ECSP12011800A - Composición farmacéutica para bajar de peso y procedimiento para obtener la misma - Google Patents
Composición farmacéutica para bajar de peso y procedimiento para obtener la mismaInfo
- Publication number
- ECSP12011800A ECSP12011800A ECSP12011800A ECSP12011800A EC SP12011800 A ECSP12011800 A EC SP12011800A EC SP12011800 A ECSP12011800 A EC SP12011800A EC SP12011800 A ECSP12011800 A EC SP12011800A
- Authority
- EC
- Ecuador
- Prior art keywords
- procedure
- pharmaceutical composition
- same
- lower weight
- orlistat
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- AHLBNYSZXLDEJQ-FWEHEUNISA-N orlistat Chemical compound CCCCCCCCCCC[C@H](OC(=O)[C@H](CC(C)C)NC=O)C[C@@H]1OC(=O)[C@H]1CCCCCC AHLBNYSZXLDEJQ-FWEHEUNISA-N 0.000 abstract 2
- 229960001243 orlistat Drugs 0.000 abstract 2
- PHIQHXFUZVPYII-ZCFIWIBFSA-N (R)-carnitine Chemical compound C[N+](C)(C)C[C@H](O)CC([O-])=O PHIQHXFUZVPYII-ZCFIWIBFSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- 230000004580 weight loss Effects 0.000 abstract 1
- 238000005550 wet granulation Methods 0.000 abstract 1
- 238000009736 wetting Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/205—Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Inorganic Chemistry (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Child & Adolescent Psychology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Plant Substances (AREA)
- Medicinal Preparation (AREA)
Abstract
Se describe una composición farmacéutica para bajar de peso que comprende una mezcla de Orlistat y L-Carnitina como ingredientes activos, y un vehículo farmacéuticamente aceptable. Asimismo, se describe un procedimiento para obtener dicha composición donde se realiza una humectación y granulación húmeda del Orlistat que evita que se presenten problemas de pegado o escasa fluidez de este compuesto.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2009009971A MX342962B (es) | 2009-09-18 | 2009-09-18 | Composicion farmaceutica para bajar de peso y procedimiento para obtener la misma. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP12011800A true ECSP12011800A (es) | 2012-05-30 |
Family
ID=43758159
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP12011800 ECSP12011800A (es) | 2009-09-18 | 2012-04-16 | Composición farmacéutica para bajar de peso y procedimiento para obtener la misma |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP2478902A4 (es) |
| AR (1) | AR078185A1 (es) |
| BR (1) | BR112012006013A2 (es) |
| CO (1) | CO6541522A2 (es) |
| EC (1) | ECSP12011800A (es) |
| GT (1) | GT201200079A (es) |
| MX (1) | MX342962B (es) |
| WO (1) | WO2011033356A1 (es) |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6004996A (en) | 1997-02-05 | 1999-12-21 | Hoffman-La Roche Inc. | Tetrahydrolipstatin containing compositions |
| IT1305308B1 (it) * | 1999-03-26 | 2001-05-04 | Biosint S P A | Granulato ad alto contenuto di l-carnitina o alcanoil-l-carnitina,particolarmente adatto alla produzione di compresse per compressione |
| WO2003009840A1 (en) * | 2001-07-24 | 2003-02-06 | Lonza Ag | Composition comprising at least one lipase inhibitor and carnitine |
| CN1546017A (zh) * | 2003-11-30 | 2004-11-17 | 杨喜鸿 | 奥利司他的复方制剂 |
| JP2006191830A (ja) * | 2005-01-12 | 2006-07-27 | Unitika Ltd | 脂肪の蓄積を抑制する食品 |
| TR200607613A2 (tr) * | 2006-12-29 | 2008-07-21 | NOBEL İLAÇ SAN.ve TiC.A.Ş. | Lipaz inhibitörü içeren farmasötik formülasyonlar |
| SI2002825T1 (sl) * | 2007-06-14 | 2013-10-30 | Krka | Farmacevtski sestavki, ki obsegajo orlistat |
| CN101224202A (zh) * | 2007-12-26 | 2008-07-23 | 广州康采恩医药有限公司 | 减肥组合物 |
-
2009
- 2009-09-18 MX MX2009009971A patent/MX342962B/es active IP Right Grant
-
2010
- 2010-09-13 WO PCT/IB2010/002270 patent/WO2011033356A1/es not_active Ceased
- 2010-09-13 BR BR112012006013A patent/BR112012006013A2/pt not_active Application Discontinuation
- 2010-09-13 EP EP10816760.2A patent/EP2478902A4/en not_active Withdrawn
- 2010-09-16 AR ARP100103388A patent/AR078185A1/es unknown
-
2012
- 2012-03-16 GT GT201200079A patent/GT201200079A/es unknown
- 2012-04-13 CO CO12060999A patent/CO6541522A2/es unknown
- 2012-04-16 EC ECSP12011800 patent/ECSP12011800A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GT201200079A (es) | 2014-01-27 |
| EP2478902A1 (en) | 2012-07-25 |
| AR078185A1 (es) | 2011-10-19 |
| MX342962B (es) | 2016-06-07 |
| WO2011033356A1 (es) | 2011-03-24 |
| BR112012006013A2 (pt) | 2016-06-14 |
| EP2478902A4 (en) | 2014-05-14 |
| CO6541522A2 (es) | 2012-10-16 |
| MX2009009971A (es) | 2011-03-18 |
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