ES529349A0 - Un procedimiento para la preparacion de derivados de acilmorfinano - Google Patents
Un procedimiento para la preparacion de derivados de acilmorfinanoInfo
- Publication number
- ES529349A0 ES529349A0 ES529349A ES529349A ES529349A0 ES 529349 A0 ES529349 A0 ES 529349A0 ES 529349 A ES529349 A ES 529349A ES 529349 A ES529349 A ES 529349A ES 529349 A0 ES529349 A0 ES 529349A0
- Authority
- ES
- Spain
- Prior art keywords
- acilmorfinan
- derivatives
- procedure
- preparation
- acilmorfinan derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
- C07D221/28—Morphinans
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/319,482 US4374139A (en) | 1981-11-09 | 1981-11-09 | Levorotatory N-substituted acylmorphinans useful as analgesic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8506635A1 ES8506635A1 (es) | 1985-08-01 |
| ES529349A0 true ES529349A0 (es) | 1985-08-01 |
Family
ID=23242421
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES517222A Granted ES517222A0 (es) | 1981-11-09 | 1982-11-08 | Un procedimiento para la preparacion de derivados de acilmorrfinano. |
| ES529349A Granted ES529349A0 (es) | 1981-11-09 | 1984-02-01 | Un procedimiento para la preparacion de derivados de acilmorfinano |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES517222A Granted ES517222A0 (es) | 1981-11-09 | 1982-11-08 | Un procedimiento para la preparacion de derivados de acilmorrfinano. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4374139A (es) |
| EP (1) | EP0079556A3 (es) |
| JP (1) | JPS5888364A (es) |
| KR (1) | KR840002357A (es) |
| AU (1) | AU9027682A (es) |
| CA (1) | CA1195324A (es) |
| DK (1) | DK491582A (es) |
| ES (2) | ES517222A0 (es) |
| FI (1) | FI823824L (es) |
| GR (1) | GR78317B (es) |
| HU (1) | HU187425B (es) |
| IL (1) | IL67180A0 (es) |
| MC (1) | MC1490A1 (es) |
| NO (1) | NO823707L (es) |
| NZ (1) | NZ202404A (es) |
| PH (1) | PH18458A (es) |
| PT (1) | PT75815B (es) |
| ZA (1) | ZA827905B (es) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4423221A (en) * | 1982-06-10 | 1983-12-27 | Sisa Pharmaceutical Laboratories, Inc. | 7-Carboethoxy-morphinan-6-one compounds |
| US4454141A (en) * | 1982-09-23 | 1984-06-12 | Sisa Pharmaceutical Laboratories, Inc. | Trans-B/C-7-(1-hydroxypentyl)-3-methoxy-17 methyl-6,7-didehydromorphinans, and methods of relieving pain with them |
| EP0184041A1 (en) * | 1984-11-13 | 1986-06-11 | Miles Inc. | 6-Methylene morphinan purification technique |
| US4929622A (en) * | 1987-09-24 | 1990-05-29 | Hoechst-Roussel Pharmaceuticals, Inc. | 2,6-Methanopyrrolo-3-benzazocines |
| DE4304450A1 (de) * | 1993-02-13 | 1994-08-18 | Boehringer Mannheim Gmbh | System zur Zubereitung von Flüssigkeiten |
| AU2002227135B2 (en) * | 2000-10-31 | 2008-01-03 | Rensselaer Polytechnic Institute | 8- substituted-2, 6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents |
| JP4202250B2 (ja) | 2001-07-25 | 2008-12-24 | バイオマリン ファーマシューティカル インコーポレイテッド | 血液脳関門輸送を調節するための組成物および方法 |
| US20040204862A1 (en) * | 2003-04-11 | 2004-10-14 | Wainer Irving W. | Computer-based model for identification and characterization for non-competitive inhibitors of nicotinic acetylcholine receptors and related ligand-gated ion channel receptors |
| EP2671507A3 (en) | 2005-04-28 | 2014-02-19 | Proteus Digital Health, Inc. | Pharma-informatics system |
| MX2009002893A (es) | 2006-09-18 | 2009-07-10 | Raptor Pharmaceutical Inc | Tratamiento de trastornos hepaticos mediante la administracion de conjugados de la proteina asociada al receptor (rap). |
| CA2752373C (en) | 2009-02-20 | 2017-10-10 | To-Bbb Holding B.V. | Glutathione-based drug delivery system |
| IL255113B (en) | 2009-05-06 | 2022-09-01 | Laboratory Skin Care Inc | Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same |
| TR201908514T4 (tr) | 2009-12-04 | 2019-07-22 | Alkermes Pharma Ireland Ltd | İlaç doz aşimi tedavi̇si̇ i̇çi̇n morfi̇nan türevleri̇ |
| US8436175B2 (en) | 2010-03-22 | 2013-05-07 | Rensselaer Polytechnic Institute | Carboxamide bioisosteres of opiates |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
| WO2013003720A1 (en) | 2011-06-29 | 2013-01-03 | Alkermes, Inc. | Peripherally acting opioid compounds |
| US9211293B2 (en) | 2011-12-15 | 2015-12-15 | Alkermes Pharma Ireland Limited | Opioid agonist antagonist combinations |
| ES2770978T3 (es) | 2013-05-24 | 2020-07-06 | Alkermes Pharma Ireland Ltd | Análogos de morfanos y morfinanos y métodos de uso |
| EP3003311A2 (en) | 2013-05-24 | 2016-04-13 | Alkermes Pharma Ireland Limited | Methods for treating depressive symptoms |
| WO2018125716A1 (en) | 2017-01-02 | 2018-07-05 | Purdue Pharma L.P. | Morphinan derivatives and use thereof |
| EP4243768A1 (en) | 2020-11-12 | 2023-09-20 | Alkermes Pharma Ireland Limited | Immediate release multilayer tablet |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3723437A (en) * | 1970-09-15 | 1973-03-27 | American Home Prod | 4,10-(methaniminomethano phenanthrene derivatives |
| ZA73988B (en) * | 1972-03-10 | 1973-10-31 | Hoffmann La Roche | Morphinan derivatives |
| US3914233A (en) * | 1972-10-20 | 1975-10-21 | Hoffmann La Roche | 4-Hydroxy-N-substituted morphinan derivatives |
-
1981
- 1981-11-09 US US06/319,482 patent/US4374139A/en not_active Expired - Fee Related
- 1981-12-29 GR GR69729A patent/GR78317B/el unknown
-
1982
- 1982-10-28 ZA ZA827905A patent/ZA827905B/xx unknown
- 1982-11-05 NZ NZ202404A patent/NZ202404A/en unknown
- 1982-11-05 DK DK491582A patent/DK491582A/da not_active Application Discontinuation
- 1982-11-05 IL IL67180A patent/IL67180A0/xx unknown
- 1982-11-08 HU HU823578A patent/HU187425B/hu unknown
- 1982-11-08 FI FI823824A patent/FI823824L/fi not_active Application Discontinuation
- 1982-11-08 MC MC821609A patent/MC1490A1/fr unknown
- 1982-11-08 ES ES517222A patent/ES517222A0/es active Granted
- 1982-11-08 EP EP82110285A patent/EP0079556A3/de not_active Ceased
- 1982-11-08 NO NO823707A patent/NO823707L/no unknown
- 1982-11-08 CA CA000415102A patent/CA1195324A/en not_active Expired
- 1982-11-08 PH PH28105A patent/PH18458A/en unknown
- 1982-11-08 PT PT75815A patent/PT75815B/pt unknown
- 1982-11-08 JP JP57194799A patent/JPS5888364A/ja active Pending
- 1982-11-09 KR KR1019820005066A patent/KR840002357A/ko not_active Withdrawn
- 1982-11-09 AU AU90276/82A patent/AU9027682A/en not_active Abandoned
-
1984
- 1984-02-01 ES ES529349A patent/ES529349A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| MC1490A1 (fr) | 1983-09-12 |
| KR840002357A (ko) | 1984-06-25 |
| PT75815A (en) | 1982-12-01 |
| GR78317B (es) | 1984-09-26 |
| EP0079556A3 (de) | 1983-08-24 |
| US4374139A (en) | 1983-02-15 |
| NZ202404A (en) | 1985-11-08 |
| DK491582A (da) | 1983-05-10 |
| JPS5888364A (ja) | 1983-05-26 |
| FI823824A0 (fi) | 1982-11-08 |
| PH18458A (en) | 1985-07-18 |
| ES8506635A1 (es) | 1985-08-01 |
| HU187425B (en) | 1986-01-28 |
| CA1195324A (en) | 1985-10-15 |
| ES8500948A1 (es) | 1984-12-01 |
| ES517222A0 (es) | 1984-12-01 |
| ZA827905B (en) | 1983-08-31 |
| FI823824A7 (fi) | 1983-05-10 |
| EP0079556A2 (de) | 1983-05-25 |
| IL67180A0 (en) | 1983-03-31 |
| PT75815B (en) | 1986-01-21 |
| FI823824L (fi) | 1983-05-10 |
| NO823707L (no) | 1983-05-10 |
| AU9027682A (en) | 1983-05-19 |
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