FR2491073A1 - Nouveaux derives 1-n- (a-hydroxy-o-aminoalcanoyl des 5,3',4'-tridesoxy- ou 5,3',4'-tridesoxy-6'-n-methyl- ou 5,3',4',6''-tetradesoxykanamycine b, leurs procedes de production et les compositions antibacteriennes les renfermant - Google Patents

Nouveaux derives 1-n- (a-hydroxy-o-aminoalcanoyl des 5,3',4'-tridesoxy- ou 5,3',4'-tridesoxy-6'-n-methyl- ou 5,3',4',6''-tetradesoxykanamycine b, leurs procedes de production et les compositions antibacteriennes les renfermant Download PDF

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Publication number
FR2491073A1
FR2491073A1 FR8115781A FR8115781A FR2491073A1 FR 2491073 A1 FR2491073 A1 FR 2491073A1 FR 8115781 A FR8115781 A FR 8115781A FR 8115781 A FR8115781 A FR 8115781A FR 2491073 A1 FR2491073 A1 FR 2491073A1
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FR
France
Prior art keywords
formula
amino
group
hydroxy
str2
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8115781A
Other languages
English (en)
French (fr)
Other versions
FR2491073B1 (2
Inventor
Hamao Umezawa
Shinichi Kondo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Microbial Chemistry Research Foundation
Original Assignee
Microbial Chemistry Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP55109854A external-priority patent/JPS5753496A/ja
Priority claimed from JP56058389A external-priority patent/JPS57175198A/ja
Application filed by Microbial Chemistry Research Foundation filed Critical Microbial Chemistry Research Foundation
Publication of FR2491073A1 publication Critical patent/FR2491073A1/fr
Application granted granted Critical
Publication of FR2491073B1 publication Critical patent/FR2491073B1/fr
Granted legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FR8115781A 1980-08-12 1981-08-10 Nouveaux derives 1-n- (a-hydroxy-o-aminoalcanoyl des 5,3',4'-tridesoxy- ou 5,3',4'-tridesoxy-6'-n-methyl- ou 5,3',4',6''-tetradesoxykanamycine b, leurs procedes de production et les compositions antibacteriennes les renfermant Granted FR2491073A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP55109854A JPS5753496A (en) 1980-08-12 1980-08-12 1-n-acyl derivative of 5,3',4'-trideoxykanamycin b or 5,3',4',6'- tetradeoxykanamycin b, and their preparation
JP56058389A JPS57175198A (en) 1981-04-20 1981-04-20 1-n-acyl derivative of 5,3,4-trideoxy-6-n-methylkanamycin b and their preparation

Publications (2)

Publication Number Publication Date
FR2491073A1 true FR2491073A1 (fr) 1982-04-02
FR2491073B1 FR2491073B1 (2) 1984-08-03

Family

ID=26399440

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8115781A Granted FR2491073A1 (fr) 1980-08-12 1981-08-10 Nouveaux derives 1-n- (a-hydroxy-o-aminoalcanoyl des 5,3',4'-tridesoxy- ou 5,3',4'-tridesoxy-6'-n-methyl- ou 5,3',4',6''-tetradesoxykanamycine b, leurs procedes de production et les compositions antibacteriennes les renfermant

Country Status (9)

Country Link
KR (1) KR850000979B1 (2)
CA (1) CA1175816A (2)
CH (1) CH648564A5 (2)
DE (1) DE3131731C2 (2)
ES (4) ES504697A0 (2)
FR (1) FR2491073A1 (2)
GB (1) GB2082575B (2)
IT (1) IT1167959B (2)
NL (1) NL8103639A (2)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2242400A1 (2) * 1973-08-29 1975-03-28 Microbial Chem Res Found

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2242400A1 (2) * 1973-08-29 1975-03-28 Microbial Chem Res Found

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
JOURNAL OF ANTIBIOTICS, volume 34, no. 12, décembre 1981 (TOKYO, JP) "Chemical modification of 5,3',4'-trideoxykanamycin B", pages 1635-1640 *
THE JAPANESE JOURNAL OF ANTIBIOTICS, volume 32 supplément, décembre 1979 (TOKYO, JP) S. FUKATSU "Industrial chemical synthesis of dideoxykanamycin B", pages S-178-186 *

Also Published As

Publication number Publication date
ES8401093A1 (es) 1983-12-16
ES8308334A1 (es) 1983-08-16
ES514622A0 (es) 1983-08-16
ES8301486A1 (es) 1982-12-01
ES8401092A1 (es) 1983-12-16
DE3131731C2 (de) 1984-02-16
IT8109493A0 (it) 1981-08-07
ES514621A0 (es) 1983-12-16
FR2491073B1 (2) 1984-08-03
ES514620A0 (es) 1983-12-16
GB2082575A (en) 1982-03-10
ES504697A0 (es) 1982-12-01
KR850000979B1 (ko) 1985-07-05
KR830006325A (ko) 1983-09-24
GB2082575B (en) 1984-04-18
CA1175816A (en) 1984-10-09
CH648564A5 (de) 1985-03-29
DE3131731A1 (de) 1982-03-11
NL8103639A (nl) 1982-03-01
IT1167959B (it) 1987-05-20

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