ES8304076A1 - "procedimiento de preparacion de compuestos del tipo arilbencensulfonamida". - Google Patents

"procedimiento de preparacion de compuestos del tipo arilbencensulfonamida".

Info

Publication number
ES8304076A1
ES8304076A1 ES513138A ES513138A ES8304076A1 ES 8304076 A1 ES8304076 A1 ES 8304076A1 ES 513138 A ES513138 A ES 513138A ES 513138 A ES513138 A ES 513138A ES 8304076 A1 ES8304076 A1 ES 8304076A1
Authority
ES
Spain
Prior art keywords
processes
preparation
radical
group
arylbenzenesulfonamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES513138A
Other languages
English (en)
Other versions
ES513138A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Choay SA
Original Assignee
Choay SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8111858A external-priority patent/FR2507598A1/fr
Priority claimed from FR8111859A external-priority patent/FR2507474A1/fr
Application filed by Choay SA filed Critical Choay SA
Publication of ES513138A0 publication Critical patent/ES513138A0/es
Publication of ES8304076A1 publication Critical patent/ES8304076A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/34—Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE COMPUESTOS DE TIPO ARILBENCENSULFONAMIDA, DE FORMULA GENERAL (I), EN DONDE AR REPRESENTA UN RADICAL; R , R Y R REPRESENTAN UN ATOMO DE HIDROGENO O DE HALOGENO; N+M+L ESTA COMPRENDIDO ENTRE 3 Y 11; R Y R REPRESENTAN UN ATOMO DE HIDROGENO O UN RADICAL ALCOHILO; R REPRESENTA UN GRUPO HIDROXI O UN RADICAL OR , EN DONDE R REPRESENTA UN GRUPO ALQUILO, Y DE SUS SALES. CONSISTE EN HACER REACCIONAR UN SULFOHALOGENURO ARSO X, SIENDO X UN HALOGENO, CON UN AMINO-ESTER DE FORMULA (II) O CON UN CLORHIDRATO DE FORMULA (III), EN PRESENCIA DE UNA BASE ORGANICA. DE APLICACION EN LA PREPARACION DE MEDICAMENTOS POR SUS PROPIEDADES NORMOLIPEMIANTES.
ES513138A 1981-06-16 1982-06-16 "procedimiento de preparacion de compuestos del tipo arilbencensulfonamida". Expired ES8304076A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8111858A FR2507598A1 (fr) 1981-06-16 1981-06-16 Nouveaux composes du type arylbenzenesulfonamide, leurs procedes de preparation et leurs applications a titre de substance active de medicaments normolipemiants
FR8111859A FR2507474A1 (en) 1981-06-16 1981-06-16 Benzene, thiophene and pyrimidine sulphonamido alkanoic acid derivs. - are normolipaemic cpds. with good therapeutic index, have low toxicity

Publications (2)

Publication Number Publication Date
ES513138A0 ES513138A0 (es) 1983-03-16
ES8304076A1 true ES8304076A1 (es) 1983-03-16

Family

ID=26222437

Family Applications (1)

Application Number Title Priority Date Filing Date
ES513138A Expired ES8304076A1 (es) 1981-06-16 1982-06-16 "procedimiento de preparacion de compuestos del tipo arilbencensulfonamida".

Country Status (7)

Country Link
US (2) US4613618A (es)
EP (1) EP0068968B1 (es)
CA (1) CA1214170A (es)
DE (1) DE3266360D1 (es)
DK (1) DK271282A (es)
ES (1) ES8304076A1 (es)
IE (1) IE53577B1 (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4885027A (en) * 1985-04-05 1989-12-05 Chevron Research Company Herbicidal arylmethylenesulfonamido-acetamide and thioacetamide derivatives
FR2598412B1 (fr) * 1986-03-12 1988-10-21 Sanofi Sa Nouveaux derives de diarylcetones et leurs procedes de preparation et les compositions pharmaceutiques les contenant
AU627434B2 (en) * 1987-08-20 1992-08-27 Boehringer Mannheim Gmbh W-arylsulphonamidoalkanoic acids for treatment of thromboxane mediated diseases
JPH02501142A (ja) * 1987-08-20 1990-04-19 スミス・クライン・アンド・フレンチ・ラボラトリース・リミテッド 生物学的に活性な化合物
IT1228454B (it) * 1989-02-22 1991-06-19 Roussel Maestretti S P A Milan Derivati del 1-arilsolfonil 2 piperidone, loro procedimento di preparazione e loro impiego come farmaci.
IL94805A (en) * 1989-06-28 1994-04-12 Ciba Geigy Ag (Arylsulfonamido- and pyridyl- or imidazolyl-)-substituted carboxylic acids, processfor their preparation and pharmaceutical compositions containing them
US5153214A (en) * 1989-06-28 1992-10-06 Ciba-Geigy Corporation Certain (arylsulfonamido- and imidazolyl-)-substituted carboxylic acids and derivatives thereof and use for suppressing thromboxane activity
US5025025A (en) * 1989-06-28 1991-06-18 Ciba-Geigy Corporation (Arylsulfonamido- and pyridyl-)-substituted carboxylic acids and derivatives thereof and use for suppressing thromboxane activity
EP0817643B1 (en) * 1995-03-31 2007-03-21 Emisphere Technologies, Inc. Compounds and compositions for delivering active agents
EP1792624A1 (en) * 1995-03-31 2007-06-06 Emisphere Technologies, Inc. Modified amino acids and compositions comprising them for delivering active agents
US6001347A (en) 1995-03-31 1999-12-14 Emisphere Technologies, Inc. Compounds and compositions for delivering active agents
UA67754C2 (uk) * 1997-10-10 2004-07-15 Пфайзер, Інк. Агоністи простагландину, фармацевтична композиція на їх основі (варіанти), спосіб нарощення та збереження кісткової маси у хребетних та спосіб лікування (варіанти)
AP2002002555A0 (en) 1999-12-22 2002-06-30 Pfizer Prod Inc EP4 Receptor selective agonists in the treatment of osteoporosis.
NZ523017A (en) * 2000-06-29 2004-10-29 Emisphere Tech Inc Compounds and compositions for delivering active agents and preparation method thereof
WO2003057650A2 (en) * 2002-01-09 2003-07-17 Emisphere Technologies, Inc. Polymorphs of sodium 4-[(4-chloro-2-hydroxybenzoyl)amino]butanoate
KR100463418B1 (ko) * 2002-11-11 2004-12-23 한국전자통신연구원 Ｃｅｌｐ 음성 부호화기에서 사용되는 가변적인 고정코드북 검색방법 및 장치

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE566666A (es) *
NL47894C (es) * 1900-01-01
US2142847A (en) * 1937-10-30 1939-01-03 Calco Chemical Co Inc Aminoarylsulphonylamino aliphatic acids and their salts
GB562349A (en) * 1943-02-12 1944-06-28 Wellcome Found Improvements relating to the manufacture of sulphanilamide derivatives
US2592105A (en) * 1948-11-16 1952-04-08 Sterling Drug Inc Iodinated aminophenylsulfonylamino carboxylic acids
DE1101408B (de) * 1959-02-10 1961-03-09 Chemische Werke Radebeul Veb Verfahren zur Herstellung von blutzuckersenkend wirkenden Sulfonylaminocarbonsaeurederivaten
GB1194388A (en) * 1966-11-08 1970-06-10 American Cyanamid Co Preparation of N-(2-Carbamoylethyl) and N,N-Bis(2-Carbamoylethyl) Sulfonamides
FR7477M (es) * 1968-04-16 1969-12-01
CA1072359A (en) * 1974-10-08 1980-02-26 Hiroyuki Konishi Method for controlling the growth of plants
US4349378A (en) * 1978-07-25 1982-09-14 Fbc Limited Compounds useful as pesticides

Also Published As

Publication number Publication date
US4761430A (en) 1988-08-02
ES513138A0 (es) 1983-03-16
IE53577B1 (en) 1988-12-21
DE3266360D1 (en) 1985-10-24
EP0068968B1 (fr) 1985-09-18
DK271282A (da) 1982-12-17
CA1214170A (fr) 1986-11-18
IE821434L (en) 1982-12-16
EP0068968A1 (fr) 1983-01-05
US4613618A (en) 1986-09-23

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