ES8507614A1 - Un procedimiento para la preparacion de nuevos antibioticos glicopeptidos n-acilados. - Google Patents

Un procedimiento para la preparacion de nuevos antibioticos glicopeptidos n-acilados.

Info

Publication number
ES8507614A1
ES8507614A1 ES536876A ES536876A ES8507614A1 ES 8507614 A1 ES8507614 A1 ES 8507614A1 ES 536876 A ES536876 A ES 536876A ES 536876 A ES536876 A ES 536876A ES 8507614 A1 ES8507614 A1 ES 8507614A1
Authority
ES
Spain
Prior art keywords
formula
procedure
acylated
glycopeptide antibiotics
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES536876A
Other languages
English (en)
Other versions
ES536876A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES536876A0 publication Critical patent/ES536876A0/es
Publication of ES8507614A1 publication Critical patent/ES8507614A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07G—COMPOUNDS OF UNKNOWN CONSTITUTION
    • C07G11/00—Antibiotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/19—Antibiotic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/27—Cyclic peptide or cyclic protein

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Fodder In General (AREA)
  • Feed For Specific Animals (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE ANTIBIOTICOS GLICOPEPTIDOS N-ACILADOS, DE FORMULA (I), EN LA QUE W ES EL RESTO DE UN GLICOPEPTIDO ANTIBIOTICO Y R ES UN GRUPO ACILO.CONSISTE EN LA REACCION DE ACILACION DE UN ANTIBIOTICO PARENTAL, DE FORMULA (II), CON UN DERIVADO ACTIVO DE UN COMPUESTO DE FORMULA (III), (IV), O (V), EN LAS QUE W TIENE EL MISMO SIGNIFICADO QUE EN LA FORMULA (I), P, R Y SE VALEN 0 O 1, M Y N VALEN 0-10, Y LOS DEMAS SIMBOLOS REPRESENTAN VARIOS TIPOS DE RADICALES; SEGUIDA DE LA EVENTUAL SEPARACION DEL GRUPO PROTECTOR DEL AMINO.ESTOS COMPUESTOS TIENEN APLICACIONES COMO ADITIVOS DE PIENSOS.
ES536876A 1983-10-21 1984-10-18 Un procedimiento para la preparacion de nuevos antibioticos glicopeptidos n-acilados. Expired ES8507614A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/544,336 US4497802A (en) 1983-10-21 1983-10-21 N-Acyl glycopeptide derivatives

Publications (2)

Publication Number Publication Date
ES536876A0 ES536876A0 (es) 1985-09-01
ES8507614A1 true ES8507614A1 (es) 1985-09-01

Family

ID=24171768

Family Applications (1)

Application Number Title Priority Date Filing Date
ES536876A Expired ES8507614A1 (es) 1983-10-21 1984-10-18 Un procedimiento para la preparacion de nuevos antibioticos glicopeptidos n-acilados.

Country Status (15)

Country Link
US (1) US4497802A (es)
EP (1) EP0142940A3 (es)
JP (1) JPS60172997A (es)
KR (1) KR860001280B1 (es)
AU (1) AU3374984A (es)
DK (1) DK501384A (es)
ES (1) ES8507614A1 (es)
FI (1) FI844043L (es)
GB (1) GB2148304B (es)
GR (1) GR80689B (es)
HU (1) HUT35697A (es)
IL (1) IL73251A0 (es)
PL (1) PL250043A1 (es)
PT (1) PT79374B (es)
ZA (1) ZA848154B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU579120B2 (en) * 1983-12-16 1988-11-17 Gruppo Lepetit S.P.A. Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
GB8415092D0 (en) * 1984-06-13 1984-07-18 Lepetit Spa Ester derivatives
GB8415093D0 (en) * 1984-06-13 1984-07-18 Lepetit Spa Antibiotic l 17392
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4639433A (en) * 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
GB8522574D0 (en) * 1985-09-12 1985-10-16 Lepetit Spa Amides of teicoplanin compounds
PT86457B (pt) * 1986-12-30 1990-11-20 Smithkline Beecham Corp Processo para a preparacao de glicopeptidos glicosilados e de composicoes que os contem
US4882313A (en) * 1987-07-31 1989-11-21 Smithkline Beckman Corporation Carboxamide derivatives of glycopeptides
EP0368949A1 (en) * 1988-02-10 1990-05-23 Beecham Group Plc Novel antibiotic compounds
EP0409045B1 (en) * 1989-07-18 1997-11-19 Biosearch Italia S.p.A. Pentapeptide antibiotics derived from dalbaheptides
DE69908819T2 (de) 1998-12-23 2004-05-06 Theravance, Inc., South San Francisco Glycopeptid-derivate und pharmazeutische zusammensetzungen, die sie enthalten
US20030211204A1 (en) * 2002-05-10 2003-11-13 Fields Christine C. Method of preparing beverages and beverage concentrates nutritionally supplemented with minerals
CA2588285A1 (en) * 2004-11-29 2006-06-01 National University Corporation Nagoya University Glycopeptide antibiotic monomer derivatives
CA2623239C (en) 2005-09-22 2016-07-12 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
JP5192384B2 (ja) 2005-09-22 2013-05-08 メディバス エルエルシー ビス−（α−アミノ）−ジオール−ジエステル含有ポリ（エステルアミド）およびポリ（エステルウレタン）組成物および使用の方法
CN101959900A (zh) 2007-12-26 2011-01-26 盐野义制药株式会社 糖肽类抗生素糖基化衍生物
EP2260060A4 (en) 2008-04-01 2013-01-16 Univ Cornell ORGANIC SOLUBLE CHITOSA SALT AND CHITOSAN DERIVED BIOMATERIALS MANUFACTURED THEREFROM
IN2013CH04314A (es) 2013-09-23 2015-08-28 Jawaharlal Nehru Ct For Advanced Scient Res Jncasr

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2990329A (en) * 1957-02-11 1961-06-27 Abbott Lab Preparation of ristocetin a salts
US3928571A (en) * 1972-12-15 1975-12-23 Lilly Co Eli Ruminant feed utilization improvement
US4115552A (en) * 1976-04-19 1978-09-19 Eli Lilly And Company Factor A and B of antibiotic A-4696
US4029769A (en) * 1976-05-24 1977-06-14 Eli Lilly And Company Antibiotic A-35512B aglycone
US4083964A (en) * 1976-05-24 1978-04-11 Eli Lilly And Company Antibiotic A-35512 for increasing feed utilization efficiency in an animal
US4322406A (en) * 1980-12-18 1982-03-30 Eli Lilly And Company Antibiotic A-4696 factors B1, B2, B3, C1a, C3 and E1
US4322343A (en) * 1980-12-18 1982-03-30 Eli Lilly And Company Pseudo-aglycone of actaplanin

Also Published As

Publication number Publication date
GB8426210D0 (en) 1984-11-21
HUT35697A (en) 1985-07-29
AU3374984A (en) 1985-04-26
US4497802A (en) 1985-02-05
PT79374B (en) 1986-11-14
GR80689B (en) 1985-02-20
FI844043A7 (fi) 1985-04-22
EP0142940A3 (en) 1985-07-10
ES536876A0 (es) 1985-09-01
FI844043A0 (fi) 1984-10-15
JPS60172997A (ja) 1985-09-06
ZA848154B (en) 1985-12-24
DK501384D0 (da) 1984-10-19
EP0142940A2 (en) 1985-05-29
IL73251A0 (en) 1985-01-31
PT79374A (en) 1984-11-01
KR860001280B1 (ko) 1986-09-05
PL250043A1 (en) 1985-07-16
GB2148304A (en) 1985-05-30
FI844043L (fi) 1985-04-22
KR850003409A (ko) 1985-06-17
GB2148304B (en) 1987-03-04
DK501384A (da) 1985-04-22

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