EP1906958A4 - Pyrazolo[3,4-b]pyridin-2-yl]-benzoesäure- derivate als hiv integrase-hemmer - Google Patents

Pyrazolo[3,4-b]pyridin-2-yl]-benzoesäure- derivate als hiv integrase-hemmer

Info

Publication number
EP1906958A4
EP1906958A4 EP06790527A EP06790527A EP1906958A4 EP 1906958 A4 EP1906958 A4 EP 1906958A4 EP 06790527 A EP06790527 A EP 06790527A EP 06790527 A EP06790527 A EP 06790527A EP 1906958 A4 EP1906958 A4 EP 1906958A4
Authority
EP
European Patent Office
Prior art keywords
baczoic
pyrazolo
pyridin
inhibitors
acid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
EP06790527A
Other languages
English (en)
French (fr)
Other versions
EP1906958A2 (de
Inventor
Brent Richard Stranix
Dominik Herbart
Valerie Perron
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ambrilia Biopharma Inc
Original Assignee
Ambrilia Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ambrilia Biopharma Inc filed Critical Ambrilia Biopharma Inc
Publication of EP1906958A2 publication Critical patent/EP1906958A2/de
Publication of EP1906958A4 publication Critical patent/EP1906958A4/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
EP06790527A 2005-06-27 2006-06-27 Pyrazolo[3,4-b]pyridin-2-yl]-benzoesäure- derivate als hiv integrase-hemmer Pending EP1906958A4 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69383305P 2005-06-27 2005-06-27
PCT/CA2006/001049 WO2007000043A2 (en) 2005-06-27 2006-06-27 Pyrazolo[3,4-b]pyridin-2-yl]-benzoic acid derivatives as hiv integrase inhibitors

Publications (2)

Publication Number Publication Date
EP1906958A2 EP1906958A2 (de) 2008-04-09
EP1906958A4 true EP1906958A4 (de) 2010-12-22

Family

ID=37595485

Family Applications (1)

Application Number Title Priority Date Filing Date
EP06790527A Pending EP1906958A4 (de) 2005-06-27 2006-06-27 Pyrazolo[3,4-b]pyridin-2-yl]-benzoesäure- derivate als hiv integrase-hemmer

Country Status (6)

Country Link
EP (1) EP1906958A4 (de)
JP (1) JP2008546813A (de)
CN (1) CN101243080A (de)
AU (1) AU2006264170A1 (de)
CA (1) CA2612300A1 (de)
WO (1) WO2007000043A2 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5269087B2 (ja) * 2007-11-16 2013-08-21 ギリアード サイエンシス インコーポレーテッド ヒト免疫不全ウイルス複製のインヒビター
WO2017222921A1 (en) * 2016-06-22 2017-12-28 Xavier University Of Louisiana 2-hydroxyisophthalic acid and its derivatives: methods of making and applications

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030096825A1 (en) * 2001-04-25 2003-05-22 Tao Wang Indole, azaindole and related heterocyclic amidopiperazine derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002356725B2 (en) * 2001-12-04 2008-07-17 F. Hoffmann-La Roche Ag Ring fused pyrazole derivatives
GB0230045D0 (en) * 2002-12-23 2003-01-29 Glaxo Group Ltd Compounds
AU2003286711A1 (en) * 2002-10-25 2004-05-13 Vertex Pharmaceuticals Incorporated Indazolinone compositions useful as kinase inhibitors
KR101312736B1 (ko) * 2003-02-27 2013-09-27 팔라우 파르마 에스에이 피라졸로피리딘 유도체

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030096825A1 (en) * 2001-04-25 2003-05-22 Tao Wang Indole, azaindole and related heterocyclic amidopiperazine derivatives

Also Published As

Publication number Publication date
EP1906958A2 (de) 2008-04-09
AU2006264170A1 (en) 2007-01-04
CN101243080A (zh) 2008-08-13
WO2007000043A3 (en) 2007-11-15
CA2612300A1 (en) 2007-01-04
WO2007000043A2 (en) 2007-01-04
JP2008546813A (ja) 2008-12-25

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