ES2116645T3 - Procedimiento para la preparacion de derivados de n-acil-glicina. - Google Patents

Procedimiento para la preparacion de derivados de n-acil-glicina.

Info

Publication number
ES2116645T3
ES2116645T3 ES95106329T ES95106329T ES2116645T3 ES 2116645 T3 ES2116645 T3 ES 2116645T3 ES 95106329 T ES95106329 T ES 95106329T ES 95106329 T ES95106329 T ES 95106329T ES 2116645 T3 ES2116645 T3 ES 2116645T3
Authority
ES
Spain
Prior art keywords
sub
rest
aril
branched
saturated
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES95106329T
Other languages
English (en)
Inventor
Matthias Dr Beller
Hartmut Dr Fischer
Thomas Dr Gerdau
Peter Gross
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Application granted granted Critical
Publication of ES2116645T3 publication Critical patent/ES2116645T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/08—Preparation of carboxylic acid amides from amides by reaction at nitrogen atoms of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/30—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms
    • C07C233/31—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cephalosporin Compounds (AREA)
  • Catalysts (AREA)

Abstract

LA INVENCION SE REFIERE A UN PROCESO PARA LA ELABORACION DE DERIVADOS ACILGLICINA DE LA FORMULA GENERAL (I) DONDE R{SUP.1} SIGNIFICA HIDROGENO, UN RESTO (C{SUB.1} - C{SUB.26}) ALQUIL SATURADO, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.2} - C{SUB.24}) ALQUENIL NO SATURADO UNO O MULTIPLES VECES, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.6} - C{SUB.18}) ARIL, UN RESTO (C{SUB.1} - C{SUB.10} ALQUIL (C{SUB.6} - C{SUB.18} ARIL O UN RESTO - (C{SUB.2} - C{SUB.10} ALQUENIL (C{SUB.6} - C{SUB.18} ARIL EVENTUALMENTE NO SATURADO MULTIPLES VECES, R{SUP.2} ES HIDROGENO, UN RESTO (C{SUB.1} - C{SUB.26}) SATURADO, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.2} C{SUB.23}) ALQUENIL NO SATURADO UNA O MULTIPLES VECES, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.6} - C{SUB.18}) ARIL, UN RESTO (C{SUB.1} - C{SUB.10} ALQUIL - (C{SUB.6} C{SUB.18} O UN RESTO - (C{SUB.2} - C{SUB.10} - ALQUENIL (C{SUB.6} - C{SUB.18}) ARIL EVENTUALMENTE NO SATURADO MULTIPLES VECES Y R{SUP.3}SIGNIFICA HIDROGENO, UN RESTO (C{SUB.1} - C{SUB.10}) ALQUIL SATURADO, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.2} - C{SUB.10) ALQUENIL NO SATURADO UNA O MULTIPLES VECES, DE CADENA RECTA, RAMIFICADA O CICLICA, UN RESTO (C{SUB.6} C{SUB.18}) - ARIL, UN RESTO (C{SUB.1} - C{SUB.10} ALQUENIL (C{SUB.6} - C{SUB.18} O UN RESTO - (C{SUB.2} - C{SUB.10} ALQUENIL - (C{SUB.6} -C{SUB.18}) ARIL EVENTUALMENTE NO SATURADO MULTIPLES VECES, CARACTERIZANDOSE PORQUE UNA AMIDA DE ACIDO CARBOXILICO DE LA FORMULA GENERAL (II) DONDE R{SUP.1} Y R{SUP.2} POSEEN EL SIGNIFICADO ANTES DADO SE TRANSFORMAN CON UN ALDEHIDO CON LA FORMULA R{SUP.3}CHO EN PRESENCIA DE UN DISOLVENTE Y UN ACIDO PARA LA OBTENCION DE UN ACIL AMINO METILOL DE LA FORMULA (III) Y ESTE COMPUESTO A CONTINUACION, DESPUES DE LA ADICION DE UN CATALIZADOR DE COBALTO CARBONIL, SE CARBONILIZA EN UNA TEMPERATURA DESDE 20 HASTA 150 TA 150 BAR.
ES95106329T 1994-05-02 1995-04-27 Procedimiento para la preparacion de derivados de n-acil-glicina. Expired - Lifetime ES2116645T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4415312A DE4415312A1 (de) 1994-05-02 1994-05-02 Verfahren zur Herstellung von N-Acylglycinderivaten

Publications (1)

Publication Number Publication Date
ES2116645T3 true ES2116645T3 (es) 1998-07-16

Family

ID=6516994

Family Applications (1)

Application Number Title Priority Date Filing Date
ES95106329T Expired - Lifetime ES2116645T3 (es) 1994-05-02 1995-04-27 Procedimiento para la preparacion de derivados de n-acil-glicina.

Country Status (19)

Country Link
US (1) US5650537A (es)
EP (1) EP0680948B1 (es)
JP (1) JPH0848660A (es)
KR (1) KR950032085A (es)
CN (1) CN1120533A (es)
AT (1) ATE164832T1 (es)
AU (1) AU697803B2 (es)
BG (1) BG62649B1 (es)
BR (1) BR9501851A (es)
CA (1) CA2148335A1 (es)
CZ (1) CZ111295A3 (es)
DE (2) DE4415312A1 (es)
ES (1) ES2116645T3 (es)
HU (1) HU216071B (es)
PL (1) PL308418A1 (es)
RU (1) RU2140903C1 (es)
SI (1) SI9500148A (es)
TW (1) TW336928B (es)
ZA (1) ZA953435B (es)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19642494A1 (de) * 1996-10-15 1998-04-16 Clariant Gmbh Verwendung von Sarkosinaten als Asphalten-Dispergatoren
DE19650501A1 (de) * 1996-12-05 1998-06-10 Hoechst Ag Verfahren zur Wiedergewinnung von bei der Herstellung von N-Acyl-alpha-aminosäurederivaten durch Amidocarbonylierung eingesetzten Cobaltcarbonylkatalysatoren
AU740288B2 (en) * 1997-02-13 2001-11-01 Monsanto Company Method of preparing amino carboxylic acids
US6232494B1 (en) 1998-02-12 2001-05-15 Monsanto Company Process for the preparation of N-(phosphonomethyl)glycine by oxidizing N-substituted N-(phosphonomethyl)glycine
CN1210283C (zh) * 1998-02-12 2005-07-13 孟山都技术有限责任公司 通过氧化n－取代的草甘膦制备草甘膦的方法
US6417133B1 (en) 1998-02-25 2002-07-09 Monsanto Technology Llc Deeply reduced oxidation catalyst and its use for catalyzing liquid phase oxidation reactions
AU754281B2 (en) 1998-08-12 2002-11-14 Monsanto Company Continuous process for the preparation of N-(phosphonomethyl) iminodiacetic acid
DE60115019T2 (de) * 2000-05-22 2006-08-03 Monsanto Technology Llc. Reaktionssysteme zur herstellung von n-(phosphonomethyl)glyzin verbindungen
US7293871B2 (en) 2000-11-27 2007-11-13 Ophthonix, Inc. Apparatus and method of correcting higher-order aberrations of the human eye
GB0112324D0 (en) * 2001-05-21 2001-07-11 Croda Int Plc Compounds
RU2324676C2 (ru) * 2002-04-29 2008-05-20 Байокон Лимитид Кристаллический n-(транс-4-изопропилциклогексилкарбонил)-d-фенилаланин формы с для лечения сахарного диабета типа 2 и способ его получения
UA92134C2 (ru) * 2003-07-09 2010-10-11 Чугай Сейяку Кабушики Кайша Соединение, обладающее анти-вгс действием, и фармацевтическая композиция, содержащая его
GB0413090D0 (en) 2004-06-11 2004-07-14 Degussa Process for preparing amino acids using the amidocarbonylation reaction (2)
GB0413092D0 (en) * 2004-06-11 2004-07-14 Degussa Process for preparing amino acids using the amidocarbonylation reaction (1)
AR051926A1 (es) 2004-09-15 2007-02-21 Monsanto Technology Llc Catalizadores de oxidacion, procedimientos de preparacion de dichos catalizadores y proceso para la elaboracion de n-( fosfonometil)glicina o una sal de la misma
RU2417218C2 (ru) * 2005-03-29 2011-04-27 Эдвард Так ВЕЙ Эфиры n-алкилкарбониламинокислот и n-алкилкарбониламинолактоны и их применение
DE102007055265A1 (de) * 2007-11-20 2009-05-28 Clariant International Ltd. Verfahren zur Herstellung von Acylglycinaten
US8252953B2 (en) 2008-05-01 2012-08-28 Monsanto Technology Llc Metal utilization in supported, metal-containing catalysts
RU2517179C2 (ru) * 2008-08-15 2014-05-27 Дзе Проктер Энд Гэмбл Компани Синтез производных циклогексана, используемых в потребительских товарах в качестве оказывающих сенсорное воздействие веществ
DE102011107503A1 (de) * 2011-07-15 2012-03-01 Clariant International Ltd. Verfahren zur Herstellung von Acylglycinaten und Zusammensetzungen enthaltend derartige Verbindungen
CN102268101A (zh) * 2011-08-31 2011-12-07 南京财经大学 一种高纯度紫菜多糖的酶辅助提取方法
KR101253462B1 (ko) 2012-10-22 2013-04-10 재 욱 한 진열대용 수직프레임 및 이를 이용한 다용도 조립식 진열대
EP2805976A1 (en) 2013-05-24 2014-11-26 Huntsman International Llc Aldehyde comprising compositions suitable for making curable polyisocyanate compositions
CN111518047B (zh) * 2019-02-01 2024-05-24 鲁南制药集团股份有限公司 Magl抑制剂及制备方法和用途
CN111518048B (zh) * 2019-02-01 2024-04-30 鲁南制药集团股份有限公司 Magl抑制剂、制备方法和用途
CN111518049B (zh) * 2019-02-01 2024-05-03 鲁南制药集团股份有限公司 Magl抑制剂、制备方法及用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR862365A (fr) * 1938-12-15 1941-03-05 Du Pont Production d'esters d'alcoylolamides
DE849554C (de) * 1943-03-26 1952-09-15 Ciba Geigy Verfahren zur Herstellung von neuen Amidabkoemmlingen
US4918222A (en) * 1984-07-27 1990-04-17 Texaco Inc. Process for synthesis of N-acetylglycine
US4891442A (en) * 1987-03-09 1990-01-02 Texaco Inc. Process for synthesis of β-phenylalanine
DE3917880A1 (de) * 1989-06-01 1990-12-06 Kali Chemie Ag Neue acylaminosaeurederivate enthaltende arzneimittel und diaetetika
GB2252770A (en) * 1991-02-14 1992-08-19 Shell Int Research The preparation of n-acyl-alpha-amino acids

Also Published As

Publication number Publication date
TW336928B (en) 1998-07-21
SI9500148A (en) 1995-12-31
HU9501217D0 (en) 1995-06-28
JPH0848660A (ja) 1996-02-20
EP0680948B1 (de) 1998-04-08
AU697803B2 (en) 1998-10-15
BR9501851A (pt) 1996-04-09
EP0680948A1 (de) 1995-11-08
BG62649B1 (bg) 2000-04-28
US5650537A (en) 1997-07-22
RU2140903C1 (ru) 1999-11-10
RU95106642A (ru) 1997-01-10
ATE164832T1 (de) 1998-04-15
KR950032085A (ko) 1995-12-20
AU1771995A (en) 1995-11-09
HUT71261A (en) 1995-11-28
BG99598A (en) 1996-04-30
ZA953435B (en) 1996-01-17
CA2148335A1 (en) 1995-11-03
HU216071B (hu) 1999-04-28
CN1120533A (zh) 1996-04-17
PL308418A1 (en) 1995-11-13
DE59501814D1 (de) 1998-05-14
DE4415312A1 (de) 1995-11-09
CZ111295A3 (en) 1995-12-13

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