ES390459A1 - Oestrone derivative and a process for its manufacture - Google Patents
Oestrone derivative and a process for its manufactureInfo
- Publication number
- ES390459A1 ES390459A1 ES390459A ES390459A ES390459A1 ES 390459 A1 ES390459 A1 ES 390459A1 ES 390459 A ES390459 A ES 390459A ES 390459 A ES390459 A ES 390459A ES 390459 A1 ES390459 A1 ES 390459A1
- Authority
- ES
- Spain
- Prior art keywords
- free
- formula
- manufacture
- oxo group
- see formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 238000000034 method Methods 0.000 title abstract 2
- DNXHEGUUPJUMQT-CBZIJGRNSA-N Estrone Chemical class OC1=CC=C2[C@H]3CC[C@](C)(C(CC4)=O)[C@@H]4[C@@H]3CCC2=C1 DNXHEGUUPJUMQT-CBZIJGRNSA-N 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000004043 oxo group Chemical group O=* 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- XCIXKGXIYUWCLL-UHFFFAOYSA-N cyclopentanol Chemical compound OC1CCCC1 XCIXKGXIYUWCLL-UHFFFAOYSA-N 0.000 abstract 1
- 230000001076 estrogenic effect Effects 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 150000003431 steroids Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/168—Steroids
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/184—Hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Polymers & Plastics (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Husbandry (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Procedure to obtain a new steroid of high oestrogenic efficacy, with the formula: ** (See formula) ** characterized in that a compound of formula: ** (See formula) ** wherein R stands for a free or ketalized oxo group, or a free or esterified hydroxy group, is etherified in the 3-position with cyclopentanol and the residue R is optionally transformed into a free oxo group. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH621770A CH536826A (en) | 1970-04-24 | 1970-04-24 | Process for the production of a new, highly estrogenic steroid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES390459A1 true ES390459A1 (en) | 1973-06-01 |
Family
ID=4306123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES390459A Expired ES390459A1 (en) | 1970-04-24 | 1971-04-22 | Oestrone derivative and a process for its manufacture |
Country Status (17)
| Country | Link |
|---|---|
| AT (1) | AT307639B (en) |
| BE (1) | BE766182A (en) |
| CA (1) | CA925852A (en) |
| CH (2) | CH536826A (en) |
| CS (1) | CS151091B2 (en) |
| DE (1) | DE2118996A1 (en) |
| DK (2) | DK129451B (en) |
| ES (1) | ES390459A1 (en) |
| FI (1) | FI48827C (en) |
| FR (1) | FR2092080B1 (en) |
| GB (1) | GB1330071A (en) |
| IE (1) | IE35071B1 (en) |
| IL (1) | IL36652A (en) |
| NL (1) | NL7105576A (en) |
| PL (1) | PL73563B1 (en) |
| SE (1) | SE385588B (en) |
| SU (1) | SU399117A3 (en) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1866M (en) * | 1961-04-07 | 1963-06-17 | Vismara Francesco Spa | New ethers of estrogen hormones. |
| FR1434172A (en) * | 1963-12-24 | 1966-04-08 | Ciba Geigy | Process for preparing new substituted estrones |
| BE755689A (en) * | 1969-09-03 | 1971-03-03 | Upjohn Co | NEW 7 BETA-ALKYL-19- NORTESTOSTERONES MANUFACTURING PROCESS |
-
1970
- 1970-04-24 CH CH621770A patent/CH536826A/en not_active IP Right Cessation
- 1970-04-24 CH CH1870072A patent/CH534140A/en not_active IP Right Cessation
-
1971
- 1971-04-16 CA CA110524A patent/CA925852A/en not_active Expired
- 1971-04-19 IL IL36652A patent/IL36652A/en unknown
- 1971-04-20 DE DE19712118996 patent/DE2118996A1/en active Pending
- 1971-04-20 IE IE489/71A patent/IE35071B1/en unknown
- 1971-04-21 GB GB1042771*[A patent/GB1330071A/en not_active Expired
- 1971-04-22 FR FR7114320A patent/FR2092080B1/fr not_active Expired
- 1971-04-22 ES ES390459A patent/ES390459A1/en not_active Expired
- 1971-04-22 PL PL1971147685A patent/PL73563B1/pl unknown
- 1971-04-23 CS CS2984A patent/CS151091B2/cs unknown
- 1971-04-23 BE BE766182A patent/BE766182A/en unknown
- 1971-04-23 AT AT350971A patent/AT307639B/en not_active IP Right Cessation
- 1971-04-23 FI FI711129A patent/FI48827C/en active
- 1971-04-23 SU SU1649255A patent/SU399117A3/ru active
- 1971-04-23 NL NL7105576A patent/NL7105576A/xx unknown
- 1971-04-23 SE SE7105301A patent/SE385588B/en unknown
- 1971-04-23 DK DK196971AA patent/DK129451B/en unknown
-
1972
- 1972-08-18 DK DK411972AA patent/DK128110B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CH534140A (en) | 1973-02-28 |
| SE385588B (en) | 1976-07-12 |
| SU399117A3 (en) | 1973-09-27 |
| DK128110B (en) | 1974-03-04 |
| CA925852A (en) | 1973-05-08 |
| FI48827B (en) | 1974-09-30 |
| FI48827C (en) | 1975-01-10 |
| IL36652A0 (en) | 1971-06-23 |
| CH536826A (en) | 1973-05-15 |
| NL7105576A (en) | 1971-10-26 |
| DK129451C (en) | 1975-04-28 |
| FR2092080B1 (en) | 1974-10-18 |
| AT307639B (en) | 1973-05-25 |
| IE35071B1 (en) | 1975-10-29 |
| GB1330071A (en) | 1973-09-12 |
| DK129451B (en) | 1974-10-14 |
| DE2118996A1 (en) | 1971-11-11 |
| CS151091B2 (en) | 1973-09-17 |
| IE35071L (en) | 1971-10-24 |
| IL36652A (en) | 1974-07-31 |
| PL73563B1 (en) | 1974-10-30 |
| FR2092080A1 (en) | 1972-01-21 |
| BE766182A (en) | 1971-10-25 |
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