HRP20010531A2 - New biphenyl and biphenyl-analogous compounds as integrin antagonists - Google Patents

New biphenyl and biphenyl-analogous compounds as integrin antagonists Download PDF

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Publication number
HRP20010531A2
HRP20010531A2 HR20010531A HRP20010531A HRP20010531A2 HR P20010531 A2 HRP20010531 A2 HR P20010531A2 HR 20010531 A HR20010531 A HR 20010531A HR P20010531 A HRP20010531 A HR P20010531A HR P20010531 A2 HRP20010531 A2 HR P20010531A2
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HR
Croatia
Prior art keywords
substituted
butyl
phenyl
optionally substituted
group
Prior art date
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HR20010531A
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English (en)
Croatian (hr)
Inventor
Markus Albers
Klaus Urbahns
Andrea Vaupel
Michael Haerter
Delf Schmidt
Beatrix Stelte-Ludwig
Christoph Gerdes
Elke Stahl
Joerg Keldenich
Ulf Brueggemeier
Klemens Lustig
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Bayer Ag
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Publication of HRP20010531A2 publication Critical patent/HRP20010531A2/hr

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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ES2200617B1 (es) 2001-01-19 2005-05-01 Almirall Prodesfarma, S.A. Derivados de urea como antagonistas de integrinas alfa 4.
RU2003126913A (ru) * 2001-02-02 2005-03-10 Шеринг Корпорейшн (US) 3,4-дизамещенные циклобутен-1,2-дионы, как антагонисты хемокинового рецептора схс
PL208928B1 (pl) * 2001-04-16 2011-06-30 Pharmacopeia 3, 4-di-podstawione cyklobuten-1, 2-diony jako ligandy receptora CXC chemokiny
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JP2005505595A (ja) 2001-10-12 2005-02-24 シェーリング　コーポレイション Ｃｘｃ−ケモカインレセプターアンタゴニストとしての３，４−二置換マレイミド化合物
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SK8432001A3 (en) 2001-12-03
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MA25331A1 (fr) 2001-12-31
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ID30235A (id) 2001-11-15
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AU761407B2 (en) 2003-06-05
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HUP0105432A3 (en) 2002-12-28
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