ECSP22031078A - Usos del complejo de metabolito antagonista del receptor de angiotensina ii e inhibidor de nep en el tratamiento de la insuficiencia card?aca - Google Patents
Usos del complejo de metabolito antagonista del receptor de angiotensina ii e inhibidor de nep en el tratamiento de la insuficiencia card?acaInfo
- Publication number
- ECSP22031078A ECSP22031078A ECSENADI202231078A ECDI202231078A ECSP22031078A EC SP22031078 A ECSP22031078 A EC SP22031078A EC SENADI202231078 A ECSENADI202231078 A EC SENADI202231078A EC DI202231078 A ECDI202231078 A EC DI202231078A EC SP22031078 A ECSP22031078 A EC SP22031078A
- Authority
- EC
- Ecuador
- Prior art keywords
- heart failure
- angiotensin
- receptor antagonist
- treatment
- nep inhibitor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
Los usos de un complejo de un metabolito antagonista del receptor de angiotensina II y un inhibidor de NEP para la insuficiencia card?aca, se relacionan espec?ficamente los usos del complejo en la preparaci?n de un medicamento para su uso en la insuficiencia card?aca con fracci?n de expulsi?n reducida (HFrEF).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201910890853 | 2019-09-20 | ||
| CN202010901984 | 2020-09-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP22031078A true ECSP22031078A (es) | 2022-08-31 |
Family
ID=74883393
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSENADI202231078A ECSP22031078A (es) | 2019-09-20 | 2022-04-19 | Usos del complejo de metabolito antagonista del receptor de angiotensina ii e inhibidor de nep en el tratamiento de la insuficiencia card?aca |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US12508246B2 (es) |
| EP (1) | EP4032532B1 (es) |
| JP (1) | JP7316449B2 (es) |
| KR (1) | KR102752382B1 (es) |
| CN (2) | CN115487175B (es) |
| AU (1) | AU2020348813B2 (es) |
| CA (1) | CA3151788A1 (es) |
| CO (1) | CO2022004910A2 (es) |
| EC (1) | ECSP22031078A (es) |
| MX (1) | MX2022003408A (es) |
| TW (1) | TWI809313B (es) |
| WO (1) | WO2021052441A1 (es) |
| ZA (1) | ZA202204370B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021052441A1 (zh) | 2019-09-20 | 2021-03-25 | 深圳信立泰药业股份有限公司 | 血管紧张素ii受体拮抗剂代谢产物与nep抑制剂的复合物治疗心衰的用途 |
| TWI894333B (zh) * | 2020-08-17 | 2025-08-21 | 大陸商深圳信立泰藥業股份有限公司 | 血管收縮素ii受體拮抗劑代謝產物與nep抑制劑的複合物用於心臟衰竭的應用 |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2004203284A1 (en) * | 1998-11-06 | 2004-08-12 | G.D. Searle & Co. | Combination therapy of angiotensin converting enzyme inhibitor and aldosterone antagonist for reducing morbidity and mortality from cardiovascular disease |
| GB0211230D0 (en) * | 2002-05-16 | 2002-06-26 | Medinnova Sf | Treatment of heart failure |
| US20060014828A1 (en) * | 2004-07-16 | 2006-01-19 | Nitromed, Inc. | Compositions and methods related to heart failure |
| AR057882A1 (es) | 2005-11-09 | 2007-12-26 | Novartis Ag | Compuestos de accion doble de bloqueadores del receptor de angiotensina e inhibidores de endopeptidasa neutra |
| WO2010113993A1 (ja) | 2009-04-01 | 2010-10-07 | 三井化学株式会社 | オレフィンの製造方法 |
| AR089954A1 (es) | 2012-02-15 | 2014-10-01 | Theravance Inc | Forma cristalina del ester 5-metil-2-oxo-[1,3]dioxol-4-ilmetilico del acido (2s,4r)-5-bifenil-4-il-2-hidroximetil-2-metil-4-[(1h-[1,2,3]triazol-4-carbonil)amino]pentanoico |
| DK3626270T3 (da) | 2013-08-26 | 2024-01-15 | Novartis Ag | Behandling af kardiovaskulære sygdomme |
| CN105503760A (zh) * | 2014-10-10 | 2016-04-20 | 上海翰森生物医药科技有限公司 | 结晶型ARB-NEPi双阳离子复合物及其制备方法和应用 |
| CN106138041A (zh) * | 2015-04-15 | 2016-11-23 | 苏州朗科生物技术有限公司 | 一种双重作用的氯沙坦复合物 |
| CN106146472A (zh) * | 2015-04-15 | 2016-11-23 | 苏州朗科生物技术有限公司 | 一种双重作用的阿利沙坦复合物 |
| PL4212152T3 (pl) * | 2015-05-11 | 2025-08-11 | Novartis Ag | Schemat dawkowania sakubitrylu-walsartanu do leczenia przewlekłej skurczowej niewydolności serca |
| WO2017006254A1 (en) | 2015-07-08 | 2017-01-12 | Novartis Ag | Drug combination comprising an angiotensin ii receptor antagonist, a neutral endopeptidase inhibitor and a mineralcorticoid receptor antagonist |
| CN105669581B (zh) | 2015-11-09 | 2017-03-22 | 成都苑东生物制药股份有限公司 | 一种血管紧张受体拮抗剂和中性内肽酶抑制剂复合物 |
| WO2017125031A1 (zh) * | 2016-01-20 | 2017-07-27 | 深圳信立泰药业股份有限公司 | 血管紧张素ii受体拮抗剂代谢产物与nep抑制剂的复合物及其制备方法 |
| TWI731943B (zh) | 2016-03-08 | 2021-07-01 | 美商施萬生物製藥研發Ip有限責任公司 | 結晶型(2s,4r)-5-(5’-氯-2’-氟-[1,1’-聯苯]-4-基)-2-(乙氧基甲基)-4-(3-羥基異㗁唑-5-甲醯胺基)-2-甲基戊酸及其用途 |
| CN106177960B (zh) * | 2016-08-01 | 2019-01-08 | 珠海赛隆药业股份有限公司(长沙)医药研发中心 | 血管紧张素受体拮抗剂和脑啡肽酶抑制剂的复合物及其用途 |
| CN106924241A (zh) * | 2017-04-28 | 2017-07-07 | 广州医科大学 | 川陈皮素在预防或治疗心衰药物中的应用 |
| SG11202112723PA (en) | 2019-05-19 | 2021-12-30 | Myokardia Inc | Treatment of systolic dysfunction and heart failure with reduced ejection fraction with the compound(r)-4-(1-((3-(difluoromethyl)-1-methyl-1h-pyrazol-4-yl)sulfonyl)-1-fluoroethyl)-n-(isoxazol-3-yl)piperidine-1-carboxamide |
| WO2020238885A1 (zh) | 2019-05-30 | 2020-12-03 | 深圳信立泰药业股份有限公司 | 血管紧张素ii受体拮抗剂代谢产物与nep抑制剂的复合物的治疗方法 |
| WO2021052441A1 (zh) * | 2019-09-20 | 2021-03-25 | 深圳信立泰药业股份有限公司 | 血管紧张素ii受体拮抗剂代谢产物与nep抑制剂的复合物治疗心衰的用途 |
| TWI894333B (zh) | 2020-08-17 | 2025-08-21 | 大陸商深圳信立泰藥業股份有限公司 | 血管收縮素ii受體拮抗劑代謝產物與nep抑制劑的複合物用於心臟衰竭的應用 |
-
2020
- 2020-09-18 WO PCT/CN2020/116023 patent/WO2021052441A1/zh not_active Ceased
- 2020-09-18 CN CN202211186846.XA patent/CN115487175B/zh active Active
- 2020-09-18 EP EP20866108.2A patent/EP4032532B1/en active Active
- 2020-09-18 AU AU2020348813A patent/AU2020348813B2/en active Active
- 2020-09-18 KR KR1020217042035A patent/KR102752382B1/ko active Active
- 2020-09-18 CA CA3151788A patent/CA3151788A1/en active Pending
- 2020-09-18 TW TW109132385A patent/TWI809313B/zh active
- 2020-09-18 CN CN202080008624.1A patent/CN113286585B/zh active Active
- 2020-09-18 US US17/761,543 patent/US12508246B2/en active Active
- 2020-09-18 MX MX2022003408A patent/MX2022003408A/es unknown
- 2020-09-18 JP JP2022513095A patent/JP7316449B2/ja active Active
-
2022
- 2022-04-19 CO CONC2022/0004910A patent/CO2022004910A2/es unknown
- 2022-04-19 EC ECSENADI202231078A patent/ECSP22031078A/es unknown
- 2022-04-19 ZA ZA2022/04370A patent/ZA202204370B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20220395491A1 (en) | 2022-12-15 |
| AU2020348813A1 (en) | 2022-04-14 |
| KR20220012317A (ko) | 2022-02-03 |
| CA3151788A1 (en) | 2021-03-25 |
| EP4032532A1 (en) | 2022-07-27 |
| TW202114652A (zh) | 2021-04-16 |
| CO2022004910A2 (es) | 2022-05-31 |
| TWI809313B (zh) | 2023-07-21 |
| CN115487175A (zh) | 2022-12-20 |
| CN113286585A (zh) | 2021-08-20 |
| JP2022545904A (ja) | 2022-11-01 |
| KR102752382B1 (ko) | 2025-01-09 |
| AU2020348813B2 (en) | 2025-09-11 |
| MX2022003408A (es) | 2022-07-12 |
| CN115487175B (zh) | 2024-05-14 |
| ZA202204370B (en) | 2022-11-30 |
| EP4032532A4 (en) | 2023-10-04 |
| WO2021052441A1 (zh) | 2021-03-25 |
| JP7316449B2 (ja) | 2023-07-27 |
| EP4032532B1 (en) | 2026-08-12 |
| US12508246B2 (en) | 2025-12-30 |
| CN113286585B (zh) | 2022-11-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CO2023011071A2 (es) | Agonistas del receptor gpcr, composiciones farmacéuticas que los comprenden y métodos para su uso | |
| MX2020013624A (es) | Agonistas del receptor glp-1 y usos de los mismos. | |
| CL2019001465A1 (es) | Nuevos compuestos como agonistas peptídicos trigonales de los receptores de glp1/glucagón/gip. | |
| CL2020003174S1 (es) | Dispositivo para administración de dosis. | |
| MX2020004467A (es) | Metodos para el tratamiento o la prevencion del asma mediante la administracion de antagonista de il-4r. | |
| CL2019002470A1 (es) | Combinaciones de un derivado de 4-pirimidinsulfamida con ingredientes activos para el tratamiento de enfermedades relacionadas con endotelina. | |
| CL2017003351A1 (es) | Anticuerpo anti receptor de transferrina humana que pasan a través de la barrera hematoencefálica. | |
| DOP2018000297A (es) | Derivado de glucagon, conjugado del mismo, composición que comprende el mismo y uso terapéutico del mismo | |
| CL2008003222A1 (es) | Peptidos con actividad antagonista de glucagon y composicion farmaceutica que los comprende, utiles para el tratamiento de la hiperglicemia, para suprimir el apetito, reducir el aumento de peso y para tratar el desgaste catabolico. | |
| MX2019003780A (es) | Uso de la combinación de anticuerpo anti-pd-1 e inhibidor de vegfr en la preparación de medicamentos para el tratamiento de cánceres. | |
| CL2019000245A1 (es) | Moduladores nmda espiro-lactam y métodos de uso de los mismos. | |
| CO2017002160A2 (es) | Derivados de pirimidina sustituidos con heterociclilo opcionalmente condensados útiles para el tratamiento de enfermedades inflamatorias, metabólicas, oncológicas y autoinmunitarias | |
| AR111360A1 (es) | Tratamiento usando células t de receptor quimérico incorporando células t polifuncionales optimizadas | |
| MX2016010998A (es) | Terapia celular adoptiva que usa un agonista de receptor huérfano gamma relacionado con receptor de ácido retinoico y métodos terapéuticos relacionados. | |
| CO2021015793A2 (es) | Métodos para tratar o prevenir el asma mediante la administración un antagonista de il-33 | |
| CL2022001692A1 (es) | Compuestos activos frente a receptores nucleares | |
| CO2017008031A2 (es) | Compuestos con actividad antagonista de los receptores muscarínicos y actividad agonista del receptor beta2 adrenérgico | |
| MX2021008268A (es) | Tratamiento de cefalea por uso excesivo de medicamentos usando anticuerpos anti-cgrp o anti-cgrp-r. | |
| PE20211196A1 (es) | Metodos para tratar inflamacion mediada por il-6 sin inmunosupresion | |
| CL2018003045A1 (es) | Semaglutida en afecciones cardiovasculares. | |
| ECSP19062381A (es) | Moduladores del receptor de estrógeno | |
| CO7461127A2 (es) | Código para la configuración de un dispositivo de atención al paciente | |
| CO2022004910A2 (es) | Un complejo de metabolito antagonista del receptor de angiotensina ii e inhibidor de nep en el tratamiento de la insuficiencia cardíaca | |
| MX376160B (es) | Compuestos que tienen actividad antagonista del receptor muscarínico y actividad agonista del receptor beta2 adrenérgico. | |
| CR20120617A (es) | Combinación de inhibidores de xantna oxidasa y antagonistas del receptor de angiotensina ii y su uso |