ECSP993134A - 1,2,3,4- TETRAHIDROQUINOLINAS -2-SUBSTITUTED 4- CARBOXIAMINO SUBSTITUTED - Google Patents
1,2,3,4- TETRAHIDROQUINOLINAS -2-SUBSTITUTED 4- CARBOXIAMINO SUBSTITUTEDInfo
- Publication number
- ECSP993134A ECSP993134A ECSP993134A ECSP993134A EC SP993134 A ECSP993134 A EC SP993134A EC SP993134 A ECSP993134 A EC SP993134A EC SP993134 A ECSP993134 A EC SP993134A
- Authority
- EC
- Ecuador
- Prior art keywords
- substituted
- inhibitors
- levels
- cholesterol
- triglycerides
- Prior art date
Links
- 238000008214 LDL Cholesterol Methods 0.000 abstract 2
- HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 abstract 2
- 239000003112 inhibitor Substances 0.000 abstract 2
- 150000002632 lipids Chemical class 0.000 abstract 2
- 150000003626 triacylglycerols Chemical class 0.000 abstract 2
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 108010023302 HDL Cholesterol Proteins 0.000 abstract 1
- 108010010234 HDL Lipoproteins Proteins 0.000 abstract 1
- 102000015779 HDL Lipoproteins Human genes 0.000 abstract 1
- 241000282414 Homo sapiens Species 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 235000012000 cholesterol Nutrition 0.000 abstract 1
- 239000003354 cholesterol ester transfer protein inhibitor Substances 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Inhibidores de la proteína de transferencia de colesteril éster, composiciones farmacéuticas que contienen tales inhibidores y el uso de tales inhibidores para elevar ciertos niveles de lípidos en plasma, incluyendo colesterol de lipoproteínas de alta densidad, y para reducir ciertos otros niveles de lípidos en plasma, tales como el colesterol LDL y los triglicéridos y, por consiguiente, para tratar enfermedades que se excerban por los bajos niveles de colesterol HDL y/o altos niveles de colesterol LDL y triglicéridos, tales como la aterosclerósis y enfermedades cardiovasculares en algunos mamíferos, incluyendo los seres humanos.Cholesteryl ester transfer protein inhibitors, pharmaceutical compositions containing such inhibitors, and the use of such inhibitors to raise certain plasma lipid levels, including high-density lipoprotein cholesterol, and to reduce certain other plasma lipid levels, such as LDL cholesterol and triglycerides and, consequently, to treat diseases that are exacerbated by low levels of HDL cholesterol and / or high levels of LDL cholesterol and triglycerides, such as atherosclerosis and cardiovascular diseases in some mammals, including human beings.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993134 ECSP993134A (en) | 1999-09-10 | 1999-09-10 | 1,2,3,4- TETRAHIDROQUINOLINAS -2-SUBSTITUTED 4- CARBOXIAMINO SUBSTITUTED |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993134 ECSP993134A (en) | 1999-09-10 | 1999-09-10 | 1,2,3,4- TETRAHIDROQUINOLINAS -2-SUBSTITUTED 4- CARBOXIAMINO SUBSTITUTED |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP993134A true ECSP993134A (en) | 1999-10-29 |
Family
ID=42044122
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP993134 ECSP993134A (en) | 1999-09-10 | 1999-09-10 | 1,2,3,4- TETRAHIDROQUINOLINAS -2-SUBSTITUTED 4- CARBOXIAMINO SUBSTITUTED |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP993134A (en) |
-
1999
- 1999-09-10 EC ECSP993134 patent/ECSP993134A/en unknown
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