ES457174A1 - Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas. - Google Patents

Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas.

Info

Publication number: ES457174A1
Authority: ES; Spain
Prior art keywords: cephalosporins; oxa; dethia; arylmalonamido; broad
Prior art date: 1976-03-25
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES457174A

Other languages

English (en)

Spanish (es)

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Shionogi and Co Ltd

Original Assignee

Shionogi and Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-03-25

Filing date

1977-03-24

Publication date

1978-08-16

1976-03-25 Priority claimed from JP3340176A external-priority patent/JPS52122386A/ja

1976-04-30 Priority claimed from JP5029576A external-priority patent/JPS52133997A/ja

1977-03-24 Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd

1978-08-16 Publication of ES457174A1 publication Critical patent/ES457174A1/es

Status Expired legal-status Critical Current

Links

229940124587 cephalosporin Drugs 0.000 title abstract 3
239000003242 anti bacterial agent Substances 0.000 title 1
-1 3-thienyl phenyl Chemical group 0.000 abstract 4
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
125000000175 2-thienyl group Chemical group S1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
241000894006 Bacteria Species 0.000 abstract 1
229930186147 Cephalosporin Natural products 0.000 abstract 1
241000589516 Pseudomonas Species 0.000 abstract 1
230000000844 anti-bacterial effect Effects 0.000 abstract 1
150000001780 cephalosporins Chemical class 0.000 abstract 1
125000005982 diphenylmethyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])(*)C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 abstract 1
WWYDYZMNFQIYPT-UHFFFAOYSA-N ru78191 Chemical compound OC(=O)C(C(O)=O)C1=CC=CC=C1 WWYDYZMNFQIYPT-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

ES457174A 1976-03-25 1977-03-24 Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas. Expired ES457174A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP3340176A JPS52122386A (en)	1976-03-25	1976-03-25	Cephalosporin analogous compounds as antibacterials
JP5029576A JPS52133997A (en)	1976-04-30	1976-04-30	Cephalosporin antibiotics

Publications (1)

Publication Number	Publication Date
ES457174A1 true ES457174A1 (es)	1978-08-16

Family

ID=26372085

Family Applications (5)

Application Number	Title	Priority Date	Filing Date
ES457174A Expired ES457174A1 (es)	1976-03-25	1977-03-24	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas.
ES469285A Expired ES469285A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas
ES469284A Expired ES469284A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas.
ES469286A Expired ES469286A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar sales de arilmalonamido-1- oxadestiacefalosporinas
ES469287A Expired ES469287A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas

Family Applications After (4)

Application Number	Title	Priority Date	Filing Date
ES469285A Expired ES469285A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas
ES469284A Expired ES469284A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas.
ES469286A Expired ES469286A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar sales de arilmalonamido-1- oxadestiacefalosporinas
ES469287A Expired ES469287A1 (es)	1976-03-25	1978-04-28	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas

Country Status (19)

Country	Link
AR (1)	AR224606A1 (fr)
BG (1)	BG31074A3 (fr)
CY (1)	CY1158A (fr)
DD (1)	DD129792A5 (fr)
DE (1)	DE2713370C2 (fr)
DK (1)	DK161331C (fr)
ES (5)	ES457174A1 (fr)
GR (1)	GR61146B (fr)
HK (1)	HK46882A (fr)
HU (1)	HU172720B (fr)
IE (1)	IE44794B1 (fr)
IL (1)	IL51743A (fr)
MX (1)	MX4348E (fr)
NO (2)	NO158505C (fr)
NZ (1)	NZ183687A (fr)
PT (1)	PT66346B (fr)
RO (2)	RO78228A (fr)
SE (1)	SE443143B (fr)
YU (2)	YU44039B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1557552A (en) *	1977-02-15	1979-12-12	Shionogi & Co	1 oxadethiacepham compounds
US4252953A (en) *	1979-05-01	1981-02-24	Eli Lilly And Company	Antibiotic crystalline epimer
JPS60123490A (ja) *	1983-12-07	1985-07-02	Shionogi & Co Ltd	マロニルオキサセフェムカルボン酸誘導体

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL178005C (nl) *	1972-11-06	1986-01-02	Merck & Co Inc	Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
US3962232A (en) *	1973-11-05	1976-06-08	Eli Lilly And Company	7-methoxycephalosporins
GB1449420A (en) *	1973-11-26	1976-09-15	Sankyo Co	7alpha-methoxycephalosporing derivatives

1977
- 1977-03-23 SE SE7703325A patent/SE443143B/xx not_active IP Right Cessation
- 1977-03-23 GR GR53086A patent/GR61146B/el unknown
- 1977-03-23 NO NO771023A patent/NO158505C/no unknown
- 1977-03-23 CY CY1158A patent/CY1158A/xx unknown
- 1977-03-24 ES ES457174A patent/ES457174A1/es not_active Expired
- 1977-03-24 IE IE622/77A patent/IE44794B1/en not_active IP Right Cessation
- 1977-03-24 PT PT66346A patent/PT66346B/pt unknown
- 1977-03-24 BG BG035796A patent/BG31074A3/xx unknown
- 1977-03-24 DD DD7700198053A patent/DD129792A5/xx unknown
- 1977-03-24 NZ NZ183687A patent/NZ183687A/xx unknown
- 1977-03-24 HU HU77SI00001565A patent/HU172720B/hu not_active IP Right Cessation
- 1977-03-24 DK DK131277A patent/DK161331C/da not_active IP Right Cessation
- 1977-03-24 RO RO7799076A patent/RO78228A/fr unknown
- 1977-03-24 RO RO7789781A patent/RO71742A/fr unknown
- 1977-03-25 IL IL51743A patent/IL51743A/xx unknown
- 1977-03-25 DE DE2713370A patent/DE2713370C2/de not_active Expired - Lifetime
- 1977-03-25 AR AR266992A patent/AR224606A1/es active
- 1977-03-25 MX MX775582U patent/MX4348E/es unknown
1978
- 1978-04-28 ES ES469285A patent/ES469285A1/es not_active Expired
- 1978-04-28 ES ES469284A patent/ES469284A1/es not_active Expired
- 1978-04-28 ES ES469286A patent/ES469286A1/es not_active Expired
- 1978-04-28 ES ES469287A patent/ES469287A1/es not_active Expired
1982
- 1982-11-11 HK HK468/82A patent/HK46882A/xx unknown
1983
- 1983-08-23 YU YU1738/83A patent/YU44039B/xx unknown
- 1983-08-23 YU YU1737/83A patent/YU44038B/xx unknown
1986
- 1986-05-28 NO NO862107A patent/NO862107L/no unknown

Also Published As

Publication number	Publication date
PT66346B (en)	1978-08-16
DE2713370C2 (de)	1994-04-21
CY1158A (en)	1983-01-28
BG31074A3 (en)	1981-10-15
HK46882A (en)	1982-11-19
ES469286A1 (es)	1979-09-16
NZ183687A (en)	1979-01-11
DD129792A5 (de)	1978-02-08
IE44794B1 (en)	1982-04-07
IE44794L (en)	1977-09-25
DK161331C (da)	1991-12-09
DE2713370A1 (de)	1977-09-29
YU173883A (en)	1983-12-31
YU44038B (en)	1990-02-28
DK161331B (da)	1991-06-24
DK131277A (da)	1977-09-26
NO862107L (no)	1977-09-27
GR61146B (en)	1978-09-27
HU172720B (hu)	1978-11-28
MX4348E (es)	1982-04-05
RO71742A (fr)	1982-02-26
ES469285A1 (es)	1979-09-16
RO78228A (fr)	1982-02-01
NO158505B (no)	1988-06-13
SE443143B (sv)	1986-02-17
PT66346A (en)	1977-04-01
YU44039B (en)	1990-02-28
AR224606A1 (es)	1981-12-30
ES469287A1 (es)	1979-09-16
SE7703325L (sv)	1977-09-26
ES469284A1 (es)	1978-11-16
NO158505C (no)	1988-09-21
NO771023L (no)	1977-09-27
YU173783A (en)	1983-12-31
IL51743A (en)	1980-10-26

Legal Events

Date	Code	Title	Description
1998-12-16	FD1A	Patent lapsed	Effective date: 19981103

Publication	Publication Date	Title
ES8106908A1 (es)	1981-09-01	Un procedimiento para la preparacion de (6r,7r)-7-((z)-2- (2-aminotiazol-4-il)-2-(2-carboxiprop-2-oxiimino)acetami- do)-3-(1-piridiniometil)cef-3-em-4-carboxilato pentahidrata-do
ES8704955A1 (es)	1987-04-16	Un proceso para la produccion de un compuesto de cefalospo- rina
ES8606361A1 (es)	1986-04-16	Un procedimiento para la preparacion de nuevos derivados de cefalosporina.
FR2509312B1 (fr)	1984-06-29
GR890100162A (en)	1990-01-19	7-(2-(s-amino1,2,4-thiadiazol-3yl)-2-(substituted-iminoacetamido)-3-(3-(quaternaryammonio)-1-propen-1-y)-3-cephem-4-carboxy-lates of the formula
IE782546L (en)	1979-06-24	Amino-thiazolyl cephalosporins
ES457174A1 (es)	1978-08-16	Un procedimiento para preparar arilmalonamido-1-oxadestiace-falosporinas.
ES403305A1 (es)	1975-05-01	Un procedimiento para producir nuevos compuestos de cefa- losporina.
MY8500128A (en)	1985-12-31	New cephalosporin derivatives, their production and use as antimicrobial agents
SE7810295L (sv)	1979-10-20	Substituerad kinolinkarboxylsyra
HK27784A (en)	1984-03-30	A solid cephalosporin salt
IE45559L (en)	1978-02-17	ß-LACTAM COMPOUNDS
ES8102590A1 (es)	1981-02-16	Metodo de producir antibioticos del tipo basado en streptomyces.
ES486023A1 (es)	1980-09-01	Un procedimiento para la preparacion de antibioticos de ce- falosporina
ES464008A1 (es)	1978-08-01	Un procedimiento para preparar nuevas beta-lactamas monoci- clicas con actividad antibacteriana.
ES8204436A1 (es)	1982-05-01	Un procedimiento para la preparacion de derivados del acido 2-b-clorometil-2&-metilpenam-3&-carboxilico.
ES8705431A1 (es)	1987-05-01	Un metodo para producir derivados de acido 2-(4-amino susti-tuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carbo-xilico
AU7357981A (en)	1982-02-04	Cephalosporins
GB1501643A (en)	1978-02-22	Antibacterial substituted azetidinones
ES8702428A1 (es)	1986-12-16	Un metodo para producir antibiotico tan-588 y-o n-desacetil-antibiotico tan-588
FR2301260A1 (fr)	1976-09-17	Nouveau procede de
TW371304B (en)	1999-10-01	Cephem compounds having antibacterial activity, their production and pharmaceutical composition
FR2361893A2 (fr)	1978-03-17	Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
IE772501L (en)	1978-06-11	Clavulanic acid ethers
ES8107309A1 (es)	1980-12-16	Un procedimiento de produccion de derivados de 7 -metoxice- falosporina