ECSP14033496A - THIAZOLS SUBSTITUTED BY CARBOXAMIDE OR SULFONAMIDE AND RELATED DERIVATIVES AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTOR - Google Patents
THIAZOLS SUBSTITUTED BY CARBOXAMIDE OR SULFONAMIDE AND RELATED DERIVATIVES AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTORInfo
- Publication number
- ECSP14033496A ECSP14033496A ECIEPI201433496A ECPI201433496A ECSP14033496A EC SP14033496 A ECSP14033496 A EC SP14033496A EC IEPI201433496 A ECIEPI201433496 A EC IEPI201433496A EC PI201433496 A ECPI201433496 A EC PI201433496A EC SP14033496 A ECSP14033496 A EC SP14033496A
- Authority
- EC
- Ecuador
- Prior art keywords
- gamma
- ror
- modulators
- sulfonamide
- nuclear receptor
- Prior art date
Links
- 229940124530 sulfonamide Drugs 0.000 title abstract 2
- 150000003456 sulfonamides Chemical group 0.000 title abstract 2
- 150000003857 carboxamides Chemical group 0.000 title 1
- 102000004164 orphan nuclear receptors Human genes 0.000 title 1
- 108090000629 orphan nuclear receptors Proteins 0.000 title 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 cyclic carboxamide Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La invención provee moduladores para el receptor nuclear huérfano ROR[gamma] y métodos para tratar enfermedades mediadas por ROR[gamma] mediante la administración de estos moduladores novedosos de ROR[gamma] a un humano o mamífero que los necesite. Específicamente, la presente invención provee compuestos cíclicos que contienen carboxamida o sulfonamida de Fórmula (1), (1'), (100), (100'), (200) y (200'), y los enantiómeros, diastereómeros, tautómeros, N-óxidos, solvatos y sales farmacéuticamente aceptables de los mismos.The invention provides modulators for the orphan nuclear receptor ROR [gamma] and methods of treating ROR [gamma] mediated diseases by administering these novel modulators of ROR [gamma] to a human or mammal in need thereof. Specifically, the present invention provides cyclic carboxamide or sulfonamide-containing compounds of Formula (1), (1 '), (100), (100'), (200) and (200 '), and the enantiomers, diastereomers, tautomers, N-oxides, solvates and pharmaceutically acceptable salts thereof.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261653556P | 2012-05-31 | 2012-05-31 | |
| EP12004186 | 2012-05-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP14033496A true ECSP14033496A (en) | 2015-09-30 |
Family
ID=71943845
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECIEPI201433496A ECSP14033496A (en) | 2012-05-31 | 2014-12-30 | THIAZOLS SUBSTITUTED BY CARBOXAMIDE OR SULFONAMIDE AND RELATED DERIVATIVES AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTOR |
Country Status (2)
| Country | Link |
|---|---|
| EC (1) | ECSP14033496A (en) |
| PE (1) | PE20200480A1 (en) |
-
2013
- 2013-05-29 PE PE2020000002A patent/PE20200480A1/en unknown
-
2014
- 2014-12-30 EC ECIEPI201433496A patent/ECSP14033496A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PE20200480A1 (en) | 2020-03-03 |
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