ECSP099599A - Procedimientos para la preparación de compuestos de urea sustituidos con piperidinilo - Google Patents

Procedimientos para la preparación de compuestos de urea sustituidos con piperidinilo

Info

Publication number
ECSP099599A
ECSP099599A EC2009009599A ECSP099599A ECSP099599A EC SP099599 A ECSP099599 A EC SP099599A EC 2009009599 A EC2009009599 A EC 2009009599A EC SP099599 A ECSP099599 A EC SP099599A EC SP099599 A ECSP099599 A EC SP099599A
Authority
EC
Ecuador
Prior art keywords
piperidinyl
procedures
preparation
urea compounds
compounds replaced
Prior art date
Application number
EC2009009599A
Other languages
English (en)
Inventor
Richard D Gless Jr
Original Assignee
Arete Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arete Therapeutics Inc filed Critical Arete Therapeutics Inc
Publication of ECSP099599A publication Critical patent/ECSP099599A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/96Sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Se describen procedimientos para la síntesis de compuestos de urea sustituidos con piperidinilo. Esta invención también se refiere a intermediarios novedosos preparados durante esta síntesis.
EC2009009599A 2007-01-29 2009-08-27 Procedimientos para la preparación de compuestos de urea sustituidos con piperidinilo ECSP099599A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88711407P 2007-01-29 2007-01-29
US97217707P 2007-09-13 2007-09-13

Publications (1)

Publication Number Publication Date
ECSP099599A true ECSP099599A (es) 2009-09-29

Family

ID=39493517

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2009009599A ECSP099599A (es) 2007-01-29 2009-08-27 Procedimientos para la preparación de compuestos de urea sustituidos con piperidinilo

Country Status (15)

Country Link
US (1) US20080207908A1 (es)
EP (1) EP2125729A1 (es)
JP (1) JP2010516785A (es)
KR (1) KR20090107045A (es)
CN (1) CN101663273A (es)
AR (1) AR065079A1 (es)
AU (1) AU2008210723A1 (es)
BR (1) BRPI0807125A2 (es)
CA (1) CA2675448A1 (es)
EA (1) EA200901063A1 (es)
EC (1) ECSP099599A (es)
IL (1) IL199654A0 (es)
MX (1) MX2009008093A (es)
TW (1) TW200838851A (es)
WO (1) WO2008094862A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090197916A1 (en) * 2007-01-29 2009-08-06 Arete Therapeutics, Inc Soluble epoxide hydrolase inhibitors for treatment of metabolic syndrome and related disorders
CN115109841B (zh) * 2022-06-23 2025-11-04 苏州拉索生物芯片科技有限公司 一种芯片微球氨基封闭方法及应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9216298D0 (en) * 1991-08-15 1992-09-16 Ici Plc Piperidine derivatives
US7081454B2 (en) * 2001-03-28 2006-07-25 Bristol-Myers Squibb Co. Tyrosine kinase inhibitors
CA2533749C (en) * 2003-08-01 2012-07-10 Chugai Seiyaku Kabushiki Kaisha Piperidine compounds useful as malonyl-coa decarboxylase inhibitors
TW200808723A (en) * 2006-03-13 2008-02-16 Univ California Conformationally restricted urea inhibitors of soluble epoxide hydrolase

Also Published As

Publication number Publication date
WO2008094862A1 (en) 2008-08-07
CA2675448A1 (en) 2008-08-07
CN101663273A (zh) 2010-03-03
JP2010516785A (ja) 2010-05-20
MX2009008093A (es) 2009-08-12
TW200838851A (en) 2008-10-01
AR065079A1 (es) 2009-05-13
IL199654A0 (en) 2010-04-15
US20080207908A1 (en) 2008-08-28
BRPI0807125A2 (pt) 2014-04-08
EA200901063A1 (ru) 2009-12-30
KR20090107045A (ko) 2009-10-12
AU2008210723A1 (en) 2008-08-07
EP2125729A1 (en) 2009-12-02

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