ES8507155A3 - Metodo para la obtencion de esteroides de la serie de prednisolona - Google Patents
Metodo para la obtencion de esteroides de la serie de prednisolonaInfo
- Publication number
- ES8507155A3 ES8507155A3 ES538539A ES538539A ES8507155A3 ES 8507155 A3 ES8507155 A3 ES 8507155A3 ES 538539 A ES538539 A ES 538539A ES 538539 A ES538539 A ES 538539A ES 8507155 A3 ES8507155 A3 ES 8507155A3
- Authority
- ES
- Spain
- Prior art keywords
- steroid
- 17alpha
- formula
- prednisolone
- series
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000003431 steroids Chemical class 0.000 title abstract 3
- 150000003117 prednisolones Chemical class 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 238000005886 esterification reaction Methods 0.000 abstract 2
- 229910052736 halogen Chemical group 0.000 abstract 2
- 150000002367 halogens Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 230000007062 hydrolysis Effects 0.000 abstract 2
- 238000006460 hydrolysis reaction Methods 0.000 abstract 2
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 238000006136 alcoholysis reaction Methods 0.000 abstract 1
- 230000008030 elimination Effects 0.000 abstract 1
- 238000003379 elimination reaction Methods 0.000 abstract 1
- 230000032050 esterification Effects 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
Landscapes
- Steroid Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE ESTEROIDES DE LA SERIE DE PREDNISOLONA, DE FORMULA (I), EN LA QUE Y Y Z PUEDENSER HIDROGENO O UN HALOGENO; Y Z ADEMAS UN ALQUILO INFERIOR.CONSISTE EN LA ORTOESTERIFICACION DE UN ESTEROIDE, DE FORMULA (II) PARA FORMAR UN COMPUESTO DE FORMULA (III), EN LA QUE R Y RK SON GRUPOS ALQUILICO DE 1-6 ATOMOS DE CARBONO; SEGUIDA DE LA HIDROLISIS DEL ORTOESTER PARA FORMAR UN 17BAB-ESTER; ESTERIFICACION DE ESTER PARA FORMAR UN 17BAB,21-DIESTER EN EL QUE EL NUEVO GRUPO ACILO TIENE 2-7 ATOMOS DE CARBONO. ELIMINACION DEL GRUPO 17BAB-ACILOXI; OXIDACION SELECTIVA DEL BDB 16-21-ESTER FORMADO; E HIDROLISIS O ALCOHOLISIS DEL 16BAB,17BAB-DIHIDROXI-21-ESTER, ULTIMAMENTE PRODUCIDO.ESTOS COMPUESTOS TIENEN APLICACIONES PARA FINES TERAPEUTICOS Y COMO INTERMEDIOS PARA LA PREPARACION DE DERIVADOS.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES538539A ES8507155A3 (es) | 1984-12-12 | 1984-12-12 | Metodo para la obtencion de esteroides de la serie de prednisolona |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES538539A ES8507155A3 (es) | 1984-12-12 | 1984-12-12 | Metodo para la obtencion de esteroides de la serie de prednisolona |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES538539A0 ES538539A0 (es) | 1985-09-01 |
| ES8507155A3 true ES8507155A3 (es) | 1985-09-01 |
Family
ID=8488307
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES538539A Expired ES8507155A3 (es) | 1984-12-12 | 1984-12-12 | Metodo para la obtencion de esteroides de la serie de prednisolona |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES8507155A3 (es) |
-
1984
- 1984-12-12 ES ES538539A patent/ES8507155A3/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES538539A0 (es) | 1985-09-01 |
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