HRP20020536A2 - Substituted pyrroles - Google Patents
Substituted pyrroles Download PDFInfo
- Publication number
- HRP20020536A2 HRP20020536A2 HR20020536A HRP20020536A HRP20020536A2 HR P20020536 A2 HRP20020536 A2 HR P20020536A2 HR 20020536 A HR20020536 A HR 20020536A HR P20020536 A HRP20020536 A HR P20020536A HR P20020536 A2 HRP20020536 A2 HR P20020536A2
- Authority
- HR
- Croatia
- Prior art keywords
- methyl
- indol
- pyrrole
- compound
- dione
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17155799P | 1999-12-22 | 1999-12-22 | |
| PCT/EP2000/013026 WO2001046178A2 (en) | 1999-12-22 | 2000-12-21 | Substituierte bisindolymaleimide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20020536A2 true HRP20020536A2 (en) | 2004-08-31 |
Family
ID=22624198
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20020536A HRP20020536A2 (en) | 1999-12-22 | 2000-12-21 | Substituted pyrroles |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US6281356B1 (cs) |
| EP (1) | EP1242409A2 (cs) |
| JP (1) | JP2003518112A (cs) |
| KR (1) | KR100508741B1 (cs) |
| CN (1) | CN1193027C (cs) |
| AR (1) | AR027035A1 (cs) |
| AU (1) | AU782920B2 (cs) |
| BR (1) | BR0016516A (cs) |
| CA (1) | CA2394852A1 (cs) |
| CO (1) | CO5090902A1 (cs) |
| CZ (1) | CZ20022492A3 (cs) |
| HR (1) | HRP20020536A2 (cs) |
| HU (1) | HUP0204572A3 (cs) |
| IL (1) | IL150200A0 (cs) |
| JO (1) | JO2199B1 (cs) |
| MA (1) | MA26860A1 (cs) |
| MX (1) | MXPA02006162A (cs) |
| MY (1) | MY133682A (cs) |
| NO (1) | NO20022927L (cs) |
| NZ (1) | NZ519359A (cs) |
| PE (1) | PE20011098A1 (cs) |
| PL (1) | PL357603A1 (cs) |
| RU (1) | RU2261862C2 (cs) |
| UY (1) | UY26498A1 (cs) |
| WO (1) | WO2001046178A2 (cs) |
| YU (1) | YU46302A (cs) |
| ZA (1) | ZA200204313B (cs) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030139373A1 (en) * | 2001-11-20 | 2003-07-24 | Breimer Lars Holger | Method for cancer therapy |
| TW200918046A (en) * | 2002-04-03 | 2009-05-01 | Novartis Ag | Indolylmaleimide derivatives |
| GB0303319D0 (en) | 2003-02-13 | 2003-03-19 | Novartis Ag | Organic compounds |
| RU2441000C2 (ru) * | 2009-11-27 | 2012-01-27 | Общество с ограниченной ответственностью "Молекулярные Технологии" | 4-(1-(4-(4-метоксифенилтио)-2,5-диоксо-2,5-дигидро-1н-пирро-3-ил)-1н-индол-3-ил)бутилкарбамимидотиоат и способ его применения |
| US20140303121A1 (en) | 2013-03-15 | 2014-10-09 | Plexxikon Inc. | Heterocyclic compounds and uses thereof |
| DK2970265T3 (en) | 2013-03-15 | 2018-10-01 | Plexxikon Inc | HETEROCYCLIC COMPOUNDS AND APPLICATIONS THEREOF |
| DK3272745T3 (da) | 2016-07-21 | 2019-09-02 | Inst Farmakologii Polskiej Akademii Nauk | Imidazolylsubstituerede indolderivater, der binder 5-ht7-serotoninreceptor, og farmaceutiske sammensætninger deraf |
| US10717735B2 (en) | 2017-10-13 | 2020-07-21 | Plexxikon Inc. | Solid forms of a compound for modulating kinases |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ227850A (en) | 1988-02-10 | 1991-11-26 | Hoffmann La Roche | Indole substituted pyrrole derivatives; preparatory process and medicaments for use against inflammatory immunological, bronchopulmonary or vascular disorders |
| DE3942991A1 (de) * | 1989-12-27 | 1991-07-04 | Goedecke Ag | Maleinimid-derivate und deren verwendung als arzneimittel |
| US5380746A (en) | 1989-05-05 | 1995-01-10 | Goedecke Aktiengesellschaft | Bis-(1H-indol-3-YL)-maleinimide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them |
| CA2015996C (en) * | 1989-05-05 | 2001-08-28 | Hartmut Osswald | Bis-(1h-indol-3-yl)-maleinimide derivatives and their use as pharmaceuticals |
| CA2046801C (en) * | 1990-08-07 | 2002-02-26 | Peter D. Davis | Substituted pyrroles |
| US5547976A (en) * | 1992-03-20 | 1996-08-20 | Burroughs Wellcome Co. | Further indole derivatives with antiviral activity |
| AU3761393A (en) | 1992-03-20 | 1993-10-21 | Wellcome Foundation Limited, The | Indole derivatives with antiviral activity |
| DE4217964A1 (de) * | 1992-05-30 | 1993-12-02 | Goedecke Ag | Indolocarbazol-Imide und deren Verwendung |
| PE91698A1 (es) | 1996-07-29 | 1998-12-24 | Hoffmann La Roche | Pirroles sustituidos |
| PE91498A1 (es) | 1996-07-29 | 1998-12-22 | Hoffmann La Roche | Pirroles sustituidos |
| PE91598A1 (es) | 1996-07-29 | 1998-12-24 | Hoffmann La Roche | Pirroles sustituidos |
| PT1064279E (pt) * | 1998-03-17 | 2003-10-31 | Hoffmann La Roche | Bisindolilmaleimidas substituidas para a inibicao da proliferacao celular |
-
2000
- 2000-12-15 US US09/737,685 patent/US6281356B1/en not_active Expired - Fee Related
- 2000-12-19 JO JO2000203A patent/JO2199B1/en active
- 2000-12-20 AR ARP000106792A patent/AR027035A1/es not_active Application Discontinuation
- 2000-12-20 MY MYPI20006018A patent/MY133682A/en unknown
- 2000-12-20 CO CO00096628A patent/CO5090902A1/es unknown
- 2000-12-21 JP JP2001547088A patent/JP2003518112A/ja active Pending
- 2000-12-21 CN CNB008173885A patent/CN1193027C/zh not_active Expired - Fee Related
- 2000-12-21 HR HR20020536A patent/HRP20020536A2/hr not_active Application Discontinuation
- 2000-12-21 PE PE2000001386A patent/PE20011098A1/es not_active Application Discontinuation
- 2000-12-21 AU AU37267/01A patent/AU782920B2/en not_active Ceased
- 2000-12-21 WO PCT/EP2000/013026 patent/WO2001046178A2/en not_active Ceased
- 2000-12-21 YU YU46302A patent/YU46302A/sh unknown
- 2000-12-21 MX MXPA02006162A patent/MXPA02006162A/es not_active Application Discontinuation
- 2000-12-21 CA CA002394852A patent/CA2394852A1/en not_active Abandoned
- 2000-12-21 CZ CZ20022492A patent/CZ20022492A3/cs unknown
- 2000-12-21 NZ NZ519359A patent/NZ519359A/en unknown
- 2000-12-21 RU RU2002119557/04A patent/RU2261862C2/ru not_active IP Right Cessation
- 2000-12-21 HU HU0204572A patent/HUP0204572A3/hu unknown
- 2000-12-21 UY UY26498A patent/UY26498A1/es not_active Application Discontinuation
- 2000-12-21 KR KR10-2002-7008019A patent/KR100508741B1/ko not_active Expired - Fee Related
- 2000-12-21 IL IL15020000A patent/IL150200A0/xx unknown
- 2000-12-21 PL PL00357603A patent/PL357603A1/xx not_active Application Discontinuation
- 2000-12-21 EP EP00991984A patent/EP1242409A2/en not_active Withdrawn
- 2000-12-21 BR BR0016516-6A patent/BR0016516A/pt not_active IP Right Cessation
-
2002
- 2002-05-29 ZA ZA200204313A patent/ZA200204313B/en unknown
- 2002-06-18 NO NO20022927A patent/NO20022927L/no not_active Application Discontinuation
- 2002-06-21 MA MA26707A patent/MA26860A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR0016516A (pt) | 2002-09-17 |
| JO2199B1 (en) | 2003-12-23 |
| NO20022927D0 (no) | 2002-06-18 |
| KR100508741B1 (ko) | 2005-08-17 |
| AU782920B2 (en) | 2005-09-08 |
| HK1054382A1 (en) | 2003-11-28 |
| CO5090902A1 (es) | 2001-10-30 |
| MA26860A1 (fr) | 2004-12-20 |
| PE20011098A1 (es) | 2001-10-26 |
| UY26498A1 (es) | 2001-06-29 |
| CA2394852A1 (en) | 2001-06-28 |
| IL150200A0 (en) | 2002-12-01 |
| CZ20022492A3 (cs) | 2003-02-12 |
| AU3726701A (en) | 2001-07-03 |
| MXPA02006162A (es) | 2002-12-05 |
| MY133682A (en) | 2007-11-30 |
| CN1193027C (zh) | 2005-03-16 |
| WO2001046178A3 (en) | 2001-12-06 |
| KR20020062365A (ko) | 2002-07-25 |
| EP1242409A2 (en) | 2002-09-25 |
| HUP0204572A3 (en) | 2004-07-28 |
| HUP0204572A2 (en) | 2003-05-28 |
| CN1411457A (zh) | 2003-04-16 |
| US6281356B1 (en) | 2001-08-28 |
| RU2002119557A (ru) | 2004-01-10 |
| ZA200204313B (en) | 2003-08-29 |
| JP2003518112A (ja) | 2003-06-03 |
| RU2261862C2 (ru) | 2005-10-10 |
| WO2001046178A2 (en) | 2001-06-28 |
| NZ519359A (en) | 2004-04-30 |
| PL357603A1 (en) | 2004-07-26 |
| YU46302A (sh) | 2005-06-10 |
| NO20022927L (no) | 2002-06-18 |
| AR027035A1 (es) | 2003-03-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A1OB | Publication of a patent application | ||
| ARAI | Request for the grant of a patent on the basis of the submitted results of a substantive examination of a patent application | ||
| OBST | Application withdrawn |