ES2074113T3 - Nuevos derivados de acido pirazolil acrilico, utiles como fungicidas sistemicos para la proteccion de plantas y materiales. - Google Patents
Nuevos derivados de acido pirazolil acrilico, utiles como fungicidas sistemicos para la proteccion de plantas y materiales.Info
- Publication number
- ES2074113T3 ES2074113T3 ES90124128T ES90124128T ES2074113T3 ES 2074113 T3 ES2074113 T3 ES 2074113T3 ES 90124128 T ES90124128 T ES 90124128T ES 90124128 T ES90124128 T ES 90124128T ES 2074113 T3 ES2074113 T3 ES 2074113T3
- Authority
- ES
- Spain
- Prior art keywords
- cyano
- nitro
- alkoxy
- halogen
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000002253 acid Substances 0.000 title 1
- 239000000417 fungicide Substances 0.000 title 1
- 239000000463 material Substances 0.000 title 1
- 230000009885 systemic effect Effects 0.000 title 1
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 4
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 4
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical group 0.000 abstract 3
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 3
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- 239000011593 sulfur Substances 0.000 abstract 2
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 2
- 125000000027 (C1-C10) alkoxy group Chemical group 0.000 abstract 1
- BBJHZSSIHPFLNS-UHFFFAOYSA-N 2-(1h-pyrazol-5-yl)prop-2-enoic acid Chemical class OC(=O)C(=C)C=1C=CNN=1 BBJHZSSIHPFLNS-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical group C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 1
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 1
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 1
- 125000005199 aryl carbonyloxy group Chemical group 0.000 abstract 1
- 230000000855 fungicidal effect Effects 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000005553 heteroaryloxy group Chemical group 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
UN DERIVADO DE ACIDO ACRILICO DE PIRAZOLILO QUE TIENE UNA ACTIVIDAD FUNGICIDA EN LAS PLANTAS, DE FORMULA DONDE: R SUB 1 Y R SUB 2 SON INDEPENDIENTEMENTE HIDROGENO O ALQUILO C SUB 1 C SUB 5; A ES UN GRUPO DE LA FORMULA: DONDE X ES INDEPENDIENTEMENTE HIDROGENO, HALOGENO, CIANO; NITRO; ALQUILO C SUB 1 10, ALQUENILO C SUB 2 UENILOXI C SUB 2 LQUICARBONILO C SUB 2 IDOS ENTRE HALOGENO , NITRO, CIANO, TRIFLUOROMETILO Y ALCOXI C SUB 1 ILCARBONILOXI C SUB 4 UB 13, ARILO C SUB 6 ETEROARILO C SUB 2 ENTRE OXIGENO, AZUFRE Y NITROGENO, HETEROARILOXI C SUB 2 C SUB 13 CON 1 TROGENO, ARALQUILO C SUB 7 SUB 12 OPCIONALMENTE SUSTITUIDO CON UNO O MAS SUSTITUTOS ELEGIDOS ENTRE HALOGENO , NITRO, CIANO, TRIFLUOROMETILO, ALQUILO C SUB 1 ANILLO FUNDIDO CON EL ANILLO DE BENCENO O EL ANILLO DE TIAZOL A LOS QUE ESTAN UNIDOS; Y B ES METOXICARBONILO O CIANO.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP32303589 | 1989-12-13 | ||
| JP7976390 | 1990-03-28 | ||
| JP27372490 | 1990-10-12 | ||
| JP02324113A JP3018490B2 (ja) | 1989-12-13 | 1990-11-27 | ピラゾリルアクリル酸誘導体、これを有効成分とする農園芸用殺菌剤およびその中間体 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2074113T3 true ES2074113T3 (es) | 1995-09-01 |
Family
ID=27466350
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES90124128T Expired - Lifetime ES2074113T3 (es) | 1989-12-13 | 1990-12-13 | Nuevos derivados de acido pirazolil acrilico, utiles como fungicidas sistemicos para la proteccion de plantas y materiales. |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US5055477A (es) |
| EP (1) | EP0433899B1 (es) |
| AT (1) | ATE121080T1 (es) |
| DE (1) | DE69018592T2 (es) |
| ES (1) | ES2074113T3 (es) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW201737B (es) * | 1990-10-31 | 1993-03-11 | Mitsubishi Chemicals Co Ltd | |
| HU9301218D0 (en) * | 1992-05-13 | 1993-08-30 | Sandoz Ag | Method for producing new pyrazole derivatives |
| JP3217191B2 (ja) * | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| CZ194795A3 (en) * | 1993-01-29 | 1995-12-13 | Ciba Geigy Ag | Derivatives of pyrazolylacrylic acid, process of their preparation and intermediates therefor, microbicides containing such acids and their use |
| AU693454B2 (en) * | 1993-05-27 | 1998-07-02 | Shell Internationale Research Maatschappij B.V. | Herbicidal thiazole derivatives |
| FR2705962B1 (fr) * | 1993-06-03 | 1995-07-13 | Rhone Poulenc Agrochimie | Arylpyrazoles fongicides. |
| EP0658547B1 (en) * | 1993-12-14 | 1998-03-11 | Mitsubishi Chemical Corporation | N-pyrazolyl carbamate derivative, agricultural/horticultural fungicide containing the same as active ingredient and production intermediate thereof |
| GB9417971D0 (en) * | 1994-09-07 | 1994-10-26 | Sandoz Ltd | Novel process |
| ES2274553T3 (es) * | 1998-03-27 | 2007-05-16 | Sds Biotech K.K. | Derivados de acido pirazolil acrilico y de acido pirazolil oximino-acetico, su preparacion y su utilizacion como fungicidas. |
| ATE268990T1 (de) * | 1999-09-24 | 2004-07-15 | Agro Kanesho Co Ltd | Insektizide und akarizide |
| ES2248581T3 (es) | 2001-03-12 | 2006-03-16 | Intercept Pharmaceuticals, Inc. | Esteroides como agonistas de fxr. |
| EP1513817A1 (en) * | 2002-05-24 | 2005-03-16 | Takeda Pharmaceutical Company Limited | 1, 2-azole derivatives with hypoglycemic and hypolipidemic activity |
| US10987362B2 (en) | 2004-03-12 | 2021-04-27 | Intercept Pharmaceuticals, Inc. | Treatment of fibrosis using FXR ligands |
| PL1734970T3 (pl) | 2004-03-12 | 2015-05-29 | Intercept Pharmaceuticals Inc | Leczenie zwłóknienia z zastosowaniem ligandów FXR |
| US20080051418A1 (en) * | 2004-11-26 | 2008-02-28 | Tsuyoshi Maekawa | Arylalkanoic Acid Derivative |
| ITMI20050912A1 (it) * | 2005-05-19 | 2006-11-20 | Erregierre Spa | Processo di preparazione di acidi 3-a-ya(b)-diidrossi-6-a(b)-alchil-5b-colanici |
| KR101555716B1 (ko) | 2007-01-19 | 2015-09-25 | 인터셉트 파마슈티컬즈, 인크. | Tgr5 조절제로서의 23-치환 담즙산 및 이의 사용 방법 |
| WO2010014836A2 (en) * | 2008-07-30 | 2010-02-04 | Intercept Pharmaceuticals, Inc. | Tgr5 modulators and methods of use thereof |
| DK2698375T3 (en) * | 2008-11-19 | 2018-05-28 | Intercept Pharmaceuticals Inc | TGR5 modulators and methods for using them |
| SI3336097T1 (sl) | 2012-06-19 | 2021-07-30 | Intercept Pharmaceuticals, Inc. | Priprava nekristalinične oblike obetiholne kisline |
| US9982008B2 (en) | 2012-06-19 | 2018-05-29 | Intercept Pharmaceuticals, Inc. | Preparation and uses of obeticholic acid |
| CN104672013A (zh) * | 2015-02-11 | 2015-06-03 | 吉林省柳俐粮食有限公司 | 一种防治稻瘟病的富硒水稻生产方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5661358A (en) * | 1979-10-24 | 1981-05-26 | Ishihara Sangyo Kaisha Ltd | Pyrazole derivative and herbicide containing the same |
| JPS57203069A (en) * | 1981-06-10 | 1982-12-13 | Nippon Tokushu Noyaku Seizo Kk | Pyrazole derivative, its preparation, and herbicide |
| NZ213630A (en) * | 1984-10-19 | 1990-02-26 | Ici Plc | Acrylic acid derivatives and fungicidal compositions |
| DE3519282A1 (de) * | 1985-05-30 | 1986-12-04 | Basf Ag, 6700 Ludwigshafen | Acrylsaeureester und fungizide, die diese verbindungen enthalten |
| DE3807232A1 (de) * | 1988-03-05 | 1989-09-14 | Bayer Ag | Substituierte acrylsaeureester |
-
1990
- 1990-12-13 ES ES90124128T patent/ES2074113T3/es not_active Expired - Lifetime
- 1990-12-13 US US07/625,762 patent/US5055477A/en not_active Expired - Fee Related
- 1990-12-13 DE DE69018592T patent/DE69018592T2/de not_active Expired - Fee Related
- 1990-12-13 AT AT90124128T patent/ATE121080T1/de active
- 1990-12-13 EP EP90124128A patent/EP0433899B1/en not_active Expired - Lifetime
-
1991
- 1991-07-17 US US07/734,292 patent/US5128481A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US5128481A (en) | 1992-07-07 |
| DE69018592D1 (de) | 1995-05-18 |
| ATE121080T1 (de) | 1995-04-15 |
| DE69018592T2 (de) | 1995-10-05 |
| US5055477A (en) | 1991-10-08 |
| EP0433899B1 (en) | 1995-04-12 |
| EP0433899A1 (en) | 1991-06-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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