesto inhibidor de glicógeno fosforilasa y composicion farmaceutica del mismo | |
| BR112014024220A2 (pt) | genes que codificam celulase | |
| CL2011000165A1 (es) | Compuestos derivados de indolinonas; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento y/o la prevencion del cancer, infecciones, enfermedades inflamatorias y autoinmunes. | |
| CL2007001748A1 (es) | Compuesto derivado de 2-arilamino-4-aminopirimidinas, inhibidores de la proteina quinasa c-alfa; composiciones farmaceuticas que los contienen; y su uso para tratar o prevenir la diabetes, el cancer, enfermedades cardiovasculares y otras. | |
| PE20142284A1 (es) | Procedimiento de fabricacion de una forma de dosificacion farmaceutica que comprende nifedipina y candesartan cilexetilo | |
| ECSP089024A (es) | Camsilato de (s)-(-)-amlodipino o hidrato del mismo y composición farmacéutica que comprende el mismo | |
| EA200701995A1 (ru) | Способы уменьшения кальцификации | |
| MX2009005400A (es) | Metodo para el diagnostico y tratamiento del glioma. |