ES408415A1 - Procedimiento para la preparacion de nuevas tiazolo (5,4-d)pirimidinas. - Google Patents

Procedimiento para la preparacion de nuevas tiazolo (5,4-d)pirimidinas.

Info

Publication number: ES408415A1
Authority: ES; Spain
Prior art keywords: general formula; alcohol; hexahydro; radicals; radical
Prior art date: 1971-11-11
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES408415A

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Boehringer Ingelheim Pharma GmbH and Co KG

Original Assignee

Dr Karl Thomae GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-11-11

Filing date

1972-11-09

Publication date

1975-11-16

1971-11-11 Priority claimed from DE2155963A external-priority patent/DE2155963A1/de

1972-10-05 Priority claimed from DE19722248792 external-priority patent/DE2248792A1/de

1972-11-09 Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH

1975-11-16 Publication of ES408415A1 publication Critical patent/ES408415A1/es

Status Expired legal-status Critical Current

Links

-1 5,7-diamino-substituted thiazolo(5,4-d)pyrimidines Chemical class 0.000 title abstract 5
150000003839 salts Chemical class 0.000 title abstract 3
150000003254 radicals Chemical class 0.000 abstract 4
150000001875 compounds Chemical class 0.000 abstract 3
LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 2
GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 abstract 2
150000001412 amines Chemical class 0.000 abstract 2
125000001841 imino group Chemical group [H]N=* 0.000 abstract 2
238000000034 method Methods 0.000 abstract 2
150000007522 mineralic acids Chemical class 0.000 abstract 2
150000007524 organic acids Chemical class 0.000 abstract 2
OQFUNFPIPRUQAE-UHFFFAOYSA-N 1,4-thiazepane Chemical compound C1CNCCSC1 OQFUNFPIPRUQAE-UHFFFAOYSA-N 0.000 abstract 1
SLRMQYXOBQWXCR-UHFFFAOYSA-N 2154-56-5 Chemical compound [CH2]C1=CC=CC=C1 SLRMQYXOBQWXCR-UHFFFAOYSA-N 0.000 abstract 1
CDGFEINVQHEUQV-UHFFFAOYSA-N [1,3]thiazolo[5,4-d]pyrimidine Chemical compound N1=CN=C2SC=NC2=C1 CDGFEINVQHEUQV-UHFFFAOYSA-N 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
125000000472 sulfonyl group Chemical group *S(*)(=O)=O 0.000 abstract 1
BRNULMACUQOKMR-UHFFFAOYSA-N thiomorpholine Chemical compound C1CSCCN1 BRNULMACUQOKMR-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

ES408415A 1971-11-11 1972-11-09 Procedimiento para la preparacion de nuevas tiazolo (5,4-d)pirimidinas. Expired ES408415A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE2155963A DE2155963A1 (de)	1971-11-11	1971-11-11	Neue thiazolo eckige klammer auf 5,4-d eckige klammer zu pyrimidine
DE19722248792 DE2248792A1 (de)	1972-10-05	1972-10-05	Neue thiazolo eckige klammer auf 5,4-d eckige klammer zu pyrimidine

Publications (1)

Publication Number	Publication Date
ES408415A1 true ES408415A1 (es)	1975-11-16

Family

ID=25762007

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ES408415A Expired ES408415A1 (es)	1971-11-11	1972-11-09	Procedimiento para la preparacion de nuevas tiazolo (5,4-d)pirimidinas.

Country Status (4)

Country	Link
US (1)	US3850917A (es)
AT (1)	AT321295B (es)
BG (2)	BG20363A3 (es)
ES (1)	ES408415A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0101518B1 (en) *	1982-02-19	1986-03-12	Mochida Pharmaceutical Co., Ltd.	Thiazolopyrimidine derivative
US5057517A (en) *	1987-07-20	1991-10-15	Merck & Co., Inc.	Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents
US7129239B2 (en) *	2002-10-28	2006-10-31	Pfizer Inc.	Purine compounds and uses thereof
ATE510841T1 (de) *	2007-06-12	2011-06-15	Hoffmann La Roche	Thiazoliopyrimidine und ihre verwendung als hemmer der phosphatidylinositol-3 kinase
CN101932587A (zh) *	2007-09-24	2010-12-29	吉宁特有限公司	噻唑并嘧啶pi3k抑制剂化合物及使用方法
SG182247A1 (en) *	2009-05-27	2012-08-30	Hoffmann La Roche	Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
MX2011012520A (es)	2009-05-27	2011-12-12	Hoffmann La Roche	Compuestos inhibidores de pi3k de pirimidina biciclicos selectivos para p110 delta y metodos de uso de los mismos.

1972
- 1972-11-02 AT AT929972A patent/AT321295B/de not_active IP Right Cessation
- 1972-11-09 US US00305128A patent/US3850917A/en not_active Expired - Lifetime
- 1972-11-09 BG BG023403A patent/BG20363A3/xx unknown
- 1972-11-09 BG BG021813A patent/BG20108A3/xx unknown
- 1972-11-09 ES ES408415A patent/ES408415A1/es not_active Expired

Also Published As

Publication number	Publication date
BG20363A3 (bg)	1975-11-05
US3850917A (en)	1974-11-26
BG20108A3 (bg)	1975-10-30
AT321295B (de)	1975-03-25

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