ECSP992959A - Inhibidores de proteasa de bis- aminometil carbonilo - Google Patents
Inhibidores de proteasa de bis- aminometil carboniloInfo
- Publication number
- ECSP992959A ECSP992959A ECSP992959A ECSP992959A EC SP992959 A ECSP992959 A EC SP992959A EC SP992959 A ECSP992959 A EC SP992959A EC SP992959 A ECSP992959 A EC SP992959A
- Authority
- EC
- Ecuador
- Prior art keywords
- diseases
- protease inhibitors
- bis
- aminometil
- cartilage
- Prior art date
Links
- 229940042399 direct acting antivirals protease inhibitors Drugs 0.000 title abstract 2
- 239000000137 peptide hydrolase inhibitor Substances 0.000 title abstract 2
- UGFAIRIUMAVXCW-UHFFFAOYSA-N Carbon monoxide Chemical class [O+]#[C-] UGFAIRIUMAVXCW-UHFFFAOYSA-N 0.000 title 1
- 206010065687 Bone loss Diseases 0.000 abstract 2
- 210000000845 cartilage Anatomy 0.000 abstract 2
- 230000015556 catabolic process Effects 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 238000006731 degradation reaction Methods 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 239000011159 matrix material Substances 0.000 abstract 2
- RSBQFKJVGZVGFM-UHFFFAOYSA-N 1,3-diaminopropan-2-one Chemical group NCC(=O)CN RSBQFKJVGZVGFM-UHFFFAOYSA-N 0.000 abstract 1
- 208000037147 Hypercalcaemia Diseases 0.000 abstract 1
- 208000029725 Metabolic bone disease Diseases 0.000 abstract 1
- 208000010191 Osteitis Deformans Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 208000027868 Paget disease Diseases 0.000 abstract 1
- 102000035195 Peptidases Human genes 0.000 abstract 1
- 108091005804 Peptidases Proteins 0.000 abstract 1
- 239000004365 Protease Substances 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- -1 captesin K Substances 0.000 abstract 1
- 208000024693 gingival disease Diseases 0.000 abstract 1
- 208000007565 gingivitis Diseases 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 230000000148 hypercalcaemia Effects 0.000 abstract 1
- 208000030915 hypercalcemia disease Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000003211 malignant effect Effects 0.000 abstract 1
- 208000027202 mammary Paget disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 1
- 201000001245 periodontitis Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona inhibidores de proteasa de bis-aminometil-carbonilo y sales, hidratos o solvatos de los mismos aceptables farmacéuticamente, que inhiben proteasas, incluyendo la captesina K, composiciones farmacéuticas de tales compuestos, y métodos para tratar enfermedades de una excesiva pérdida ósea o degradación de cartilago o de matriz, incluyendo osteoporosis; enfermedades gingivales incluyendo gingivitis y periodontitis; artritis más especificamente osteoartritis y artritis reumatoide; enfermedad de paget; hipercalcemia de enfermedades malignas; y enfermedades óseas metabólicas, que comprende inhibir dicha pérdida de hueso o dicha excesiva degradación de cartilago o de matriz administrando a un paciente que lo necesite un compuesto según la presente invención.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992959 ECSP992959A (es) | 1999-05-20 | 1999-05-20 | Inhibidores de proteasa de bis- aminometil carbonilo |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992959 ECSP992959A (es) | 1999-05-20 | 1999-05-20 | Inhibidores de proteasa de bis- aminometil carbonilo |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992959A true ECSP992959A (es) | 1999-10-06 |
Family
ID=42043948
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992959 ECSP992959A (es) | 1999-05-20 | 1999-05-20 | Inhibidores de proteasa de bis- aminometil carbonilo |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992959A (es) |
-
1999
- 1999-05-20 EC ECSP992959 patent/ECSP992959A/es unknown
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