ES463871A1 - Procedimiento para la obtencion de lactamas - Google Patents
Procedimiento para la obtencion de lactamasInfo
- Publication number
- ES463871A1 ES463871A1 ES463871A ES463871A ES463871A1 ES 463871 A1 ES463871 A1 ES 463871A1 ES 463871 A ES463871 A ES 463871A ES 463871 A ES463871 A ES 463871A ES 463871 A1 ES463871 A1 ES 463871A1
- Authority
- ES
- Spain
- Prior art keywords
- opt
- alkyl
- substd
- halo
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 241000589516 Pseudomonas Species 0.000 title abstract 2
- 229940088710 antibiotic agent Drugs 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 229930186147 Cephalosporin Natural products 0.000 title 1
- 229930182555 Penicillin Natural products 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 229940124587 cephalosporin Drugs 0.000 title 1
- 150000001780 cephalosporins Chemical class 0.000 title 1
- 229940049954 penicillin Drugs 0.000 title 1
- -1 RO-phenyl Chemical group 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000001475 halogen functional group Chemical group 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- GRVDJDISBSALJP-UHFFFAOYSA-N methyloxidanyl Chemical compound [O]C GRVDJDISBSALJP-UHFFFAOYSA-N 0.000 abstract 2
- 125000000896 monocarboxylic acid group Chemical group 0.000 abstract 2
- 125000004299 tetrazol-5-yl group Chemical group [H]N1N=NC(*)=N1 0.000 abstract 2
- 125000001544 thienyl group Chemical group 0.000 abstract 2
- 125000001359 1,2,3-triazol-4-yl group Chemical group [H]N1N=NC([*])=C1[H] 0.000 abstract 1
- 125000004521 1,3,4-thiadiazol-2-yl group Chemical group S1C(=NN=C1)* 0.000 abstract 1
- 241000588722 Escherichia Species 0.000 abstract 1
- 241000588748 Klebsiella Species 0.000 abstract 1
- 125000003668 acetyloxy group Chemical group [H]C([H])([H])C(=O)O[*] 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 239000003782 beta lactam antibiotic agent Substances 0.000 abstract 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
- 125000002150 cyclohexa-1,4-dienyl group Chemical group [H]C1=C([H])C([H])(*)C([H])=C([H])C1([H])[H] 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- IPZJQDSFZGZEOY-UHFFFAOYSA-N dimethylmethylene Chemical compound C[C]C IPZJQDSFZGZEOY-UHFFFAOYSA-N 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000000654 isopropylidene group Chemical group C(C)(C)=* 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000002132 β-lactam antibiotic Substances 0.000 abstract 1
- 229940124586 β-lactam antibiotics Drugs 0.000 abstract 1
- 150000003952 β-lactams Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Abstract
Procedimiento para la obtención de lactamas, de fórmula general: **(Fórmula)** donde Z significa fenilo, RO-fenilo, ciclohexen-1-ilo, ciclohexa-1, 4-dienilo o tienilo, R y R1, en cada caso, significan H ó alquilo-(O)n-CO-, n representa O ó 1, R2 y R3, en cada caso, significan H, halógeno, NO2, NH2, alquilamino, dialquilamino o acilamino, ó juntos significan -CH=CH-CH=CH-, donde en el resto mencionado en último lugar también un grupo CH puede estar sustituido por N y/o un átomo de H por R4, o dos átomos de H por R4 y R5, R4 y R5, en cada caso, significan alquilo, alcoxi, dialquilamino ó halógeno o juntos -CH=CH- CH=CH-.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19772710979 DE2710979A1 (de) | 1977-03-14 | 1977-03-14 | Lactame, verfahren zu ihrer herstellung und diese verbindungen enthaltende mittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES463871A1 true ES463871A1 (es) | 1979-01-01 |
Family
ID=6003546
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES463871A Expired ES463871A1 (es) | 1977-03-14 | 1977-11-04 | Procedimiento para la obtencion de lactamas |
Country Status (7)
| Country | Link |
|---|---|
| AT (1) | ATA788777A (es) |
| DD (1) | DD134100A5 (es) |
| DE (1) | DE2710979A1 (es) |
| ES (1) | ES463871A1 (es) |
| GR (1) | GR63172B (es) |
| NZ (1) | NZ186671A (es) |
| PL (1) | PL205285A1 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2924948A1 (de) * | 1979-06-21 | 1981-01-22 | Thomae Gmbh Dr K | Neue cephalosporine, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| DE3134776A1 (de) * | 1981-09-02 | 1983-03-10 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue 6(alpha)-methoxy-penicilline, ihre salze, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| FR2874922A1 (fr) * | 2004-07-30 | 2006-03-10 | Palumed Sa | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
| FR2873695A1 (fr) * | 2004-07-30 | 2006-02-03 | Palumed Sa | Molecules hybrides qa ou q est une aminoquinoleine et a est un antibiotique ou un inhibiteur de resistance), leur synthese et leurs utilisations en tant qu'agent antibacterien |
| EP1771456A2 (fr) * | 2004-07-30 | 2007-04-11 | Palumed SA | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
-
1977
- 1977-03-14 DE DE19772710979 patent/DE2710979A1/de not_active Withdrawn
- 1977-11-04 AT AT788777A patent/ATA788777A/de not_active Application Discontinuation
- 1977-11-04 ES ES463871A patent/ES463871A1/es not_active Expired
-
1978
- 1978-03-10 DD DD20411478A patent/DD134100A5/xx unknown
- 1978-03-13 NZ NZ18667178A patent/NZ186671A/xx unknown
- 1978-03-13 PL PL20528578A patent/PL205285A1/xx unknown
- 1978-03-14 GR GR55703A patent/GR63172B/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GR63172B (en) | 1979-09-28 |
| DD134100A5 (de) | 1979-02-07 |
| ATA788777A (de) | 1980-11-15 |
| NZ186671A (en) | 1980-03-05 |
| DE2710979A1 (de) | 1978-09-21 |
| PL205285A1 (pl) | 1979-06-04 |
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