ES557045A0 - Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas - Google Patents

Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Info

Publication number
ES557045A0
ES557045A0 ES557045A ES557045A ES557045A0 ES 557045 A0 ES557045 A0 ES 557045A0 ES 557045 A ES557045 A ES 557045A ES 557045 A ES557045 A ES 557045A ES 557045 A0 ES557045 A0 ES 557045A0
Authority
ES
Spain
Prior art keywords
arylmethanones
oxadiazol
preparing
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES557045A
Other languages
English (en)
Other versions
ES8800917A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Hoechst Roussel Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharmaceuticals Inc filed Critical Hoechst Roussel Pharmaceuticals Inc
Publication of ES8800917A1 publication Critical patent/ES8800917A1/es
Publication of ES557045A0 publication Critical patent/ES557045A0/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
ES557045A 1985-01-22 1986-09-01 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas Expired ES8800917A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/693,509 US4562186A (en) 1985-01-22 1985-01-22 (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use

Publications (2)

Publication Number Publication Date
ES8800917A1 ES8800917A1 (es) 1987-12-01
ES557045A0 true ES557045A0 (es) 1987-12-01

Family

ID=24784962

Family Applications (2)

Application Number Title Priority Date Filing Date
ES551041A Expired ES8705868A1 (es) 1985-01-22 1986-01-20 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas
ES557045A Expired ES8800917A1 (es) 1985-01-22 1986-09-01 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES551041A Expired ES8705868A1 (es) 1985-01-22 1986-01-20 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Country Status (8)

Country Link
US (1) US4562186A (es)
EP (1) EP0189080A3 (es)
JP (1) JPS61167674A (es)
DK (1) DK30186A (es)
ES (2) ES8705868A1 (es)
GR (1) GR860142B (es)
IE (1) IE860177L (es)
PT (1) PT81880B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4562186A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use
US7576220B2 (en) * 2006-04-06 2009-08-18 Rikkyo Gakuin Method of producing 1,2,4-oxadiazole derivatives
CN113195461A (zh) * 2018-10-01 2021-07-30 Pi工业有限公司 新型恶二唑类化合物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL256329A (es) * 1959-09-29
BE738276A (en) * 1968-09-01 1970-02-16 Prepn of 3-acyl-1,2,4-oxadiazoles useful in syn - of medicaments, in plant protection and as inter
GB1227978A (es) * 1968-09-13 1971-04-15
FR2053742A5 (en) * 1969-07-16 1971-04-16 Berlin Chemie Veb Prepn of 3-acyl-1,2,4-oxadiazoles useful in syn - of medicaments, in plant protection and as inter
IL42363A0 (en) * 1972-07-04 1973-07-30 Lepetit Spa 1,2,4-oxadiazole derivatives
US4160829A (en) * 1972-12-22 1979-07-10 Gist-Brocades N.V. Antibacterial 1,2,4-oxadiazolylacetamido cephalosporins
JPS58150576A (ja) * 1982-03-03 1983-09-07 Sumitomo Chem Co Ltd 新規な1,2,4−オキサジアゾ−ル誘導体
US4562186A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use
US4562187A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (Isoxazol-3-yl)arylmethanones, compositions and pharmaceutical use

Also Published As

Publication number Publication date
EP0189080A2 (en) 1986-07-30
ES8705868A1 (es) 1987-05-16
GR860142B (en) 1986-05-16
ES8800917A1 (es) 1987-12-01
EP0189080A3 (en) 1987-07-15
DK30186A (da) 1986-07-23
PT81880B (en) 1987-11-12
ES551041A0 (es) 1987-05-16
IE860177L (en) 1986-07-22
DK30186D0 (da) 1986-01-21
JPS61167674A (ja) 1986-07-29
US4562186A (en) 1985-12-31
PT81880A (en) 1986-02-01

Similar Documents

Publication Publication Date Title
ES548135A0 (es) Un procedimiento para preparar dioxafosforinanos
ES553989A0 (es) Procedimiento para preparar 2,2,6,6-tetraalquil-4-piperidilaminas
ES551517A0 (es) Un procedimiento para preparar aril-hidroxamatos
ES549713A0 (es) Un procedimiento para preparar 1,4-dihidropiridinas
ES543929A0 (es) Un procedimiento para preparar un p-isononanoiloxibenceno- sulfonato
ES549860A0 (es) Un procedimiento para preparar aminoacil-ladanos
AR231308A1 (es) Un procedimiento para preparar 1-be-d-ribofuranosil-1,2,4-triazolcarboxamida rivavirina
ES552032A0 (es) Un procedimiento para preparar derivados de 1,8-naftiridina
ES546157A0 (es) Un procedimiento para preparar quinolonas
ES542149A0 (es) Un procedimiento para preparar hidroxi-4-2h-1-benzotiopiran-2-onas
ES557659A0 (es) Un procedimiento para preparar derivados de ciclopentil-eter.
ES544864A0 (es) Un procedimiento para preparar 4-acetoxi-3-hidroxietilazeti-zin-2-ona
ES549472A0 (es) Un procedimiento para preparar 1-beta-d-ribofuranosil-1,2,4-triazol-3-carboxamida.
ES552772A0 (es) Un procedimiento para producir 2,3,4-tri-o-acil-d- y-o l-hexosas
ES552138A0 (es) Un procedimiento para preparar poliarilen-polieteres
ES557056A0 (es) Un procedimiento para preparar el compuesto 3(s)-3-amino-2-oxo-4,4-dimetil-1-azetidinilsulfato
ES544381A0 (es) Un procedimiento para preparar 5-desoxi-l-arabinosa
AR241134A1 (es) Un procedimiento para preparar w-lactamas
ES557568A0 (es) Un procedimiento para preparar etil-alfa-(1-carboxi-etil)-ami-no-gamma-fenilbutirato
ES552724A0 (es) Un procedimiento para preparar nuevos compuestos de 2-oxa-0 aza-pregnano.
ES551361A0 (es) Un metodo para preparar 6-cloro-2-metil-1h-2,3,4,5-tetrahidro-3-benzazepen-n-oxido.
ES540589A0 (es) Un procedimiento para preparar 2-arilimidazo (4,5-c) piridi-nas.
ES557045A0 (es) Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas
ES554201A0 (es) Un procedimiento para preparar etanobenzazepinas
ES557636A0 (es) Un procedimiento para preparar derivados de 3-amino-4-oxo-2,3,4,5-benzoxapina