ES557261A1 - Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos - Google Patents

Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos

Info

Publication number
ES557261A1
ES557261A1 ES557261A ES557261A ES557261A1 ES 557261 A1 ES557261 A1 ES 557261A1 ES 557261 A ES557261 A ES 557261A ES 557261 A ES557261 A ES 557261A ES 557261 A1 ES557261 A1 ES 557261A1
Authority
ES
Spain
Prior art keywords
formula
group
azacycloalkenes
azacycloalkanes
trisubstituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES557261A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES557261A1 publication Critical patent/ES557261A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • G—PHYSICS
    • G05—CONTROLLING; REGULATING
    • G05B—CONTROL OR REGULATING SYSTEMS IN GENERAL; FUNCTIONAL ELEMENTS OF SUCH SYSTEMS; MONITORING OR TESTING ARRANGEMENTS FOR SUCH SYSTEMS OR ELEMENTS
    • G05B2219/00—Program-control systems
    • G05B2219/30—Nc systems
    • G05B2219/35—Nc in input of data, input till input file format
    • G05B2219/35287—Verify, check program by drawing, display part, testpiece

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Azacicloalcanos ó bien azacicloalquenos 1,3,4-trisustituidos de la formula**formula** en la que R significa un resto 3-indol, en caso dado sustituido, alk significa alquileno inferior, que separa el resto R del átomo de hidrógeno por 1 a 3 átomos de carbono, R1 significa carboxi en cado dado esterificado ó amidado y R2 significa un grupo hidroxi en cado dado eterificado ó acilado ó un grupo amino en caso dado acilado, y sus tautómeros y/ó sales, tienen efecto nootrópico y pueden encontrar aplicación como nootrópicos. Se obtienen por ejemplo, porque en un compuesto de la fórmula **formula** en la que X4 significa un resto transformable en un grupo R2, se transforma X4 en un grupo R2
ES557261A 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos Expired ES557261A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1385 1985-01-03
CH305385 1985-07-15

Publications (1)

Publication Number Publication Date
ES557261A1 true ES557261A1 (es) 1987-10-01

Family

ID=25683258

Family Applications (5)

Application Number Title Priority Date Filing Date
ES550634A Expired ES8704896A1 (es) 1985-01-03 1986-01-02 Procedimiento para la obtencion de azacicloalcanos y azaci- cloalquenos 1,3,4-trisustituidos
ES557260A Expired ES557260A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos
ES557262A Expired ES557262A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos
ES557263A Expired ES557263A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de alanincompuestos n-sustituidos
ES557261A Expired ES557261A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos

Family Applications Before (4)

Application Number Title Priority Date Filing Date
ES550634A Expired ES8704896A1 (es) 1985-01-03 1986-01-02 Procedimiento para la obtencion de azacicloalcanos y azaci- cloalquenos 1,3,4-trisustituidos
ES557260A Expired ES557260A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos
ES557262A Expired ES557262A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de azacicloalcanos y azacicloalquenos 1,3,4-trisustituidos
ES557263A Expired ES557263A1 (es) 1985-01-03 1986-12-16 Procedimiento para la obtencion de alanincompuestos n-sustituidos

Country Status (10)

Country Link
EP (1) EP0187122A3 (es)
KR (1) KR870006037A (es)
AU (1) AU5178486A (es)
DK (1) DK786A (es)
ES (5) ES8704896A1 (es)
FI (1) FI855183A7 (es)
GR (1) GR860004B (es)
HU (1) HUT40108A (es)
NO (1) NO860007L (es)
PT (1) PT81780B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2249548B (en) * 1988-06-03 1992-10-14 Wyeth John & Brother Ltd Aralkyl amine intermediates
GB8813185D0 (en) * 1988-06-03 1988-07-06 Wyeth John & Brother Ltd New method & amines used therein
EP1831165A1 (en) * 2004-12-20 2007-09-12 F. Hoffmann-Roche AG 4-aminopiperidine derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3075986A (en) * 1958-01-09 1963-01-29 Rhone Poulenc Sa (1-piperdidylalkyl) derivatives of 3-indole
US3183235A (en) * 1961-06-27 1965-05-11 Sterling Drug Inc 1-[3-, 2-, and 1-indolyl-lower-alkanoyl] piperidines
US3238215A (en) * 1963-10-17 1966-03-01 Sterling Drug Inc 1-[(3-, 2-, and 1-indolyl)-lower-alkyl-, lower-alkenyl-, and lower-alkynyl]piperidines
US3821387A (en) * 1965-10-23 1974-06-28 Robins Co Inc A H The treatment of parkinsonism with 3-(omega-substituted alkyl)-indoles
GB1189064A (en) * 1967-05-01 1970-04-22 Sterling Drug Inc Indole Derivatives
DE3233553A1 (de) * 1982-09-10 1984-03-15 Merck Patent Gmbh, 6100 Darmstadt Pyrrolderivate
DE3342632A1 (de) * 1983-11-25 1985-06-05 Merck Patent Gmbh, 6100 Darmstadt Indolderivate

Also Published As

Publication number Publication date
AU5178486A (en) 1986-07-10
ES557262A1 (es) 1987-10-01
FI855183A0 (fi) 1985-12-30
DK786A (da) 1986-07-04
PT81780A (de) 1986-02-01
ES8704896A1 (es) 1987-04-16
EP0187122A3 (de) 1987-12-16
ES557263A1 (es) 1987-10-01
ES557260A1 (es) 1987-10-01
FI855183A7 (fi) 1986-07-04
NO860007L (no) 1986-07-04
DK786D0 (da) 1986-01-02
EP0187122A2 (de) 1986-07-09
GR860004B (en) 1986-04-25
PT81780B (de) 1987-11-05
ES550634A0 (es) 1987-04-16
KR870006037A (ko) 1987-07-08
HUT40108A (en) 1986-11-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19881116