ES8201550A1 - Procedimiento para la preparacion de 4-(4-alquil-4-aroil-1- piperidino) butirofenona - Google Patents
Procedimiento para la preparacion de 4-(4-alquil-4-aroil-1- piperidino) butirofenonaInfo
- Publication number
- ES8201550A1 ES8201550A1 ES496204A ES496204A ES8201550A1 ES 8201550 A1 ES8201550 A1 ES 8201550A1 ES 496204 A ES496204 A ES 496204A ES 496204 A ES496204 A ES 496204A ES 8201550 A1 ES8201550 A1 ES 8201550A1
- Authority
- ES
- Spain
- Prior art keywords
- alkyl
- oxo
- compounds
- butyrophenones
- aroyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 230000000561 anti-psychotic effect Effects 0.000 abstract 1
- -1 aryl Grignard reagents Chemical class 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8894279A | 1979-10-27 | 1979-10-27 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES496204A0 ES496204A0 (es) | 1981-12-01 |
| ES8201550A1 true ES8201550A1 (es) | 1981-12-01 |
Family
ID=22214421
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES496204A Expired ES8201550A1 (es) | 1979-10-27 | 1980-10-23 | Procedimiento para la preparacion de 4-(4-alquil-4-aroil-1- piperidino) butirofenona |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS5673061A (fr) |
| AU (1) | AU6369480A (fr) |
| BE (1) | BE885894A (fr) |
| CA (1) | CA1148162A (fr) |
| DE (1) | DE3039974A1 (fr) |
| ES (1) | ES8201550A1 (fr) |
| FR (1) | FR2468592A1 (fr) |
| GB (1) | GB2061937A (fr) |
| IL (1) | IL61340A0 (fr) |
| IT (1) | IT1146198B (fr) |
| NL (1) | NL8005890A (fr) |
| ZA (1) | ZA806501B (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| USD473103S1 (en) | 2001-07-25 | 2003-04-15 | Calico Brands, Inc. | Utility lighter |
| PT2354124E (pt) * | 2006-12-19 | 2013-04-09 | Hoffmann La Roche | Derivados de heteroaril-pirrolidinilo e piperidinil-cetona |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE713746C (de) * | 1939-03-31 | 1941-11-18 | I G Farbenindustrie Akt Ges | Verfahren zur Darstellung von 4-Arylpiperidyl-4-ketonen |
| US3080372A (en) * | 1960-03-25 | 1963-03-05 | Res Lab Dr C Janssen | 1-aroylalkyl-4-arylpiperidine derivatives |
| CH492710A (de) * | 1968-01-11 | 1970-06-30 | Geigy Ag J R | Verfahren zur Herstellung von neuen Piperidinderivaten |
| CH498836A (de) * | 1968-12-20 | 1970-11-15 | Geigy Ag J R | Verfahren zur Herstellung von neuen Piperidinderivaten |
| US3852455A (en) * | 1970-11-27 | 1974-12-03 | Richardson Merrell Inc | 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers |
| ZA717147B (en) * | 1970-11-27 | 1972-07-26 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives |
| US3888867A (en) * | 1972-05-03 | 1975-06-10 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)4'-fluorobutyrophenone derivatives |
| US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
| SE7409245L (fr) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
| GB1535791A (en) * | 1975-05-07 | 1978-12-13 | Ferrosan Ab | Derivatives of 4-piperidinol |
| CH602642A5 (fr) * | 1975-11-14 | 1978-07-31 | Orgamol Sa | |
| US4335127A (en) * | 1979-01-08 | 1982-06-15 | Janssen Pharmaceutica, N.V. | Piperidinylalkyl quinazoline compounds, composition and method of use |
-
1980
- 1980-10-22 ZA ZA00806501A patent/ZA806501B/xx unknown
- 1980-10-23 DE DE19803039974 patent/DE3039974A1/de not_active Withdrawn
- 1980-10-23 ES ES496204A patent/ES8201550A1/es not_active Expired
- 1980-10-24 GB GB8034418A patent/GB2061937A/en not_active Withdrawn
- 1980-10-24 IT IT49998/80A patent/IT1146198B/it active
- 1980-10-24 FR FR8022862A patent/FR2468592A1/fr active Granted
- 1980-10-24 AU AU63694/80A patent/AU6369480A/en not_active Abandoned
- 1980-10-24 CA CA000363264A patent/CA1148162A/fr not_active Expired
- 1980-10-24 IL IL61340A patent/IL61340A0/xx unknown
- 1980-10-27 NL NL8005890A patent/NL8005890A/nl not_active Application Discontinuation
- 1980-10-27 BE BE0/202608A patent/BE885894A/fr not_active IP Right Cessation
- 1980-10-27 JP JP14952780A patent/JPS5673061A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FR2468592B1 (fr) | 1983-08-05 |
| ES496204A0 (es) | 1981-12-01 |
| GB2061937A (en) | 1981-05-20 |
| BE885894A (fr) | 1981-02-16 |
| JPS5673061A (en) | 1981-06-17 |
| NL8005890A (nl) | 1981-04-29 |
| ZA806501B (en) | 1981-10-28 |
| IT1146198B (it) | 1986-11-12 |
| IT8049998A0 (it) | 1980-10-24 |
| FR2468592A1 (fr) | 1981-05-08 |
| CA1148162A (fr) | 1983-06-14 |
| AU6369480A (en) | 1981-04-30 |
| DE3039974A1 (de) | 1981-05-07 |
| IL61340A0 (en) | 1980-12-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19970303 |