HRP20030174A2 - Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof - Google Patents
Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof Download PDFInfo
- Publication number
- HRP20030174A2 HRP20030174A2 HR20030174A HRP20030174A HRP20030174A2 HR P20030174 A2 HRP20030174 A2 HR P20030174A2 HR 20030174 A HR20030174 A HR 20030174A HR P20030174 A HRP20030174 A HR P20030174A HR P20030174 A2 HRP20030174 A2 HR P20030174A2
- Authority
- HR
- Croatia
- Prior art keywords
- halogen
- alkoxy
- general formula
- alkyl
- hydroxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10041671A DE10041671C1 (de) | 2000-08-10 | 2000-08-10 | Verfahren zur Herstellung von Imidazo[1,2-c][2,3]benzodiazepinen sowie Phenylessigsäureester und Oxazol-Derivate als Zwischenprodukte bei deren Herstellung |
| PCT/EP2001/008661 WO2002012247A1 (de) | 2000-08-10 | 2001-07-26 | Verfahren zur herstellung von imidazo[1,2-c][2,3]benzodiazepinen und zwischenprodukte bei deren herstellung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20030174A2 true HRP20030174A2 (en) | 2004-06-30 |
Family
ID=7653689
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20030174A HRP20030174A2 (en) | 2000-08-10 | 2001-07-26 | Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof |
Country Status (30)
| Country | Link |
|---|---|
| US (1) | US6784292B2 (cs) |
| EP (1) | EP1307460B1 (cs) |
| JP (1) | JP2004505981A (cs) |
| KR (1) | KR20030021263A (cs) |
| CN (1) | CN1205213C (cs) |
| AT (1) | ATE260921T1 (cs) |
| AU (2) | AU2001278512B2 (cs) |
| BG (1) | BG107519A (cs) |
| BR (1) | BR0112810A (cs) |
| CA (1) | CA2417804A1 (cs) |
| CZ (1) | CZ2003676A3 (cs) |
| DE (2) | DE10041671C1 (cs) |
| DK (1) | DK1307460T3 (cs) |
| EA (1) | EA005570B1 (cs) |
| EE (1) | EE200300058A (cs) |
| ES (1) | ES2217173T3 (cs) |
| HR (1) | HRP20030174A2 (cs) |
| HU (1) | HUP0301500A3 (cs) |
| IL (1) | IL154165A0 (cs) |
| MX (1) | MXPA02012913A (cs) |
| NO (1) | NO20030605D0 (cs) |
| NZ (1) | NZ523479A (cs) |
| PL (1) | PL359586A1 (cs) |
| PT (1) | PT1307460E (cs) |
| SK (1) | SK2892003A3 (cs) |
| TR (1) | TR200401281T4 (cs) |
| UA (1) | UA79737C2 (cs) |
| WO (1) | WO2002012247A1 (cs) |
| YU (1) | YU8903A (cs) |
| ZA (1) | ZA200301862B (cs) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8173806B2 (en) * | 2006-03-17 | 2012-05-08 | Mitsubishi Gas Chemical Company, Inc. | Method for production of quinazolin-4-one derivative |
| KR200453637Y1 (ko) * | 2009-06-23 | 2011-05-19 | (주)대양스톤 | 씽크대용 볼 고정장치 |
| CN104498543B (zh) * | 2015-01-22 | 2017-10-31 | 中国石油大学(华东) | 一种脂肪酶催化合成乙偶姻脂肪酸酯的方法 |
| CN104557533A (zh) * | 2015-01-22 | 2015-04-29 | 中国石油大学(华东) | 一种磷钨酸催化合成乙偶姻短链脂肪酸酯的方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19604919A1 (de) * | 1996-02-01 | 1997-08-07 | Schering Ag | Neue 2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel |
| HUP9701325A1 (hu) | 1997-07-31 | 2000-08-28 | Gyógyszerkutató Intézet Kft. | Új 2,3-benzodiazepin-származékok |
-
2000
- 2000-08-10 DE DE10041671A patent/DE10041671C1/de not_active Expired - Lifetime
-
2001
- 2001-07-26 AU AU2001278512A patent/AU2001278512B2/en not_active Ceased
- 2001-07-26 CA CA002417804A patent/CA2417804A1/en not_active Abandoned
- 2001-07-26 PL PL01359586A patent/PL359586A1/xx not_active Application Discontinuation
- 2001-07-26 PT PT01956566T patent/PT1307460E/pt unknown
- 2001-07-26 IL IL15416501A patent/IL154165A0/xx unknown
- 2001-07-26 HU HU0301500A patent/HUP0301500A3/hu unknown
- 2001-07-26 KR KR10-2003-7001796A patent/KR20030021263A/ko not_active Ceased
- 2001-07-26 ES ES01956566T patent/ES2217173T3/es not_active Expired - Lifetime
- 2001-07-26 AT AT01956566T patent/ATE260921T1/de not_active IP Right Cessation
- 2001-07-26 CN CNB018139876A patent/CN1205213C/zh not_active Expired - Fee Related
- 2001-07-26 NZ NZ523479A patent/NZ523479A/en unknown
- 2001-07-26 US US10/344,156 patent/US6784292B2/en not_active Expired - Fee Related
- 2001-07-26 DE DE50101634T patent/DE50101634D1/de not_active Expired - Fee Related
- 2001-07-26 TR TR2004/01281T patent/TR200401281T4/xx unknown
- 2001-07-26 BR BR0112810-8A patent/BR0112810A/pt not_active IP Right Cessation
- 2001-07-26 EA EA200300220A patent/EA005570B1/ru not_active IP Right Cessation
- 2001-07-26 UA UA2003032066A patent/UA79737C2/uk unknown
- 2001-07-26 AU AU7851201A patent/AU7851201A/xx active Pending
- 2001-07-26 JP JP2002518222A patent/JP2004505981A/ja active Pending
- 2001-07-26 CZ CZ2003676A patent/CZ2003676A3/cs unknown
- 2001-07-26 WO PCT/EP2001/008661 patent/WO2002012247A1/de not_active Ceased
- 2001-07-26 DK DK01956566T patent/DK1307460T3/da active
- 2001-07-26 EP EP01956566A patent/EP1307460B1/de not_active Expired - Lifetime
- 2001-07-26 HR HR20030174A patent/HRP20030174A2/hr not_active Application Discontinuation
- 2001-07-26 EE EEP200300058A patent/EE200300058A/xx unknown
- 2001-07-26 MX MXPA02012913A patent/MXPA02012913A/es active IP Right Grant
- 2001-07-26 YU YU8903A patent/YU8903A/sh unknown
- 2001-07-26 SK SK289-2003A patent/SK2892003A3/sk unknown
-
2003
- 2003-02-04 BG BG107519A patent/BG107519A/bg unknown
- 2003-02-07 NO NO20030605A patent/NO20030605D0/no not_active Application Discontinuation
- 2003-03-06 ZA ZA200301862A patent/ZA200301862B/en unknown
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| ODRP | Renewal fee for the maintenance of a patent |
Payment date: 20070627 Year of fee payment: 7 |
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| PNAN | Change of the applicant name, address/residence |
Owner name: BAYER SCHERING PHARMA AKTIENGESELLSCHAFT, DE |
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| OBST | Application withdrawn |