ES2177980T3 - Procedimiento para la preparacion de un tiazol disustituido. - Google Patents

Procedimiento para la preparacion de un tiazol disustituido.

Info

Publication number
ES2177980T3
ES2177980T3 ES97923661T ES97923661T ES2177980T3 ES 2177980 T3 ES2177980 T3 ES 2177980T3 ES 97923661 T ES97923661 T ES 97923661T ES 97923661 T ES97923661 T ES 97923661T ES 2177980 T3 ES2177980 T3 ES 2177980T3
Authority
ES
Spain
Prior art keywords
preparation
tiazol
procedure
disposed
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES97923661T
Other languages
English (en)
Inventor
Patricia A Oliver
Arthur J Cooper
John E Lallaman
Denton C Landgridge
Jieh-Heh J Tien
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Application granted granted Critical
Publication of ES2177980T3 publication Critical patent/ES2177980T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28Radicals substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Cephalosporin Compounds (AREA)
  • Application Of Or Painting With Fluid Materials (AREA)

Abstract

SE DESCRIBE UN PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE N - ((N - METIL - N - ((2 - ISOPROPIL - 4 TIAZOLIL)METIL)AMINO)CARBONIL) - AMINOACIDO.
ES97923661T 1996-06-28 1997-05-19 Procedimiento para la preparacion de un tiazol disustituido. Expired - Lifetime ES2177980T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/673,445 US6160122A (en) 1996-06-28 1996-06-28 Process for the preparation of a disubstituted thiazole

Publications (1)

Publication Number Publication Date
ES2177980T3 true ES2177980T3 (es) 2002-12-16

Family

ID=24702690

Family Applications (1)

Application Number Title Priority Date Filing Date
ES97923661T Expired - Lifetime ES2177980T3 (es) 1996-06-28 1997-05-19 Procedimiento para la preparacion de un tiazol disustituido.

Country Status (11)

Country Link
US (1) US6160122A (es)
EP (1) EP0854872B1 (es)
JP (2) JPH11512114A (es)
AT (1) ATE215535T1 (es)
CA (1) CA2229788A1 (es)
DE (1) DE69711590T2 (es)
DK (1) DK0854872T3 (es)
ES (1) ES2177980T3 (es)
MX (1) MX9801636A (es)
PT (1) PT854872E (es)
WO (1) WO1998000410A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY121765A (en) 1998-07-20 2006-02-28 Abbott Lab Polymorph of ritonavir
TR201809435T4 (tr) 2000-01-19 2018-07-23 Abbvie Inc Geliştirilmiş farmasötik formülasyonlar.
DE102012024596A1 (de) * 2012-12-13 2014-06-18 Zm Präzisionsdentaltechnik Gmbh Dentalimplantat

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5142056A (en) * 1989-05-23 1992-08-25 Abbott Laboratories Retroviral protease inhibiting compounds
DE3325734A1 (de) * 1983-07-16 1985-01-24 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von n-(3,5-dichlorphenyl)-oxazolidin-2,4-dionen
US5539122A (en) * 1989-05-23 1996-07-23 Abbott Laboratories Retroviral protease inhibiting compounds
BE1005720A3 (fr) * 1992-03-20 1993-12-28 Solvay Procede de synthese peptidique et nouveaux intermediaires de synthese.
CA2170020C (en) * 1992-12-29 2005-08-02 Dale J. Kempf Retroviral protease inhibiting compounds
BE1007183A3 (fr) * 1993-06-18 1995-04-18 Solvay Ureines derivees d'alpha, omega-diaminoacides et procede pour leur preparation.
BE1007184A3 (fr) * 1993-06-18 1995-04-18 Solvay Procede de preparation d'un amide d'alpha-aminoacide, utilisable en synthese peptidique.
KR0125117B1 (ko) * 1994-06-15 1997-12-05 성재갑 항 에이즈(aids)효과를 갖는 신규한 인간 면역 결핍 바이러스(hiv)프로테아제 억제 화합물 및 그의 제조방법

Also Published As

Publication number Publication date
PT854872E (pt) 2002-09-30
DE69711590T2 (de) 2002-11-14
CA2229788A1 (en) 1998-01-08
ATE215535T1 (de) 2002-04-15
DK0854872T3 (da) 2002-07-29
EP0854872A1 (en) 1998-07-29
US6160122A (en) 2000-12-12
JPH11512114A (ja) 1999-10-19
WO1998000410A1 (en) 1998-01-08
JP2009035560A (ja) 2009-02-19
DE69711590D1 (de) 2002-05-08
MX9801636A (es) 1998-05-31
EP0854872B1 (en) 2002-04-03

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