EE03383B1 - Kolesterooli biosünteesi inhibiitori ja kolesterooli absorptsiooni ß-laktaaminhibiitori kombinatsioon - Google Patents

Kolesterooli biosünteesi inhibiitori ja kolesterooli absorptsiooni ß-laktaaminhibiitori kombinatsioon

Info

Publication number
EE03383B1
EE03383B1 EE9400341A EE9400341A EE03383B1 EE 03383 B1 EE03383 B1 EE 03383B1 EE 9400341 A EE9400341 A EE 9400341A EE 9400341 A EE9400341 A EE 9400341A EE 03383 B1 EE03383 B1 EE 03383B1
Authority
EE
Estonia
Prior art keywords
inhibitor
cholesterol
pct
combination
lactam
Prior art date
Application number
EE9400341A
Other languages
English (en)
Estonian (et)
Other versions
EE9400341A (et
Inventor
R. Davis Harry
Original Assignee
Schering Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corporation filed Critical Schering Corporation
Publication of EE9400341A publication Critical patent/EE9400341A/xx
Publication of EE03383B1 publication Critical patent/EE03383B1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EE9400341A 1992-12-23 1994-11-23 Kolesterooli biosünteesi inhibiitori ja kolesterooli absorptsiooni ß-laktaaminhibiitori kombinatsioon EE03383B1 (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US99548892A 1992-12-23 1992-12-23

Publications (2)

Publication Number Publication Date
EE9400341A EE9400341A (et) 1996-04-15
EE03383B1 true EE03383B1 (et) 2001-04-16

Family

ID=25541876

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400341A EE03383B1 (et) 1992-12-23 1994-11-23 Kolesterooli biosünteesi inhibiitori ja kolesterooli absorptsiooni ß-laktaaminhibiitori kombinatsioon

Country Status (32)

Country Link
US (1) US5661145A (de)
EP (1) EP0675714B1 (de)
JP (1) JP3992728B2 (de)
KR (1) KR100306936B1 (de)
CN (1) CN1090479C (de)
AT (1) ATE175872T1 (de)
AU (1) AU680864B2 (de)
CA (1) CA2152351C (de)
CZ (1) CZ287125B6 (de)
DE (1) DE69323213T2 (de)
DK (1) DK0675714T3 (de)
EE (1) EE03383B1 (de)
ES (1) ES2128552T3 (de)
FI (1) FI952916A7 (de)
GR (1) GR3029405T3 (de)
HR (1) HRP931515B1 (de)
HU (1) HU221724B1 (de)
IL (1) IL108112A (de)
LT (1) LT3300B (de)
LV (1) LV10919B (de)
MX (1) MX9308053A (de)
MY (1) MY109538A (de)
NO (1) NO311325B1 (de)
NZ (1) NZ259790A (de)
PL (1) PL174128B1 (de)
SG (1) SG45147A1 (de)
SI (1) SI9300677A (de)
SK (1) SK281173B6 (de)
TW (1) TW319698B (de)
WO (1) WO1994014433A1 (de)
YU (1) YU49060B (de)
ZA (1) ZA939552B (de)

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US5633246A (en) * 1994-11-18 1997-05-27 Schering Corporation Sulfur-substituted azetidinone compounds useful as hypocholesterolemic agents
US5656624A (en) * 1994-12-21 1997-08-12 Schering Corporation 4-[(heterocycloalkyl or heteroaromatic)-substituted phenyl]-2-azetidinones useful as hypolipidemic agents
CZ127198A3 (cs) 1995-11-02 1998-12-16 Warner-Lambert Company Způsob regulace koncentrace lipidů a farmaceutická kompozice pro tento způsob
US20030153541A1 (en) * 1997-10-31 2003-08-14 Robert Dudley Novel anticholesterol compositions and method for using same
SI20109A (sl) * 1998-12-16 2000-06-30 LEK, tovarna farmacevtskih in kemi�nih izdelkov, d.d. Stabilna farmacevtska formulacija
AU4343500A (en) 1999-04-16 2000-11-02 Schering Corporation Use of azetidinone compounds
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US6979462B1 (en) * 2000-10-03 2005-12-27 Mutual Pharmaceutical Co., Inc. Stabilization of solid drug formulations
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US7071181B2 (en) 2001-01-26 2006-07-04 Schering Corporation Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
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Also Published As

Publication number Publication date
HU9501854D0 (en) 1995-08-28
PL309636A1 (en) 1995-10-30
NZ259790A (en) 1997-02-24
US5661145A (en) 1997-08-26
NO311325B1 (no) 2001-11-19
PL174128B1 (pl) 1998-06-30
HRP931515A2 (en) 1996-12-31
LTIP1514A (en) 1994-10-25
CA2152351A1 (en) 1994-07-07
MY109538A (en) 1997-02-28
NO952529L (no) 1995-06-23
EP0675714B1 (de) 1999-01-20
EP0675714A1 (de) 1995-10-11
DK0675714T3 (da) 1999-09-13
KR100306936B1 (ko) 2001-11-30
ES2128552T3 (es) 1999-05-16
LT3300B (en) 1995-06-26
SK78395A3 (en) 1996-05-08
SK281173B6 (sk) 2000-12-11
DE69323213D1 (de) 1999-03-04
HUT72081A (en) 1996-03-28
CN1090479C (zh) 2002-09-11
LV10919A (lv) 1995-12-20
MX9308053A (es) 1994-06-30
CZ287125B6 (en) 2000-09-13
HU221724B1 (hu) 2002-12-28
SG45147A1 (en) 1998-01-16
CA2152351C (en) 2009-09-22
CN1095591A (zh) 1994-11-30
FI952916L (fi) 1995-06-14
GR3029405T3 (en) 1999-05-28
FI952916A0 (fi) 1995-06-14
ZA939552B (en) 1994-10-12
ATE175872T1 (de) 1999-02-15
SI9300677A (en) 1994-09-30
AU5872094A (en) 1994-07-19
AU680864B2 (en) 1997-08-14
YU80293A (sh) 1997-12-05
LV10919B (en) 1996-04-20
NO952529D0 (no) 1995-06-23
FI952916A7 (fi) 1995-06-14
YU49060B (sh) 2003-08-29
EE9400341A (et) 1996-04-15
JP3992728B2 (ja) 2007-10-17
TW319698B (de) 1997-11-11
CZ164395A3 (en) 1996-03-13
WO1994014433A1 (en) 1994-07-07
IL108112A (en) 1999-11-30
JPH08505141A (ja) 1996-06-04
HRP931515B1 (en) 2000-02-29
IL108112A0 (en) 1994-04-12
DE69323213T2 (de) 1999-07-08

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