ES513102A0 - "procedimiento para la preparacion de derivados de n-oxaciclil-alcohilpiperidina". - Google Patents
"procedimiento para la preparacion de derivados de n-oxaciclil-alcohilpiperidina".Info
- Publication number
- ES513102A0 ES513102A0 ES513102A ES513102A ES513102A0 ES 513102 A0 ES513102 A0 ES 513102A0 ES 513102 A ES513102 A ES 513102A ES 513102 A ES513102 A ES 513102A ES 513102 A0 ES513102 A0 ES 513102A0
- Authority
- ES
- Spain
- Prior art keywords
- oxaciclil
- alcohilpiperidina
- derivatives
- procedure
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19813124366 DE3124366A1 (de) | 1981-06-20 | 1981-06-20 | N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8304974A1 ES8304974A1 (es) | 1983-03-16 |
| ES513102A0 true ES513102A0 (es) | 1983-03-16 |
Family
ID=6135055
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES513102A Granted ES513102A0 (es) | 1981-06-20 | 1982-06-15 | "procedimiento para la preparacion de derivados de n-oxaciclil-alcohilpiperidina". |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US4470989A (de) |
| EP (1) | EP0068261B1 (de) |
| JP (1) | JPS58977A (de) |
| KR (1) | KR840000540A (de) |
| AT (1) | ATE12498T1 (de) |
| AU (1) | AU551182B2 (de) |
| CA (1) | CA1175432A (de) |
| DE (2) | DE3124366A1 (de) |
| DK (1) | DK275782A (de) |
| ES (1) | ES513102A0 (de) |
| FI (1) | FI822178L (de) |
| GR (1) | GR76502B (de) |
| HU (1) | HU190989B (de) |
| IE (1) | IE53127B1 (de) |
| IL (1) | IL66084A (de) |
| NO (1) | NO822041L (de) |
| NZ (1) | NZ201006A (de) |
| PH (1) | PH18536A (de) |
| PT (1) | PT75070B (de) |
| ZA (1) | ZA824328B (de) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3366460D1 (en) * | 1982-08-05 | 1986-10-30 | Toshiba Kk | Color picture tube and method for manufacturing the same |
| US5312840A (en) * | 1986-07-10 | 1994-05-17 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education | Substituted guanidines having high binding to the sigma receptor and the use thereof |
| US5221745A (en) * | 1991-06-21 | 1993-06-22 | American Home Products Corp. | Psychotropic piperidinylmethyl benzodioxans |
| US5182292A (en) * | 1991-06-21 | 1993-01-26 | American Home Products Corporation | Psychotropic piperidinylmethyl benzodioxans |
| US5212170A (en) * | 1991-06-21 | 1993-05-18 | American Home Products Corporation | Psychotropic piperidinylmethyl benzodioxans |
| DE4140540A1 (de) * | 1991-12-09 | 1993-06-17 | Bayer Ag | Neue azaheterocyclylmethyl-chromane |
| US6096763A (en) * | 1995-02-23 | 2000-08-01 | Merck & Co., Inc. | α1a adrenergic receptor antagonists |
| GB9603457D0 (de) * | 1996-02-19 | 1996-04-17 | Merck & Co Inc | |
| US5952351A (en) * | 1995-02-23 | 1999-09-14 | Merck & Co., Inc. | Alpha 1a adrenergic receptor antagonists |
| US6025355A (en) * | 1997-05-19 | 2000-02-15 | Cambridge Neuroscience, Inc. | Pharmaceutically active compounds and methods of use |
| US6242198B1 (en) | 1996-07-25 | 2001-06-05 | Cambridge Neuroscience, Inc. | Methods of treatment of eye trauma and disorders |
| US6756389B2 (en) | 1996-08-09 | 2004-06-29 | Cambridge Neuroscience, Inc. | Pharmaceutically active compounds and methods of use |
| EE04780B1 (et) | 1999-06-02 | 2007-02-15 | Janssen Pharmaceutica N.V. | Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod |
| SK286159B6 (sk) | 1999-06-02 | 2008-04-07 | Janssen Pharmaceutica N. V. | Benzodioxánový, benzofuránový alebo benzopyránovýderivát, spôsob jeho prípravy, tento derivát na použitie ako liečivo, farmaceutická kompozícia obsahujúca tento derivát a spôsob jej prípravy |
| JO2654B1 (en) * | 2000-09-04 | 2012-06-17 | شركة جانسين فارماسوتيكا ان. في | Multiple aryl caroxa amides are useful as lipid - lowering agents |
| JO2409B1 (en) * | 2000-11-21 | 2007-06-17 | شركة جانسين فارماسوتيكا ان. في | Second-phenyl carboxy amides are useful as lipid-lowering agents |
| CA2465328C (en) * | 2001-11-01 | 2011-06-14 | Michael Francis Gross | Piperidines |
| WO2007036718A2 (en) | 2005-09-30 | 2007-04-05 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
| US8283364B2 (en) | 2005-09-30 | 2012-10-09 | Glaxo Group Limited | Compounds which have activity at M1 receptor and their uses in medicine |
| WO2007036711A1 (en) | 2005-09-30 | 2007-04-05 | Glaxo Group Limited | BENZIMIDAZOLONES WHICH HAVE ACTIVITY AT Ml RECEPTOR |
| GB0605784D0 (en) * | 2006-03-22 | 2006-05-03 | Glaxo Group Ltd | Compounds |
| WO2009037294A1 (en) | 2007-09-20 | 2009-03-26 | Glaxo Group Limited | Compounds which have activity at m1 receptor and their uses in medicine |
| GB0718415D0 (en) | 2007-09-20 | 2007-10-31 | Glaxo Group Ltd | Compounds |
| CN108358832A (zh) * | 2017-12-29 | 2018-08-03 | 上海艾康睿医药科技有限公司 | 一种合成4-[(2-氨基-4-氯)苯基]-氨基-n-哌啶甲酸乙酯的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3910930A (en) * | 1973-01-04 | 1975-10-07 | Janssen Pharmaceutica Nv | 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones |
| US4066772A (en) * | 1975-07-21 | 1978-01-03 | Janssen Pharmaceutica N.V. | 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds |
| GR71865B (de) * | 1978-03-20 | 1983-07-07 | Ciba Geigy | |
| US4181802A (en) * | 1978-05-11 | 1980-01-01 | Janssen Pharmaceutica N.V. | 1-(Heterocyclylalkyl)-1,3-dihydro-2-H-benzimidazole-2-ones |
| US4329348A (en) * | 1979-02-26 | 1982-05-11 | Ciba-Geigy Corporation | N-Oxacyclic-alkylpiperidines as psychostimulants |
-
1981
- 1981-06-20 DE DE19813124366 patent/DE3124366A1/de not_active Withdrawn
-
1982
- 1982-06-14 DE DE8282105174T patent/DE3262861D1/de not_active Expired
- 1982-06-14 AT AT82105174T patent/ATE12498T1/de active
- 1982-06-14 EP EP82105174A patent/EP0068261B1/de not_active Expired
- 1982-06-15 ES ES513102A patent/ES513102A0/es active Granted
- 1982-06-17 FI FI822178A patent/FI822178L/fi not_active Application Discontinuation
- 1982-06-17 PT PT75070A patent/PT75070B/de unknown
- 1982-06-18 PH PH27449A patent/PH18536A/en unknown
- 1982-06-18 HU HU821992A patent/HU190989B/hu unknown
- 1982-06-18 NZ NZ201006A patent/NZ201006A/en unknown
- 1982-06-18 CA CA000405525A patent/CA1175432A/en not_active Expired
- 1982-06-18 GR GR68474A patent/GR76502B/el unknown
- 1982-06-18 KR KR1019820002715A patent/KR840000540A/ko not_active Withdrawn
- 1982-06-18 DK DK275782A patent/DK275782A/da not_active Application Discontinuation
- 1982-06-18 US US06/389,677 patent/US4470989A/en not_active Expired - Fee Related
- 1982-06-18 NO NO822041A patent/NO822041L/no unknown
- 1982-06-18 IE IE1448/82A patent/IE53127B1/en unknown
- 1982-06-18 AU AU84992/82A patent/AU551182B2/en not_active Ceased
- 1982-06-18 JP JP57104048A patent/JPS58977A/ja active Pending
- 1982-06-18 IL IL66084A patent/IL66084A/xx unknown
- 1982-06-18 ZA ZA824328A patent/ZA824328B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES8304974A1 (es) | 1983-03-16 |
| IL66084A (en) | 1986-07-31 |
| PH18536A (en) | 1985-08-09 |
| CA1175432A (en) | 1984-10-02 |
| FI822178A0 (fi) | 1982-06-17 |
| IE53127B1 (en) | 1988-07-06 |
| HU190989B (en) | 1986-12-28 |
| JPS58977A (ja) | 1983-01-06 |
| DK275782A (da) | 1982-12-21 |
| AU8499282A (en) | 1983-01-06 |
| IL66084A0 (en) | 1982-09-30 |
| GR76502B (de) | 1984-08-10 |
| DE3262861D1 (en) | 1985-05-09 |
| ATE12498T1 (de) | 1985-04-15 |
| EP0068261A1 (de) | 1983-01-05 |
| DE3124366A1 (de) | 1982-12-30 |
| PT75070B (de) | 1985-01-07 |
| FI822178A7 (fi) | 1982-12-21 |
| PT75070A (de) | 1982-07-01 |
| AU551182B2 (en) | 1986-04-17 |
| KR840000540A (ko) | 1984-02-25 |
| NO822041L (no) | 1982-12-21 |
| ZA824328B (en) | 1983-04-27 |
| IE821448L (en) | 1982-12-20 |
| EP0068261B1 (de) | 1985-04-03 |
| NZ201006A (en) | 1985-12-13 |
| FI822178L (fi) | 1982-12-21 |
| US4470989A (en) | 1984-09-11 |
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