EE200300071A - Kinasoliini derivaadid - Google Patents

Kinasoliini derivaadid

Info

Publication number: EE200300071A
Authority: EE; Estonia
Prior art keywords: quinazoline derivatives; quinazoline; derivatives
Prior art date: 2000-08-21

Application number

EEP200300071A

Other languages

English (en)

Inventor

Fran�Ois Andr� Hennequin Laurent

Ple Patrick

Marie Paul Lambert Christine

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-21

Filing date

2001-08-15

Publication date

2004-12-15

2001-08-15 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2004-12-15 Publication of EE200300071A publication Critical patent/EE200300071A/et

2011-02-15 Publication of EE05387B1 publication Critical patent/EE05387B1/et

Links

125000002294 quinazolinyl group Chemical class N1=C(N=CC2=CC=CC=C12)* 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Neurology (AREA)
Immunology (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Biomedical Technology (AREA)
Oncology (AREA)
Neurosurgery (AREA)
Ophthalmology & Optometry (AREA)
Hematology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Emergency Medicine (AREA)
Vascular Medicine (AREA)
Gastroenterology & Hepatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

EEP200300071A 2000-08-21 2001-08-15 KinasoliiniÁderivaadid,ÁnendeÁvalmistamismeetodÁjaÁkasutamine EE05387B1 (et)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP00402320		2000-08-21
EP01401006		2001-04-19
PCT/GB2001/003649 WO2002016352A1 (en)	2000-08-21	2001-08-15	Quinazoline derivatives

Publications (2)

Publication Number	Publication Date
EE200300071A true EE200300071A (et)	2004-12-15
EE05387B1 EE05387B1 (et)	2011-02-15

Family

ID=26073540

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200300071A EE05387B1 (et)	2000-08-21	2001-08-15	KinasoliiniÁderivaadid,ÁnendeÁvalmistamismeetodÁjaÁkasutamine

Country Status (21)

Country	Link
US (1)	US7115615B2 (et)
EP (1)	EP1313727A1 (et)
JP (1)	JP2004506732A (et)
KR (2)	KR20080027400A (et)
CN (1)	CN100347169C (et)
AR (1)	AR033560A1 (et)
AU (2)	AU7860901A (et)
BR (1)	BR0113358A (et)
CA (1)	CA2419301C (et)
CZ (1)	CZ2003486A3 (et)
EE (1)	EE05387B1 (et)
IL (2)	IL154131A0 (et)
MX (1)	MXPA03001332A (et)
MY (1)	MY129809A (et)
NO (1)	NO326515B1 (et)
NZ (1)	NZ523702A (et)
PL (1)	PL202812B1 (et)
RU (1)	RU2267489C2 (et)
SK (1)	SK2142003A3 (et)
TW (1)	TWI280960B (et)
WO (1)	WO2002016352A1 (et)

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US6080747A (en)	1999-03-05	2000-06-27	Hughes Institute	JAK-3 inhibitors for treating allergic disorders
DE19911509A1 (de)	1999-03-15	2000-09-21	Boehringer Ingelheim Pharma	Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
SK3822002A3 (en)	1999-09-21	2002-10-08	Astrazeneca Ab	Quinazoline derivatives, process for the preparation thereof and their use
JP2003509497A (ja)	1999-09-21	2003-03-11	アストラゼネカアクチボラグ	キナゾリン化合物とそれらを含有する医薬組成物
GB9922173D0 (en)	1999-09-21	1999-11-17	Zeneca Ltd	Chemical compounds
US7160889B2 (en)	2000-04-07	2007-01-09	Astrazeneca Ab	Quinazoline compounds
UA73993C2 (uk)	2000-06-06	2005-10-17	Астразенека Аб	Хіназолінові похідні для лікування пухлин та фармацевтична композиція
AU2001292137A1 (en)	2000-10-13	2002-04-22	Astrazeneca Ab	Quinazoline derivatives
AU2001292138A1 (en)	2000-10-13	2002-04-22	Astrazeneca Ab	Quinazoline derivatives with anti-tumour activity
US20040063733A1 (en)	2000-10-25	2004-04-01	Lambert Christine Marie Paul	Quinazoline derivatives
WO2002085895A1 (en)	2001-04-19	2002-10-31	Astrazeneca Ab	Quinazoline derivatives
US7501516B2 (en)	2001-07-16	2009-03-10	Astrazeneca Ab	Quinoline derivatives and their use as tyrosine kinase inhibitors

2001
- 2001-08-15 US US10/344,678 patent/US7115615B2/en not_active Expired - Fee Related
- 2001-08-15 JP JP2002521453A patent/JP2004506732A/ja not_active Ceased
- 2001-08-15 SK SK214-2003A patent/SK2142003A3/sk not_active Application Discontinuation
- 2001-08-15 CZ CZ2003486A patent/CZ2003486A3/cs unknown
- 2001-08-15 MX MXPA03001332A patent/MXPA03001332A/es active IP Right Grant
- 2001-08-15 AU AU7860901A patent/AU7860901A/xx active Pending
- 2001-08-15 WO PCT/GB2001/003649 patent/WO2002016352A1/en not_active Ceased
- 2001-08-15 EP EP01956688A patent/EP1313727A1/en not_active Withdrawn
- 2001-08-15 RU RU2003107683/04A patent/RU2267489C2/ru not_active IP Right Cessation
- 2001-08-15 AU AU2001278609A patent/AU2001278609B2/en not_active Ceased
- 2001-08-15 IL IL15413101A patent/IL154131A0/xx unknown
- 2001-08-15 CA CA002419301A patent/CA2419301C/en not_active Expired - Fee Related
- 2001-08-15 NZ NZ523702A patent/NZ523702A/en unknown
- 2001-08-15 KR KR1020087005460A patent/KR20080027400A/ko not_active Withdrawn
- 2001-08-15 PL PL360591A patent/PL202812B1/pl not_active IP Right Cessation
- 2001-08-15 CN CNB018177409A patent/CN100347169C/zh not_active Expired - Fee Related
- 2001-08-15 BR BR0113358-6A patent/BR0113358A/pt not_active Application Discontinuation
- 2001-08-15 EE EEP200300071A patent/EE05387B1/et not_active IP Right Cessation
- 2001-08-15 KR KR1020037002441A patent/KR100821446B1/ko not_active Expired - Fee Related
- 2001-08-20 MY MYPI20013907A patent/MY129809A/en unknown
- 2001-08-21 AR ARP010103972A patent/AR033560A1/es not_active Application Discontinuation
- 2001-09-14 TW TW90122895A patent/TWI280960B/zh not_active IP Right Cessation
2003
- 2003-01-26 IL IL154131A patent/IL154131A/en not_active IP Right Cessation
- 2003-02-20 NO NO20030795A patent/NO326515B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
BR0113358A (pt)	2003-07-01
CN1471527A (zh)	2004-01-28
KR20030022416A (ko)	2003-03-15
WO2002016352A1 (en)	2002-02-28
NZ523702A (en)	2004-08-27
NO20030795L (no)	2003-04-04
CA2419301C (en)	2009-12-08
IL154131A (en)	2010-04-15
TWI280960B (en)	2007-05-11
CN100347169C (zh)	2007-11-07
MXPA03001332A (es)	2004-07-08
CA2419301A1 (en)	2002-02-28
RU2267489C2 (ru)	2006-01-10
NO326515B1 (no)	2008-12-22
EP1313727A1 (en)	2003-05-28
IL154131A0 (en)	2003-07-31
JP2004506732A (ja)	2004-03-04
AR033560A1 (es)	2003-12-26
PL360591A1 (en)	2004-09-06
KR100821446B1 (ko)	2008-04-10
NO20030795D0 (no)	2003-02-20
CZ2003486A3 (cs)	2003-05-14
MY129809A (en)	2007-05-31
EE05387B1 (et)	2011-02-15
KR20080027400A (ko)	2008-03-26
AU7860901A (en)	2002-03-04
US20040034046A1 (en)	2004-02-19
AU2001278609B2 (en)	2005-04-14
US7115615B2 (en)	2006-10-03
SK2142003A3 (en)	2003-07-01
PL202812B1 (pl)	2009-07-31

Legal Events

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2012-04-16	MM4A	Lapsed by not paying the annual fees	Effective date: 20110815

Publication	Publication Date	Title
NL300999I1 (nl)	2019-07-17	macimorelin
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PT1351959E (pt)	2005-09-30	Novos derivados de pleuromutilina
ATE280752T1 (de)	2004-11-15	Aminomethyl-phenyl-cyclohexanonderivate
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ATE374776T1 (de)	2007-10-15	Pyrrolotriazolopyrimidinonderivate
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