GT200900294A - Compuestos amino-heterocíclicos - Google Patents

Compuestos amino-heterocíclicos

Info

Publication number: GT200900294A
Authority: GT; Guatemala
Prior art keywords: amino; heterocyclic compounds; same; compounds; lso
Prior art date: 2007-05-11

Application number

GT200900294A

Other languages

English (en)

Spanish (es)

Inventor

Proulx-La France Carolina

Verhoest Patrick Robert

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-05-11

Filing date

2009-11-10

Publication date

2011-08-29

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39672073&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200900294(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-11-10 Application filed filed Critical

2011-08-29 Publication of GT200900294A publication Critical patent/GT200900294A/es

Links

150000001875 compounds Chemical class 0.000 abstract 2
208000024827 Alzheimer disease Diseases 0.000 abstract 1
101100407341 Drosophila melanogaster Pde9 gene Proteins 0.000 abstract 1
208000010877 cognitive disease Diseases 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
208000015122 neurodegenerative disease Diseases 0.000 abstract 1
230000000626 neurodegenerative effect Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
201000000980 schizophrenia Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Diabetes (AREA)
Psychiatry (AREA)
Ophthalmology & Optometry (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Hospice & Palliative Care (AREA)
Virology (AREA)
Psychology (AREA)
Molecular Biology (AREA)
Pain & Pain Management (AREA)
Obesity (AREA)
AIDS & HIV (AREA)
Tropical Medicine & Parasitology (AREA)
Emergency Medicine (AREA)
Vascular Medicine (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Hematology (AREA)
Gynecology & Obstetrics (AREA)
Reproductive Health (AREA)

GT200900294A 2007-05-11 2009-11-10 Compuestos amino-heterocíclicos GT200900294A (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US91733307P	2007-05-11	2007-05-11

Publications (1)

Publication Number	Publication Date
GT200900294A true GT200900294A (es)	2011-08-29

Family

ID=39672073

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
GT200900294A GT200900294A (es)	2007-05-11	2009-11-10	Compuestos amino-heterocíclicos

Country Status (43)

Country	Link
US (1)	US7964607B2 (sr)
EP (1)	EP2152712B1 (sr)
JP (1)	JP4579346B2 (sr)
KR (1)	KR101222330B1 (sr)
CN (1)	CN101687876B (sr)
AP (1)	AP2524A (sr)
AR (1)	AR066502A1 (sr)
AT (1)	ATE540954T1 (sr)
AU (1)	AU2008249750B2 (sr)
BR (1)	BRPI0811280B8 (sr)
CA (1)	CA2687035C (sr)
CL (1)	CL2008001374A1 (sr)
CO (1)	CO6241157A2 (sr)
CR (1)	CR11095A (sr)
CU (1)	CU23834B1 (sr)
CY (1)	CY1112332T1 (sr)
DK (1)	DK2152712T3 (sr)
DO (1)	DOP2009000258A (sr)
EA (1)	EA016510B1 (sr)
EC (1)	ECSP099728A (sr)
ES (1)	ES2377849T3 (sr)
GE (1)	GEP20125405B (sr)
GT (1)	GT200900294A (sr)
HR (1)	HRP20120105T1 (sr)
IL (1)	IL201977A (sr)
MA (1)	MA31373B1 (sr)
ME (1)	ME00954B (sr)
MX (1)	MX2009011830A (sr)
MY (1)	MY147330A (sr)
NI (1)	NI200900204A (sr)
NZ (1)	NZ580904A (sr)
PA (1)	PA8779901A1 (sr)
PE (1)	PE20090247A1 (sr)
PL (1)	PL2152712T3 (sr)
PT (1)	PT2152712E (sr)
RS (1)	RS52166B (sr)
SI (1)	SI2152712T1 (sr)
SV (1)	SV2009003411A (sr)
TN (1)	TN2009000471A1 (sr)
TW (1)	TWI362262B (sr)
UA (1)	UA94660C2 (sr)
WO (1)	WO2008139293A1 (sr)
ZA (1)	ZA200907776B (sr)

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UA105362C2 (en) *	2008-04-02	2014-05-12	Бьорингер Ингельхайм Интернациональ Гмбх	1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
CN102143965A (zh)	2008-09-08	2011-08-03	贝林格尔.英格海姆国际有限公司	吡唑并嘧啶酮及其在治疗中枢神经系统疾病中的用途
CA2894860C (en)	2008-11-19	2018-11-06	Gerhard Koenig	Treatment of cognitive disorders with (r)-7-chloro-n-(quinuclidin-3-yl)benzo[b]thiophene-2-carboxamide and pharmaceutically acceptable salts thereof
TWI404721B (zh)	2009-01-26	2013-08-11	Pfizer	胺基－雜環化合物
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JP5808319B2 (ja) *	2009-05-11	2015-11-10	フォルムファーマシューティカルズ、インコーポレイテッド	アセチルコリンエステラーゼ阻害剤と組み合わせた特定のα７ニコチン酸受容体を用いた認知障害の治療
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HRP20160473T1 (hr)	2010-09-07	2016-07-29	Astellas Pharma Inc.	Pirazolokinolinski spojevi
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EP3666272A1 (en)	2012-05-08	2020-06-17	Forum Pharmaceuticals Inc.	Use of encenicline in the treatment of cognitive impairment, alzheimer's disease, memory deficit
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AU2014250392B2 (en)	2013-04-05	2018-03-01	Eisai R&D Management Co., Ltd.	Salt of pyrazoloquinoline derivative, and crystal thereof
PE20151718A1 (es)	2013-04-05	2015-11-22	Eisai Randd Man Co Ltd	Compuestos piridinilpirazoloquinolina
CN103626774B (zh) *	2013-11-20	2015-11-04	苏州明锐医药科技有限公司	伊鲁替尼的制备方法
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BR112018000254A2 (pt)	2015-07-07	2018-09-04	H Lundbeck As	inibidores de pde9 com cadeia principal de imidazotriazinona e cadeia principal de imidazopirazinona para o tratamento de doenças periféricas
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US10550126B2 (en)	2015-10-16	2020-02-04	Abbvie Inc.	Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-A]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
US11365198B2 (en)	2015-10-16	2022-06-21	Abbvie Inc.	Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
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TWI729109B (zh) *	2016-04-12	2021-06-01	丹麥商Ｈ朗德貝克公司	作爲PDE1抑制劑的1,5-二氫-4H-吡唑并[3,4-d]嘧啶-4-酮和1,5-二氫-4H-吡唑并[4,3-c]吡啶-4-酮
AU2017292650A1 (en)	2016-07-06	2018-12-13	H. Lundbeck A/S	PDE9 inhibitors for treatment of peripheral diseases
EP3529250B1 (en)	2016-10-18	2023-12-06	H. Lundbeck A/S	Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as pde1 inhibitors
SG11201903770UA (en)	2016-10-28	2019-05-30	H Lundbeck As	Combination treatments comprising imidazopyrazinones for the treatment of psychiatric and/or cognitive disorders
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EA200901373A1 (ru)	2010-06-30
CA2687035C (en)	2011-09-20
AP2524A (en)	2012-12-04
HK1142595A1 (en)	2010-12-10
TW200902015A (en)	2009-01-16
AP2009005048A0 (en)	2009-12-31
NI200900204A (es)	2010-03-11
BRPI0811280A2 (pt)	2015-01-20
CU20090184A7 (es)	2011-07-11
TN2009000471A1 (fr)	2011-03-31
UA94660C2 (en)	2011-05-25
IL201977A (en)	2014-07-31
TWI362262B (en)	2012-04-21
MX2009011830A (es)	2009-11-13
RS52166B (sr)	2012-08-31
ES2377849T3 (es)	2012-04-02
ME00954B (me)	2012-06-20
US7964607B2 (en)	2011-06-21
AU2008249750A1 (en)	2008-11-20
WO2008139293A1 (en)	2008-11-20
CU23834B1 (es)	2012-10-15
PT2152712E (pt)	2012-02-29
EP2152712A1 (en)	2010-02-17
MA31373B1 (fr)	2010-05-03
CL2008001374A1 (es)	2008-11-14
HRP20120105T1 (hr)	2012-02-29
CN101687876A (zh)	2010-03-31
DK2152712T3 (da)	2012-03-26
CN101687876B (zh)	2012-12-12
BRPI0811280B8 (pt)	2021-05-25
BRPI0811280B1 (pt)	2021-05-11
SV2009003411A (es)	2010-05-21
KR101222330B1 (ko)	2013-01-15
EP2152712B1 (en)	2012-01-11
ZA200907776B (en)	2011-01-26
EA016510B1 (ru)	2012-05-30
AR066502A1 (es)	2009-08-26
MY147330A (en)	2012-11-30
PE20090247A1 (es)	2009-03-13
JP2010526863A (ja)	2010-08-05
CA2687035A1 (en)	2008-11-20
GEP20125405B (en)	2012-02-27
ECSP099728A (es)	2009-12-28
AU2008249750B2 (en)	2011-07-14
PA8779901A1 (es)	2008-12-18
CY1112332T1 (el)	2015-12-09
PL2152712T3 (pl)	2012-05-31
KR20100007985A (ko)	2010-01-22
CR11095A (es)	2009-12-04
DOP2009000258A (es)	2010-05-15
SI2152712T1 (sl)	2012-03-30
US20090030003A1 (en)	2009-01-29
ATE540954T1 (de)	2012-01-15
IL201977A0 (en)	2010-06-16
NZ580904A (en)	2012-02-24
CO6241157A2 (es)	2011-01-20
JP4579346B2 (ja)	2010-11-10

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