ES2157027T3 - Oxazolidinonas sustituidas y su uso como farmacos antibacterianos. - Google Patents

Oxazolidinonas sustituidas y su uso como farmacos antibacterianos.

Info

Publication number
ES2157027T3
ES2157027T3 ES97101509T ES97101509T ES2157027T3 ES 2157027 T3 ES2157027 T3 ES 2157027T3 ES 97101509 T ES97101509 T ES 97101509T ES 97101509 T ES97101509 T ES 97101509T ES 2157027 T3 ES2157027 T3 ES 2157027T3
Authority
ES
Spain
Prior art keywords
antibacterial
oxazolidinones
pharmacos
replaced
medications
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES97101509T
Other languages
English (en)
Inventor
Bernd Dr Riedl
Dieter Dr Habich
Andreas Dr Stolle
Martin Dr Ruppelt
Stephan Dr Bartel
Walter Dr Guarnieri
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Application granted granted Critical
Publication of ES2157027T3 publication Critical patent/ES2157027T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6581—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms
    • C07F9/6584—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms having one phosphorus atom as ring hetero atom
    • C07F9/65842—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring
    • C07F9/65844—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring the phosphorus atom being part of a five-membered ring which may be condensed with another ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

LA PRESENTE INVENCION TRATA DE NUEVAS OXAZOLIDINONAS DE FORMULA GENERAL (I) EN DONDE LOS SUSTITUYENTES TIENEN EL SIGNIFICADO DADO EN LA DESCRIPCION, PROCEDIMIENTO PARA SU OBTENCION Y SU UTILIZACION COMO MEDICAMENTOS, EN PARTICULAR COMO MEDICAMENTOS ANTIBACTERIANOS.
ES97101509T 1996-02-06 1997-01-31 Oxazolidinonas sustituidas y su uso como farmacos antibacterianos. Expired - Lifetime ES2157027T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19604223A DE19604223A1 (de) 1996-02-06 1996-02-06 Neue substituierte Oxazolidinone

Publications (1)

Publication Number Publication Date
ES2157027T3 true ES2157027T3 (es) 2001-08-01

Family

ID=7784633

Family Applications (1)

Application Number Title Priority Date Filing Date
ES97101509T Expired - Lifetime ES2157027T3 (es) 1996-02-06 1997-01-31 Oxazolidinonas sustituidas y su uso como farmacos antibacterianos.

Country Status (36)

Country Link
US (1) US5792765A (es)
EP (1) EP0789025B1 (es)
JP (1) JPH09316073A (es)
KR (1) KR970061888A (es)
CN (1) CN1160051A (es)
AR (1) AR005703A1 (es)
AT (1) ATE200285T1 (es)
AU (1) AU1251697A (es)
BG (1) BG101193A (es)
BR (1) BR9700885A (es)
CA (1) CA2196862A1 (es)
CO (1) CO4560411A1 (es)
CZ (1) CZ34097A3 (es)
DE (2) DE19604223A1 (es)
DK (1) DK0789025T3 (es)
EE (1) EE9700043A (es)
ES (1) ES2157027T3 (es)
GR (1) GR3036015T3 (es)
HR (1) HRP970048A2 (es)
HU (1) HUP9700358A3 (es)
ID (1) ID15881A (es)
IL (1) IL120125A0 (es)
MX (1) MX9700886A (es)
NO (1) NO970511L (es)
NZ (1) NZ314179A (es)
PL (1) PL318277A1 (es)
PT (1) PT789025E (es)
SG (1) SG50791A1 (es)
SI (1) SI0789025T1 (es)
SK (1) SK15897A3 (es)
SV (1) SV1997000009A (es)
TN (1) TNSN97032A1 (es)
TR (1) TR199700092A2 (es)
TW (1) TW350845B (es)
YU (1) YU4397A (es)
ZA (1) ZA97927B (es)

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GB9821938D0 (en) * 1998-10-09 1998-12-02 Zeneca Ltd Chemical compounds
JP2000204084A (ja) * 1998-11-11 2000-07-25 Hokuriku Seiyaku Co Ltd チオカルバミド酸誘導体
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AU1045300A (en) * 1998-11-17 2000-06-05 Bayer Aktiengesellschaft Novel heterocyclyl-substituted oxazolidone derivatives
DE69933526D1 (de) 1998-12-07 2006-11-23 Takasago Perfumery Co Ltd Verfahren zur Herstellung von optisch aktiven Oxazolidinonderivate
JP2003501351A (ja) * 1999-05-27 2003-01-14 ファルマシア・アンド・アップジョン・カンパニー 抗菌剤としての二環系オキサゾリジノン
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Also Published As

Publication number Publication date
AU1251697A (en) 1997-08-14
IL120125A0 (en) 1997-06-10
BG101193A (en) 1999-02-26
SV1997000009A (es) 1997-10-23
NO970511D0 (no) 1997-02-05
HUP9700358A2 (hu) 1998-07-28
HUP9700358A3 (en) 1999-08-30
PL318277A1 (en) 1997-08-18
CN1160051A (zh) 1997-09-24
MX9700886A (es) 1998-04-30
NO970511L (no) 1997-08-07
ATE200285T1 (de) 2001-04-15
DE59703261D1 (de) 2001-05-10
SG50791A1 (en) 1998-07-20
JPH09316073A (ja) 1997-12-09
CZ34097A3 (en) 1997-08-13
TNSN97032A1 (fr) 2005-03-15
KR970061888A (ko) 1997-09-12
TR199700092A2 (tr) 1997-08-21
EP0789025A1 (de) 1997-08-13
GR3036015T3 (en) 2001-09-28
SI0789025T1 (en) 2001-08-31
ID15881A (id) 1997-08-14
CA2196862A1 (en) 1997-08-07
TW350845B (en) 1999-01-21
CO4560411A1 (es) 1998-02-10
ZA97927B (en) 1997-08-19
DK0789025T3 (da) 2001-06-18
US5792765A (en) 1998-08-11
HU9700358D0 (en) 1997-03-28
HRP970048A2 (en) 1998-04-30
BR9700885A (pt) 1998-10-27
PT789025E (pt) 2001-07-31
EP0789025B1 (de) 2001-04-04
NZ314179A (en) 1998-12-23
EE9700043A (et) 1997-08-15
SK15897A3 (en) 1997-10-08
DE19604223A1 (de) 1997-08-07
YU4397A (sh) 1999-09-27
AR005703A1 (es) 1999-07-14

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