EE200200461A - Pteridiiniühendid psoriaasi raviks - Google Patents

Pteridiiniühendid psoriaasi raviks

Info

Publication number: EE200200461A
Authority: EE; Estonia
Prior art keywords: psoriasis; treatment; pteridine compounds; pteridine; compounds
Prior art date: 2000-02-23

Application number

EEP200200461A

Other languages

English (en)

Inventor

Bonnert Roger

Gardiner Stewart

Hunt Fraser

Walters Iain

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-02-23

Filing date

2001-02-20

Publication date

2003-12-15

2001-02-20 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2003-12-15 Publication of EE200200461A publication Critical patent/EE200200461A/et

Links

201000004681 Psoriasis Diseases 0.000 title 1
125000001042 pteridinyl group Chemical class N1=C(N=CC2=NC=CN=C12)* 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Immunology (AREA)
Pain & Pain Management (AREA)
Pulmonology (AREA)
Psychiatry (AREA)
Dermatology (AREA)
Rheumatology (AREA)
Addiction (AREA)
Diabetes (AREA)
Orthopedic Medicine & Surgery (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Cardiology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Hematology (AREA)
Physical Education & Sports Medicine (AREA)
Heart & Thoracic Surgery (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Medicinal Preparation (AREA)

EEP200200461A 2000-02-23 2001-02-20 Pteridiiniühendid psoriaasi raviks EE200200461A (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0004128A GB2359551A (en)	2000-02-23	2000-02-23	Pharmaceutically active pyrimidine derivatives
PCT/SE2001/000374 WO2001062758A1 (en)	2000-02-23	2001-02-20	Pteridine compounds for the treatment of psoriasis

Publications (1)

Publication Number	Publication Date
EE200200461A true EE200200461A (et)	2003-12-15

Family

ID=9886153

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200200461A EE200200461A (et)	2000-02-23	2001-02-20	Pteridiiniühendid psoriaasi raviks

Country Status (32)

Country	Link
US (2)	US6875868B2 (et)
EP (1)	EP1259512B1 (et)
JP (1)	JP2003524012A (et)
KR (1)	KR100795758B1 (et)
CN (1)	CN1190437C (et)
AR (1)	AR029805A1 (et)
AT (1)	ATE250605T1 (et)
AU (1)	AU782509B2 (et)
BG (1)	BG107002A (et)
BR (1)	BR0108600A (et)
CA (1)	CA2400217C (et)
CO (1)	CO5290258A1 (et)
CZ (1)	CZ20022839A3 (et)
DE (1)	DE60100851T2 (et)
DK (1)	DK1259512T3 (et)
EE (1)	EE200200461A (et)
ES (1)	ES2206402T3 (et)
GB (1)	GB2359551A (et)
HU (1)	HUP0204399A3 (et)
IL (2)	IL151132A0 (et)
IS (1)	IS6491A (et)
MX (1)	MXPA02008233A (et)
NO (1)	NO329898B1 (et)
NZ (1)	NZ520355A (et)
PL (1)	PL358004A1 (et)
PT (1)	PT1259512E (et)
RU (1)	RU2002125451A (et)
SK (1)	SK12152002A3 (et)
TR (1)	TR200302214T4 (et)
UA (1)	UA72590C2 (et)
WO (1)	WO2001062758A1 (et)
ZA (1)	ZA200206590B (et)

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US7439358B2 (en) *	2006-02-08	2008-10-21	Boehringer Ingelheim International Gmbh	Specific salt, anhydrous and crystalline form of a dihydropteridione derivative
RU2437889C2 (ru) *	2006-09-29	2011-12-27	Астразенека Аб	НОВЫЕ 5,7-ДИЗАМЕЩЕННЫЕ ПРОИЗВОДНЫЕ [1,3]ТИАЗОЛО[4,5-d]ПИРИМИДИН-2-(3Н)-АМИНА И ИХ ПРИМЕНЕНИЕ В ТЕРАПИИ
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US8546566B2 (en)	2010-10-12	2013-10-01	Boehringer Ingelheim International Gmbh	Process for manufacturing dihydropteridinones and intermediates thereof
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2000
- 2000-02-23 GB GB0004128A patent/GB2359551A/en not_active Withdrawn
2001
- 2001-02-20 PL PL01358004A patent/PL358004A1/xx not_active Application Discontinuation
- 2001-02-20 CZ CZ20022839A patent/CZ20022839A3/cs unknown
- 2001-02-20 RU RU2002125451/04A patent/RU2002125451A/ru not_active Application Discontinuation
- 2001-02-20 CN CNB018054676A patent/CN1190437C/zh not_active Expired - Fee Related
- 2001-02-20 BR BR0108600-6A patent/BR0108600A/pt not_active Application Discontinuation
- 2001-02-20 NZ NZ520355A patent/NZ520355A/en not_active IP Right Cessation
- 2001-02-20 DK DK01906493T patent/DK1259512T3/da active
- 2001-02-20 EE EEP200200461A patent/EE200200461A/et unknown
- 2001-02-20 TR TR2003/02214T patent/TR200302214T4/xx unknown
- 2001-02-20 HU HU0204399A patent/HUP0204399A3/hu unknown
- 2001-02-20 US US10/204,814 patent/US6875868B2/en not_active Expired - Fee Related
- 2001-02-20 JP JP2001562540A patent/JP2003524012A/ja active Pending
- 2001-02-20 MX MXPA02008233A patent/MXPA02008233A/es active IP Right Grant
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- 2001-02-20 ES ES01906493T patent/ES2206402T3/es not_active Expired - Lifetime
- 2001-02-20 KR KR1020027011047A patent/KR100795758B1/ko not_active Expired - Fee Related
- 2001-02-20 DE DE60100851T patent/DE60100851T2/de not_active Expired - Lifetime
- 2001-02-20 PT PT01906493T patent/PT1259512E/pt unknown
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- 2001-02-20 WO PCT/SE2001/000374 patent/WO2001062758A1/en not_active Ceased
- 2001-02-20 AT AT01906493T patent/ATE250605T1/de active
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- 2001-02-20 AU AU34316/01A patent/AU782509B2/en not_active Ceased
- 2001-02-21 AR ARP010100773A patent/AR029805A1/es not_active Application Discontinuation
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2002
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- 2002-08-22 NO NO20024005A patent/NO329898B1/no not_active IP Right Cessation
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Also Published As

Publication number	Publication date
JP2003524012A (ja)	2003-08-12
IL151132A0 (en)	2003-04-10
KR20030005207A (ko)	2003-01-17
GB2359551A (en)	2001-08-29
BG107002A (bg)	2003-04-30
CN1190437C (zh)	2005-02-23
SK12152002A3 (sk)	2003-03-04
ES2206402T3 (es)	2004-05-16
US6875868B2 (en)	2005-04-05
HUP0204399A3 (en)	2004-11-29
CO5290258A1 (es)	2003-06-27
WO2001062758A1 (en)	2001-08-30
ZA200206590B (en)	2003-11-17
IL151132A (en)	2010-11-30
US20050171345A1 (en)	2005-08-04
HK1050899A1 (en)	2003-07-11
CA2400217A1 (en)	2001-08-30
IS6491A (is)	2002-08-07
EP1259512A1 (en)	2002-11-27
AU3431601A (en)	2001-09-03
AU782509B2 (en)	2005-08-04
BR0108600A (pt)	2002-11-12
DE60100851D1 (de)	2003-10-30
NO20024005L (no)	2002-10-22
AR029805A1 (es)	2003-07-16
CN1404482A (zh)	2003-03-19
NO20024005D0 (no)	2002-08-22
UA72590C2 (uk)	2005-03-15
PL358004A1 (en)	2004-08-09
CA2400217C (en)	2009-02-17
HUP0204399A2 (en)	2003-05-28
PT1259512E (pt)	2004-02-27
US7579342B2 (en)	2009-08-25
RU2002125451A (ru)	2004-01-10
KR100795758B1 (ko)	2008-01-21
MXPA02008233A (es)	2004-04-05
GB0004128D0 (en)	2000-04-12
DK1259512T3 (da)	2003-12-29
ATE250605T1 (de)	2003-10-15
NO329898B1 (no)	2011-01-24
DE60100851T2 (de)	2004-07-15
EP1259512B1 (en)	2003-09-24
NZ520355A (en)	2005-01-28
TR200302214T4 (tr)	2004-01-21
CZ20022839A3 (cs)	2002-11-13
US20030055250A1 (en)	2003-03-20

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