ECSP982481A - Inhibidores de proteasas - Google Patents
Inhibidores de proteasasInfo
- Publication number
- ECSP982481A ECSP982481A ECSP982481A ECSP982481A EC SP982481 A ECSP982481 A EC SP982481A EC SP982481 A ECSP982481 A EC SP982481A EC SP982481 A ECSP982481 A EC SP982481A
- Authority
- EC
- Ecuador
- Prior art keywords
- disease
- cartilage
- excessive
- degeneration
- present
- Prior art date
Links
- 229940042399 direct acting antivirals protease inhibitors Drugs 0.000 title 1
- 239000000137 peptide hydrolase inhibitor Substances 0.000 title 1
- 210000000845 cartilage Anatomy 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 201000010099 disease Diseases 0.000 abstract 3
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 3
- 206010065687 Bone loss Diseases 0.000 abstract 2
- 230000007850 degeneration Effects 0.000 abstract 2
- 239000011159 matrix material Substances 0.000 abstract 2
- 102000004171 Cathepsin K Human genes 0.000 abstract 1
- 108090000625 Cathepsin K Proteins 0.000 abstract 1
- 208000037147 Hypercalcaemia Diseases 0.000 abstract 1
- 208000030136 Marchiafava-Bignami Disease Diseases 0.000 abstract 1
- 208000029725 Metabolic bone disease Diseases 0.000 abstract 1
- 208000010191 Osteitis Deformans Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 208000027868 Paget disease Diseases 0.000 abstract 1
- 102000035195 Peptidases Human genes 0.000 abstract 1
- 108091005804 Peptidases Proteins 0.000 abstract 1
- 239000004365 Protease Substances 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- 230000015556 catabolic process Effects 0.000 abstract 1
- 238000006731 degradation reaction Methods 0.000 abstract 1
- 208000007565 gingivitis Diseases 0.000 abstract 1
- 230000000148 hypercalcaemia Effects 0.000 abstract 1
- 208000030915 hypercalcemia disease Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000003211 malignant effect Effects 0.000 abstract 1
- 208000027202 mammary Paget disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 1
- 201000001245 periodontitis Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona compuestos que inhiben proteasas, incluyendo catepsina K, composiciones farmacéuticas de tales compuestos, y métodos para tratar enfermedades de excesiva pérdida ósea o degeneración de cartílago o degradación de cartílago o matriz, incluyendo osteoporosis; enfermedad gigival, incluyendo gingivitis y periodontitis; artritis, más especificamente, osteoartritis y artritis reumatoide; enfermedad de Paget; hipercalcemia de enfermedades malignas; y enfermedad ósea metabólica, que comprende inhibir dicha pérdida ósea o degeneración excesiva de cartílago o matriz administrando un compuesto de la presente invención a un paciente con necesidad de ello.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982481 ECSP982481A (es) | 1998-04-22 | 1998-04-22 | Inhibidores de proteasas |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982481 ECSP982481A (es) | 1998-04-22 | 1998-04-22 | Inhibidores de proteasas |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP982481A true ECSP982481A (es) | 1999-01-19 |
Family
ID=42043403
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP982481 ECSP982481A (es) | 1998-04-22 | 1998-04-22 | Inhibidores de proteasas |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP982481A (es) |
-
1998
- 1998-04-22 EC ECSP982481 patent/ECSP982481A/es unknown
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