ES8201966A1 - Un procedimiento de produccion de derivados de fenetilamina sulfamoil-sustituidos - Google Patents

Un procedimiento de produccion de derivados de fenetilamina sulfamoil-sustituidos

Info

Publication number
ES8201966A1
ES8201966A1 ES499224A ES499224A ES8201966A1 ES 8201966 A1 ES8201966 A1 ES 8201966A1 ES 499224 A ES499224 A ES 499224A ES 499224 A ES499224 A ES 499224A ES 8201966 A1 ES8201966 A1 ES 8201966A1
Authority
ES
Spain
Prior art keywords
group
lower alkyl
hydrogen
sulfamoyl
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES499224A
Other languages
English (en)
Other versions
ES499224A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yamanouchi Pharmaceutical Co Ltd
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11859488&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES8201966(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Publication of ES499224A0 publication Critical patent/ES499224A0/es
Publication of ES8201966A1 publication Critical patent/ES8201966A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D203/08—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring nitrogen atom
    • C07D203/10—Radicals substituted by singly bound oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE FENETILAMINA SULFAMOIL-SUSTITUIDOS DE FORMULA (I), ASI COMO DE SUS SALES, EN LA QUE R1 ES UN GRUPO AMINO A AMINO SUSTITUIDO; R2, R3, R4, R5, R6, R7, R8, R9 Y R10 PUEDEN SER VARIOS TIPOS DE RADICALES, E Y ES OXIGENO O RADICAL METILENO. CONSISTE EN LA REACCION DE UN COMPUESTO DE FORMULA (II), EN LA QUE R ES HIDROGENO O UN RADICAL ALQUILO INFERIOR, Y R1-R10 E Y TIENEN EL MISMO SIGNIFICACO QUE EN LA FORMULA (I), CON UN AGENTE HALOGENANTE, EN UN DISOLVENTE ORGANICO INERTE, A LA TEMPERATURA AMBIENTE O BAJO CALEFACCION. SI SE DESEA, EL PRODUCTO HALOGENADO OBTENIDO SE PUEDE REDUCIR CON HIDROGENO EN PRESENCIA DE UN CATALIZADOR, O SE PUEDE TRATAR CON UN ALCALI Y A CONTINUACION CON YODURO DE HIDROGENO, UN ALCOHOL Y TIOFENOL.
ES499224A 1980-02-08 1981-02-06 Un procedimiento de produccion de derivados de fenetilamina sulfamoil-sustituidos Expired ES8201966A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1438280A JPS56110665A (en) 1980-02-08 1980-02-08 Sulfamoyl-substituted phenetylamine derivative and its preparation

Publications (2)

Publication Number Publication Date
ES499224A0 ES499224A0 (es) 1982-01-01
ES8201966A1 true ES8201966A1 (es) 1982-01-01

Family

ID=11859488

Family Applications (1)

Application Number Title Priority Date Filing Date
ES499224A Expired ES8201966A1 (es) 1980-02-08 1981-02-06 Un procedimiento de produccion de derivados de fenetilamina sulfamoil-sustituidos

Country Status (17)

Country Link
US (6) US4373106A (es)
EP (1) EP0034432B1 (es)
JP (1) JPS56110665A (es)
AR (2) AR227533A1 (es)
AT (1) ATE7223T1 (es)
AU (1) AU541720B2 (es)
CA (1) CA1177849A (es)
DE (2) DE19675042I2 (es)
ES (1) ES8201966A1 (es)
GR (1) GR73827B (es)
IE (1) IE50862B1 (es)
LU (1) LU90000I2 (es)
MX (2) MX6859E (es)
NL (1) NL950014I2 (es)
PT (1) PT72460B (es)
SU (3) SU1082320A3 (es)
UA (3) UA5981A1 (es)

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US4558106A (en) * 1983-03-29 1985-12-10 Union Carbide Corporation Polymerization process using metal formate to reduce the color of thermoplastic copolymers

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AR227533A1 (es) 1982-11-15
IE50862B1 (en) 1986-08-06
NL950014I2 (nl) 1997-01-06
US4703063A (en) 1987-10-27
AU541720B2 (en) 1985-01-17
SU1248533A3 (ru) 1986-07-30
PT72460A (en) 1981-03-01
US4987152A (en) 1991-01-22
AR230433A1 (es) 1984-04-30
US4373106A (en) 1983-02-08
AU6689681A (en) 1981-08-13
LU90000I2 (fr) 1997-03-04
SU1082320A3 (ru) 1984-03-23
EP0034432B1 (en) 1984-04-25
US4868216A (en) 1989-09-19
DE3163257D1 (en) 1984-05-30
ES499224A0 (es) 1982-01-01
US4761500A (en) 1988-08-02
EP0034432A2 (en) 1981-08-26
SU1181540A3 (ru) 1985-09-23
JPS6252742B2 (es) 1987-11-06
JPS56110665A (en) 1981-09-01
CA1177849A (en) 1984-11-13
UA5980A1 (uk) 1994-12-29
US4731478A (en) 1988-03-15
DE19675042I2 (de) 2001-06-13
IE810236L (en) 1981-08-08
MX9203592A (es) 1992-07-31
PT72460B (en) 1982-02-04
GR73827B (es) 1984-05-04
ATE7223T1 (de) 1984-05-15
MX6859E (es) 1986-09-08
UA5990A1 (uk) 1994-12-29
UA5981A1 (uk) 1994-12-29
EP0034432A3 (en) 1982-03-24
NL950014I1 (nl) 1996-12-02

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