FR1614M - Nouveau dérivé d'imidazoline et ses sels d'addition acides. - Google Patents

Nouveau dérivé d'imidazoline et ses sels d'addition acides.

Info

Publication number
FR1614M
FR1614M FR879728A FR879728A FR1614M FR 1614 M FR1614 M FR 1614M FR 879728 A FR879728 A FR 879728A FR 879728 A FR879728 A FR 879728A FR 1614 M FR1614 M FR 1614M
Authority
FR
France
Prior art keywords
imidazoline
acid addition
addition salts
new derivative
derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR879728A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck KGaA
Original Assignee
E Merck AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E Merck AG filed Critical E Merck AG
Application granted granted Critical
Publication of FR1614M publication Critical patent/FR1614M/fr
Active legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR879728A 1960-11-23 1961-11-22 Nouveau dérivé d'imidazoline et ses sels d'addition acides. Active FR1614M (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DEM47194A DE1121054B (de) 1960-11-23 1960-11-23 Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen

Publications (1)

Publication Number Publication Date
FR1614M true FR1614M (fr) 1962-12-17

Family

ID=7305839

Family Applications (1)

Application Number Title Priority Date Filing Date
FR879728A Active FR1614M (fr) 1960-11-23 1961-11-22 Nouveau dérivé d'imidazoline et ses sels d'addition acides.

Country Status (6)

Country Link
US (2) US3161653A (fr)
CH (1) CH446353A (fr)
DE (1) DE1121054B (fr)
FR (1) FR1614M (fr)
GB (1) GB951989A (fr)
SE (1) SE305877B (fr)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1595234A1 (de) * 1965-04-27 1970-03-05 Roehm & Haas Gmbh Verfahren zur Herstellung oligomerer bzw. polymerer Amine
US3438995A (en) * 1968-01-08 1969-04-15 Melville Sahyun Diazaheterocyclic substituted benz-oxaheterocyclic compounds
GB1333471A (en) * 1971-01-27 1973-10-10 Labaz Imidazoline derivatives and process for preparing the same
US4978332A (en) * 1987-09-28 1990-12-18 Matrix Pharmaceutical, Inc. Treatments employing vasoconstrictive substances in combination with cytotoxic agents for introduction into cellular lesion areas
JPH10501823A (ja) * 1995-04-10 1998-02-17 バクスター、インターナショナル、インコーポレイテッド クモ膜下出血の治療における架橋ヘモグロビンの使用
WO1999032482A1 (fr) * 1997-12-19 1999-07-01 Eli Lilly And Company Composes d'imidazoline hypoglycemiques
CA2637312A1 (fr) * 2006-01-27 2007-08-02 F. Hoffmann-La Roche Ag Utilisation de 2-imidazole substitue de derives d'imidazoline
WO2008046756A1 (fr) * 2006-10-19 2008-04-24 F. Hoffmann-La Roche Ag Aminométhyl- 2 -imidazoles à affinité avec les récepteurs associés à une amine à l'état de trace
CA2666762C (fr) * 2006-10-19 2014-12-30 F. Hoffmann-La Roche Ag Aminomethyl-4-imidazoles
EP2086959B1 (fr) * 2006-11-02 2011-11-16 F. Hoffmann-La Roche AG 2-IMIDAZOLES SUBSTITUES EN TANT QUE MODULATEURS DES RECEPTEURS ASSOCIES AUX AMINES A l'ETAT DE TRACES
MX2009005047A (es) * 2006-11-16 2009-05-25 Hoffmann La Roche 4-imidazoles sustituidos.
MX2009005920A (es) * 2006-12-13 2009-06-16 Hoffmann La Roche Nuevos 2-imidazoles como ligandos para receptores asociados con trazas de amina.
US20080146523A1 (en) 2006-12-18 2008-06-19 Guido Galley Imidazole derivatives
MX2009008255A (es) * 2007-02-02 2009-08-12 Hoffmann La Roche Nuevas 2-aminooxazolinas como ligandos taar1.
KR101222412B1 (ko) * 2007-02-15 2013-01-15 에프. 호프만-라 로슈 아게 Ｔａａｒ1 리간드로서의 2-아미노옥사졸린
CN101687812A (zh) 2007-07-02 2010-03-31 弗·哈夫曼-拉罗切有限公司 对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物
WO2009003867A1 (fr) * 2007-07-03 2009-01-08 F. Hoffmann-La Roche Ag 4-imidazolines et leur utilisation comme antidépresseurs
WO2009016048A1 (fr) * 2007-07-27 2009-02-05 F. Hoffmann-La Roche Ag 2-azétidineméthaneamines et 2-pyrrolidineméthaneamines comme ligands de taar
CN101765425A (zh) * 2007-08-02 2010-06-30 弗·哈夫曼-拉罗切有限公司 苯甲酰胺衍生物用于治疗cns障碍的用途
BRPI0814758A2 (pt) * 2007-08-03 2015-03-03 Hoffmann La Roche Piridinacarboxamida e derivados de benzamida como ligantes taar1
US8242153B2 (en) * 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
CN102083805A (zh) * 2008-07-24 2011-06-01 弗·哈夫曼-拉罗切有限公司 4,5-二氢-唑-2-基衍生物
US20100311798A1 (en) * 2009-06-05 2010-12-09 Decoret Guillaume 2-aminooxazolines as taar1 ligands
US8354441B2 (en) * 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
JP6814814B2 (ja) 2016-03-17 2021-01-20 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ Ｔａａｒのアゴニストとしての活性を有する５−エチル−４−メチル−ピラゾール−３−カルボキサミド誘導体

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1049387B (de) * 1959-01-29 Ciba Aktiengesellschaft, Basel (Schweiz) Verfahren zur Herstellung eines neuen Imidazolins
US2965648A (en) * 1960-12-20 Certain i-alkenyl benzimidazoles
US2441867A (en) * 1943-11-19 1948-05-18 Recip Ab Methods of producing 2-(alpha-naphthylmethyl)-imidazoline
US2457047A (en) * 1946-02-13 1948-12-21 Monsanto Chemicals 2-(2'-thenyl)-4, 5-dihydroimidazoles and process for making the same
US2780577A (en) * 1951-05-26 1957-02-05 Burroughs Wellcome Co Inhibiting polymethylene diquaternary curariform activity by alpha-stilbazoline derivatives
US2744909A (en) * 1955-06-27 1956-05-08 Bristol Lab Inc 2-(ortho-phenylbenzyl) imidazoline and acid addition salts
US3024248A (en) * 1956-09-18 1962-03-06 Ciba Pharm Prod Inc Organic sulfur compounds and method for producing same
US2955073A (en) * 1958-06-02 1960-10-04 Burroughs Wellcome Co Method of treating febrile convulsions
NL277287A (fr) * 1958-09-02
US3010972A (en) * 1960-03-18 1961-11-28 Smith Kline French Lab Condensed cyclopropyl amine derivatives
US3042674A (en) * 1960-07-12 1962-07-03 Sahyun Xanthene and thiaxanthene cyclic amidines

Also Published As

Publication number Publication date
GB951989A (en) 1964-03-11
DE1121054B (de) 1962-01-04
SE305877B (fr) 1968-11-11
CH446353A (de) 1967-11-15
US3161653A (en) 1964-12-15
US3238101A (en) 1966-03-01

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