ES2421598T3 - Composición glucopeptídica con actividad antibiótica mejorada - Google Patents

Composición glucopeptídica con actividad antibiótica mejorada

Info

Publication number
ES2421598T3
ES2421598T3 ES04762852T ES04762852T ES2421598T3 ES 2421598 T3 ES2421598 T3 ES 2421598T3 ES 04762852 T ES04762852 T ES 04762852T ES 04762852 T ES04762852 T ES 04762852T ES 2421598 T3 ES2421598 T3 ES 2421598T3
Authority
ES
Spain
Prior art keywords
glucopeptide
composition
antibiotic activity
improved antibiotic
glycopeptides
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES04762852T
Other languages
English (en)
Inventor
Anita Mathiesen
Torben Koch
Trine Suhr-Jessen
Joern Thyme
Tiemen Reijns
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Xellia Pharmaceuticals ApS
Original Assignee
Axellia Pharmaceuticals ApS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Axellia Pharmaceuticals ApS filed Critical Axellia Pharmaceuticals ApS
Application granted granted Critical
Publication of ES2421598T3 publication Critical patent/ES2421598T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/14Peptides containing saccharide radicals; Derivatives thereof, e.g. bleomycin, phleomycin, muramylpeptides or vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Compounds Of Unknown Constitution (AREA)

Abstract

Composición antibiótica glucopeptídica apropiada para la administración como medicamento a un paciente y quecomprende: A: un antibiótico glucopeptídico en su forma glucosilada; y B: un resto de un antibiótico glucopeptídico que carece de una o varias unidades de glucosilo; siendo elcontenido de B de 14% a 73% (p/p) del contenido total de glucopéptidos y glucopéptidos desglucosilados,calculado como: 10 B / (A + B) (p/p).
ES04762852T 2003-09-17 2004-09-17 Composición glucopeptídica con actividad antibiótica mejorada Expired - Lifetime ES2421598T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03021000A EP1516626B1 (en) 2003-09-17 2003-09-17 A Teicoplanin composition with improved antibiotic activity
PCT/DK2004/000632 WO2005025599A1 (en) 2003-09-17 2004-09-17 A glycopeptide composition with improved antibiotic activity

Publications (1)

Publication Number Publication Date
ES2421598T3 true ES2421598T3 (es) 2013-09-04

Family

ID=34178422

Family Applications (2)

Application Number Title Priority Date Filing Date
ES03021000T Expired - Lifetime ES2278101T3 (es) 2003-09-17 2003-09-17 Composicion de teicoplanina con actividad antibiotica mejorada.
ES04762852T Expired - Lifetime ES2421598T3 (es) 2003-09-17 2004-09-17 Composición glucopeptídica con actividad antibiótica mejorada

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES03021000T Expired - Lifetime ES2278101T3 (es) 2003-09-17 2003-09-17 Composicion de teicoplanina con actividad antibiotica mejorada.

Country Status (14)

Country Link
US (2) US7981859B2 (es)
EP (2) EP1516626B1 (es)
JP (1) JP2007505841A (es)
CN (1) CN1871023B (es)
AT (1) ATE349224T1 (es)
AU (1) AU2004271688B2 (es)
CA (1) CA2538842C (es)
DE (1) DE60310717T2 (es)
DK (1) DK1516626T3 (es)
ES (2) ES2278101T3 (es)
NO (1) NO20061368L (es)
PT (1) PT1516626E (es)
SI (1) SI1516626T1 (es)
WO (1) WO2005025599A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1516626T3 (da) * 2003-09-17 2007-04-30 Alpharma Aps Teicoplanin-sammensætning med forbedret antibiotisk aktivitet
EP1806150A1 (en) * 2006-01-05 2007-07-11 NEED PHARMA S.r.l. Teicoplanin composition
US20070173438A1 (en) * 2006-01-13 2007-07-26 The Scripps Research Institute [PSI[CH2NH]PG4] glycopeptide antibiotic analogs
KR20100109934A (ko) 2007-12-26 2010-10-11 시오노기세야쿠 가부시키가이샤 글리코펩티드 항생 물질 배당화 유도체
CN106132980A (zh) * 2014-01-28 2016-11-16 中央研究院 肽可霉素类似物及其用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1496386A (en) * 1975-03-05 1977-12-30 Lepetit Spa Antibiotics
GB8307847D0 (en) * 1983-03-22 1983-04-27 Lepetit Spa Antibiotics l 17054 and l 17046
GB8420405D0 (en) * 1984-08-10 1984-09-12 Lepetit Spa Preparing antibiotic l 17046
GB8512795D0 (en) * 1985-05-21 1985-06-26 Lepetit Spa Increasing ratio of components of teicoplanin a2 complex
GB8608798D0 (en) 1986-04-11 1986-05-14 Lepetit Spa Recovery of glycopeptide antibiotics from aqueous solutions
GB8726859D0 (en) * 1987-11-17 1987-12-23 Lepetit Spa 22-dechlorotei-coplanins
IE64155B1 (en) * 1989-03-29 1995-07-12 Lepetit Spa New substituted alkylamide derivatives of teicoplanin
JPH0597672A (ja) * 1991-10-08 1993-04-20 Terumo Corp アミド誘導体含有固形製剤およびその製造方法
DK1516626T3 (da) 2003-09-17 2007-04-30 Alpharma Aps Teicoplanin-sammensætning med forbedret antibiotisk aktivitet

Also Published As

Publication number Publication date
PT1516626E (pt) 2007-04-30
US20070287663A1 (en) 2007-12-13
CA2538842A1 (en) 2005-03-24
US20050080004A1 (en) 2005-04-14
EP1670496B1 (en) 2013-05-22
CN1871023A (zh) 2006-11-29
DE60310717T2 (de) 2007-10-11
SI1516626T1 (sl) 2007-04-30
AU2004271688A1 (en) 2005-03-24
DK1516626T3 (da) 2007-04-30
EP1516626B1 (en) 2006-12-27
EP1670496A1 (en) 2006-06-21
CN1871023B (zh) 2012-08-22
JP2007505841A (ja) 2007-03-15
US7919470B2 (en) 2011-04-05
ATE349224T1 (de) 2007-01-15
CA2538842C (en) 2012-08-21
EP1516626A1 (en) 2005-03-23
US7981859B2 (en) 2011-07-19
AU2004271688B2 (en) 2009-05-28
DE60310717D1 (de) 2007-02-08
ES2278101T3 (es) 2007-08-01
WO2005025599A1 (en) 2005-03-24
NO20061368L (no) 2006-06-15

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