ES2148786T3 - Derivados de alfa-hidrazinoacidos y procedimiento para su preparacion. - Google Patents
Derivados de alfa-hidrazinoacidos y procedimiento para su preparacion.Info
- Publication number
- ES2148786T3 ES2148786T3 ES96930204T ES96930204T ES2148786T3 ES 2148786 T3 ES2148786 T3 ES 2148786T3 ES 96930204 T ES96930204 T ES 96930204T ES 96930204 T ES96930204 T ES 96930204T ES 2148786 T3 ES2148786 T3 ES 2148786T3
- Authority
- ES
- Spain
- Prior art keywords
- radical
- designates
- alfa
- procedure
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000002253 acid Substances 0.000 title abstract 2
- 150000003254 radicals Chemical class 0.000 abstract 3
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical class [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- -1 RADICAL PHENYL Chemical group 0.000 abstract 2
- 229910052799 carbon Inorganic materials 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical group [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 150000001723 carbon free-radicals Chemical class 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 230000001681 protective effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C281/00—Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
- C07C281/02—Compounds containing any of the groups, e.g. carbazates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
- C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
- C07K1/1072—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Analytical Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Peptides Or Proteins (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
DERIVADO DE AL - HIDRACINOACIDA DE FORMULA GENERAL (I), EN LA QUE R 1 , R 2 , R 3 DESIGNAN EL HIDROGENO O UN RADICAL CARBONADO, CUANDO R 2 Y R 3 SON DIFERENTES, C* DESIGNA UN CARBONO ASIMETRICO DE CONFIGURACION L, D O DL, R 4 Y R 5 DESIGNAN UN GRUPO PROTECTOR, CARACTERIZADO PORQUE R 4 DESIGNA UN RADICAL BENCILO ARCH 2 DE FORMULA (A), EN DONDE AR DESIGNA UN RADICAL FENILO O FENILO SUSTITUIDO POR UNO O VARIOS GRUPOS X, SIENDO X EL HIDROGENO, UN HALOGENO, UN RADICAL NITRO O UN RADICAL ALQUILO, Y PORQUE R 5 DESIGNA UN GRUPO Y - O - CO, EN EL QUE Y DESIGNA UN RADICAL CARBONADO DIFERENTE DE R 4 .
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9510685A FR2738564B1 (fr) | 1995-09-07 | 1995-09-07 | Nouveaux derives d'alpha-hydrazinoacides et procede pour les fabriquer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2148786T3 true ES2148786T3 (es) | 2000-10-16 |
Family
ID=9482477
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES96930204T Expired - Lifetime ES2148786T3 (es) | 1995-09-07 | 1996-09-04 | Derivados de alfa-hidrazinoacidos y procedimiento para su preparacion. |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5962722A (es) |
| EP (1) | EP0853612B1 (es) |
| JP (1) | JPH11512109A (es) |
| DE (1) | DE69608906T2 (es) |
| ES (1) | ES2148786T3 (es) |
| FR (1) | FR2738564B1 (es) |
| WO (1) | WO1997009303A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19623892A1 (de) * | 1996-06-06 | 1997-12-11 | Hoechst Schering Agrevo Gmbh | Substituierte Pyrazolyl-pyrazolderivate |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS51138602A (en) * | 1975-05-15 | 1976-11-30 | Shunichi Yamada | Process for preparing alpha-hydrazino carboxylic acids |
-
1995
- 1995-09-07 FR FR9510685A patent/FR2738564B1/fr not_active Expired - Fee Related
-
1996
- 1996-04-09 US US09/029,628 patent/US5962722A/en not_active Expired - Fee Related
- 1996-09-04 EP EP96930204A patent/EP0853612B1/fr not_active Expired - Lifetime
- 1996-09-04 ES ES96930204T patent/ES2148786T3/es not_active Expired - Lifetime
- 1996-09-04 DE DE69608906T patent/DE69608906T2/de not_active Expired - Fee Related
- 1996-09-04 JP JP9510904A patent/JPH11512109A/ja active Pending
- 1996-09-04 WO PCT/FR1996/001349 patent/WO1997009303A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO1997009303A1 (fr) | 1997-03-13 |
| EP0853612B1 (fr) | 2000-06-14 |
| US5962722A (en) | 1999-10-05 |
| EP0853612A1 (fr) | 1998-07-22 |
| FR2738564B1 (fr) | 1997-10-24 |
| DE69608906D1 (de) | 2000-07-20 |
| FR2738564A1 (fr) | 1997-03-14 |
| DE69608906T2 (de) | 2001-03-01 |
| JPH11512109A (ja) | 1999-10-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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