ECSP15007708A - NITROGEN-CONTAINING 5-MEMBER HETEROCYCLES REPLACED BY CARBOXAMIDE OR SULPHONAMIDE AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTOR - Google Patents
NITROGEN-CONTAINING 5-MEMBER HETEROCYCLES REPLACED BY CARBOXAMIDE OR SULPHONAMIDE AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTORInfo
- Publication number
- ECSP15007708A ECSP15007708A ECIEPI20157708A ECPI201507708A ECSP15007708A EC SP15007708 A ECSP15007708 A EC SP15007708A EC IEPI20157708 A ECIEPI20157708 A EC IEPI20157708A EC PI201507708 A ECPI201507708 A EC PI201507708A EC SP15007708 A ECSP15007708 A EC SP15007708A
- Authority
- EC
- Ecuador
- Prior art keywords
- gamma
- ror
- modulators
- nuclear receptor
- carboxamide
- Prior art date
Links
- 150000003857 carboxamides Chemical class 0.000 title 1
- 102000004164 orphan nuclear receptors Human genes 0.000 title 1
- 108090000629 orphan nuclear receptors Proteins 0.000 title 1
- FDDDEECHVMSUSB-UHFFFAOYSA-N sulfanilamide Chemical compound NC1=CC=C(S(N)(=O)=O)C=C1 FDDDEECHVMSUSB-UHFFFAOYSA-N 0.000 title 1
- 229940124530 sulfonamide Drugs 0.000 title 1
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 cyclic carboxamide Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención provee moduladores para el receptor nuclear huérfano ROR[gamma] y métodos para tratar enfermedades mediadas por ROR[gamma] mediante la administración de estos nuevos moduladores de ROR[gamma] a un humano o mamífero que los necesita. Específicamente, la presente invención provee compuestos cíclicos que contienen carboxamida de Fórmula (1) a Fórmula (5) y los enantiómeros, diastereómeros, tautómeros, N-óxidos, solvatos y sales farmacéuticamente aceptables de los mismos.The invention provides modulators for the orphan nuclear receptor ROR [gamma] and methods for treating ROR [gamma] mediated diseases by administering these novel ROR [gamma] modulators to a human or mammal in need thereof. Specifically, the present invention provides cyclic carboxamide-containing compounds of Formula (1) to Formula (5) and the enantiomers, diastereomers, tautomers, N-oxides, solvates, and pharmaceutically acceptable salts thereof.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261681296P | 2012-08-09 | 2012-08-09 | |
| EP12005789 | 2012-08-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP15007708A true ECSP15007708A (en) | 2015-12-31 |
Family
ID=70289070
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECIEPI20157708A ECSP15007708A (en) | 2012-08-09 | 2015-03-02 | NITROGEN-CONTAINING 5-MEMBER HETEROCYCLES REPLACED BY CARBOXAMIDE OR SULPHONAMIDE AS MODULATORS FOR THE ROR [GAMMA] ORPHAN NUCLEAR RECEPTOR |
Country Status (2)
| Country | Link |
|---|---|
| EC (1) | ECSP15007708A (en) |
| NI (1) | NI201500016A (en) |
-
2015
- 2015-02-06 NI NI201500016A patent/NI201500016A/en unknown
- 2015-03-02 EC ECIEPI20157708A patent/ECSP15007708A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NI201500016A (en) | 2015-09-21 |
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