HRP20000751A2 - Novel nucleosides having bicyclic sugar moiety - Google Patents

Novel nucleosides having bicyclic sugar moiety Download PDF

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Publication number
HRP20000751A2
HRP20000751A2 HR20000751A HRP20000751A HRP20000751A2 HR P20000751 A2 HRP20000751 A2 HR P20000751A2 HR 20000751 A HR20000751 A HR 20000751A HR P20000751 A HRP20000751 A HR P20000751A HR P20000751 A2 HRP20000751 A2 HR P20000751A2
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HR
Croatia
Prior art keywords
mmol
octane
dioxabicyclo
solution
title compound
Prior art date
Application number
HR20000751A
Other languages
English (en)
Croatian (hr)
Inventor
Guangyi Wang
Original Assignee
Icn Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Icn Pharmaceuticals filed Critical Icn Pharmaceuticals
Publication of HRP20000751A2 publication Critical patent/HRP20000751A2/hr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compounds Of Unknown Constitution (AREA)
HR20000751A 1998-05-26 1999-05-24 Novel nucleosides having bicyclic sugar moiety HRP20000751A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8671998P 1998-05-26 1998-05-26
PCT/US1999/011442 WO1999060855A1 (en) 1998-05-26 1999-05-24 Novel nucleosides having bicyclic sugar moiety

Publications (1)

Publication Number Publication Date
HRP20000751A2 true HRP20000751A2 (en) 2001-12-31

Family

ID=22200439

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20000751A HRP20000751A2 (en) 1998-05-26 1999-05-24 Novel nucleosides having bicyclic sugar moiety

Country Status (21)

Country Link
US (1) US6403566B1 (de)
EP (1) EP1082012A4 (de)
JP (1) JP2002516256A (de)
CN (1) CN1311630A (de)
AU (1) AU757724B2 (de)
BR (1) BR9911596A (de)
CA (1) CA2333380A1 (de)
HR (1) HRP20000751A2 (de)
HU (1) HUP0102152A3 (de)
IL (1) IL139420A0 (de)
MX (1) MXPA00011473A (de)
NO (1) NO20005938L (de)
NZ (1) NZ507913A (de)
PL (1) PL344303A1 (de)
RU (1) RU2211223C2 (de)
SI (1) SI20474A (de)
SK (1) SK17432000A3 (de)
UA (1) UA61997C2 (de)
WO (1) WO1999060855A1 (de)
YU (1) YU73600A (de)
ZA (1) ZA200006315B (de)

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US6403566B1 (en) 2002-06-11
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CN1311630A (zh) 2001-09-05
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