ECSP982530A - NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA - Google Patents

NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA

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Publication number
ECSP982530A
ECSP982530A ECSP982530A ECSP982530A EC SP982530 A ECSP982530 A EC SP982530A EC SP982530 A ECSP982530 A EC SP982530A EC SP982530 A ECSP982530 A EC SP982530A
Authority
EC
Ecuador
Prior art keywords
novel sulfonamide
protein
transferasa
farnesil
sulfonamide inhibitors
Prior art date
Application number
Other languages
Spanish (es)
Inventor
F George Njoroge
Ronald J Doll
Viyyoor Moopil Girijavallabhan
Bancha Vibulbhan
Arthur G Taveras
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP982530 priority Critical patent/ECSP982530A/en
Publication of ECSP982530A publication Critical patent/ECSP982530A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se describen novedosos compuestos de sulfonamida y composiciones farmacéuticas que son inhibidores de la enzina proteína transferasa. También se describe un método para inhibir la función Ras y, por lo tanto, para inhibir el desarrollo anormal de las células. El método consiste en administrar el novedoso compuesto de sulfonamida a un sistema biológico. Específicamente, el método inhibe el desarrollo anormal de las células en mamíferos tales como seres humanos.Novel sulfonamide compounds and pharmaceutical compositions that are inhibitors of the protein transferase enzyme are described. Also described is a method of inhibiting Ras function and, therefore, of inhibiting abnormal cell development. The method is to administer the novel sulfonamide compound to a biological system. Specifically, the method inhibits abnormal cell development in mammals such as humans.

ECSP982530 1998-06-15 1998-06-15 NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA ECSP982530A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP982530 ECSP982530A (en) 1998-06-15 1998-06-15 NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP982530 ECSP982530A (en) 1998-06-15 1998-06-15 NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA

Publications (1)

Publication Number Publication Date
ECSP982530A true ECSP982530A (en) 1999-04-13

Family

ID=42043450

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP982530 ECSP982530A (en) 1998-06-15 1998-06-15 NOVEL SULFONAMIDE INHIBITORS FROM FARNESIL - PROTEIN TRANSFERASA

Country Status (1)

Country Link
EC (1) ECSP982530A (en)

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