ES465152A1 - Procedimiento para la obtencion de derivados del acido %- (aminoacetil)fenoxiacetico. - Google Patents
Procedimiento para la obtencion de derivados del acido %- (aminoacetil)fenoxiacetico.Info
- Publication number
- ES465152A1 ES465152A1 ES465152A ES465152A ES465152A1 ES 465152 A1 ES465152 A1 ES 465152A1 ES 465152 A ES465152 A ES 465152A ES 465152 A ES465152 A ES 465152A ES 465152 A1 ES465152 A1 ES 465152A1
- Authority
- ES
- Spain
- Prior art keywords
- alpha
- ketone derivatives
- amino ketone
- formula
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/88—Unsaturated compounds containing keto groups containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Hematology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Procedimiento para la obtención de un compuesto de fórmula:***(Ver fórmula)en la que R es un radical hidroxi o metoxio una sal de adición de ácido del mismo farmacéuticamente aceptableo para un compuesto de fórmula I en la que R es un radical hidroxiuna sal de adición de base farmacéuticamente aceptable.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB48402/75A GB1559977A (en) | 1975-11-25 | 1975-11-25 | Amines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES465152A1 true ES465152A1 (es) | 1978-10-01 |
Family
ID=10448487
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES453632A Expired ES453632A1 (es) | 1975-11-25 | 1976-11-25 | Procedimiento para la obtencion de derivados del acido 4-(a-minoacetil) fenoxiacetico. |
| ES465152A Expired ES465152A1 (es) | 1975-11-25 | 1977-12-16 | Procedimiento para la obtencion de derivados del acido %- (aminoacetil)fenoxiacetico. |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES453632A Expired ES453632A1 (es) | 1975-11-25 | 1976-11-25 | Procedimiento para la obtencion de derivados del acido 4-(a-minoacetil) fenoxiacetico. |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US4105790A (es) |
| JP (2) | JPS5265240A (es) |
| AR (1) | AR215871A1 (es) |
| AT (1) | AT348993B (es) |
| AU (1) | AU503657B2 (es) |
| BE (1) | BE848707A (es) |
| CA (1) | CA1068695A (es) |
| CH (1) | CH624383A5 (es) |
| CS (1) | CS196333B2 (es) |
| DD (1) | DD127474A5 (es) |
| DE (1) | DE2653635C2 (es) |
| DK (1) | DK531276A (es) |
| ES (2) | ES453632A1 (es) |
| FI (1) | FI763399A7 (es) |
| FR (1) | FR2332747A1 (es) |
| GB (1) | GB1559977A (es) |
| IE (1) | IE44030B1 (es) |
| IL (1) | IL50904A (es) |
| IN (1) | IN145003B (es) |
| LU (1) | LU76251A1 (es) |
| NL (1) | NL7613081A (es) |
| NO (1) | NO764012L (es) |
| NZ (1) | NZ182581A (es) |
| PL (2) | PL105799B1 (es) |
| PT (1) | PT65892B (es) |
| SE (1) | SE7613079L (es) |
| SU (1) | SU722481A3 (es) |
| ZA (1) | ZA766696B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH028457U (es) * | 1988-07-01 | 1990-01-19 | ||
| JPH02130656U (es) * | 1989-03-31 | 1990-10-29 | ||
| US5348969A (en) * | 1992-04-03 | 1994-09-20 | Bristol-Myers Squibb Company | Diphenyloxazolyl-oxazoles as platelet aggregation inhibitors |
| JP3712208B2 (ja) * | 1993-06-25 | 2005-11-02 | メレルファーマスーティカルズ インコーポレイテッド | 抗ヒスタミン性の4−ジフェニルメチル/ジフェニルメトキシピペリジン誘導体類を製造する新規な中間体 |
| US6147216A (en) * | 1993-06-25 | 2000-11-14 | Merrell Pharmaceuticals Inc. | Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| US6683094B2 (en) | 1998-07-02 | 2004-01-27 | Aventis Pharmaceuticals Inc. | Antihistaminic piperidine derivatives and intermediates for the preparation thereof |
| US6700012B2 (en) | 1998-07-02 | 2004-03-02 | Aventis Pharmaceuticals Inc. | Antihistaminic piperidine derivatives and intermediates for the preparation thereof |
| FR2880887B1 (fr) * | 2005-01-14 | 2009-01-30 | Merck Sante Soc Par Actions Si | Derives d'hydroxyphenols, procedes pour leur preparation, compositions pharmaceutiques les contenant et applications en therapeutique |
| TW200740779A (en) | 2005-07-22 | 2007-11-01 | Mitsubishi Pharma Corp | Intermediate compound for synthesizing pharmaceutical agent and production method thereof |
| EP3170844A4 (en) * | 2014-07-16 | 2018-01-10 | Adeka Corporation | Photosensitive composition |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH543472A (fr) * | 1969-01-31 | 1973-10-31 | Orchimed Sa | Procédé pour la préparation d'acides phénoxyalcoyl-carboxyliques |
-
1975
- 1975-11-25 GB GB48402/75A patent/GB1559977A/en not_active Expired
-
1976
- 1976-11-08 IE IE2474/76A patent/IE44030B1/en unknown
- 1976-11-09 ZA ZA766696A patent/ZA766696B/xx unknown
- 1976-11-09 NZ NZ182581A patent/NZ182581A/xx unknown
- 1976-11-09 US US05/740,195 patent/US4105790A/en not_active Expired - Lifetime
- 1976-11-10 IN IN2024/CAL/76A patent/IN145003B/en unknown
- 1976-11-12 CA CA265,534A patent/CA1068695A/en not_active Expired
- 1976-11-14 IL IL50904A patent/IL50904A/xx unknown
- 1976-11-15 AU AU19625/76A patent/AU503657B2/en not_active Expired
- 1976-11-23 PL PL1976205925A patent/PL105799B1/pl unknown
- 1976-11-23 LU LU76251A patent/LU76251A1/xx unknown
- 1976-11-23 PL PL1976193861A patent/PL105491B1/pl unknown
- 1976-11-23 SE SE7613079A patent/SE7613079L/xx unknown
- 1976-11-24 DD DD195943A patent/DD127474A5/xx unknown
- 1976-11-24 FR FR7635385A patent/FR2332747A1/fr active Granted
- 1976-11-24 AT AT870976A patent/AT348993B/de not_active IP Right Cessation
- 1976-11-24 CH CH1480376A patent/CH624383A5/de not_active IP Right Cessation
- 1976-11-24 NL NL7613081A patent/NL7613081A/xx not_active Application Discontinuation
- 1976-11-24 CS CS767604A patent/CS196333B2/cs unknown
- 1976-11-24 NO NO764012A patent/NO764012L/no unknown
- 1976-11-24 BE BE172664A patent/BE848707A/xx not_active IP Right Cessation
- 1976-11-25 PT PT65892A patent/PT65892B/pt unknown
- 1976-11-25 AR AR265606A patent/AR215871A1/es active
- 1976-11-25 FI FI763399A patent/FI763399A7/fi not_active Application Discontinuation
- 1976-11-25 JP JP51141767A patent/JPS5265240A/ja active Granted
- 1976-11-25 ES ES453632A patent/ES453632A1/es not_active Expired
- 1976-11-25 DK DK531276A patent/DK531276A/da not_active Application Discontinuation
- 1976-11-25 DE DE2653635A patent/DE2653635C2/de not_active Expired
-
1977
- 1977-12-16 ES ES465152A patent/ES465152A1/es not_active Expired
-
1978
- 1978-02-13 SU SU782579897A patent/SU722481A3/ru active
-
1985
- 1985-11-08 JP JP60249137A patent/JPS61158922A/ja active Granted
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