HRP20040850A2 - Conjugates of biologically active compounds, methods for their preparation and use formulation and pharmaceutical applications thereof - Google Patents

Conjugates of biologically active compounds, methods for their preparation and use formulation and pharmaceutical applications thereof

Info

Publication number
HRP20040850A2
HRP20040850A2 HR20040850A HRP20040850A HRP20040850A2 HR P20040850 A2 HRP20040850 A2 HR P20040850A2 HR 20040850 A HR20040850 A HR 20040850A HR P20040850 A HRP20040850 A HR P20040850A HR P20040850 A2 HRP20040850 A2 HR P20040850A2
Authority
HR
Croatia
Prior art keywords
alkyl
alkenyl
aryl
alkynyl
heteroaryl
Prior art date
Application number
HR20040850A
Other languages
English (en)
Croatian (hr)
Inventor
Burnet Michael
Guse Jan-Hinrich
Gutke Hans-Jurgen
Beck Albert
Tsotsou Georgia
Droste-Borel Irina
Reichert Jeannette
Luyten Kattie
Busch Maximilian
Wolff Michael
Moussa Khobzaoui
Margutti Simona
Meindl Thomas
Kim Gene
Barker Laurence
Original Assignee
Synovo Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synovo Gmbh filed Critical Synovo Gmbh
Publication of HRP20040850A2 publication Critical patent/HRP20040850A2/hr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K49/00—Preparations for testing in vivo
    • A61K49/0004—Screening or testing of compounds for diagnosis of disorders, assessment of conditions, e.g. renal clearance, gastric emptying, testing for diabetes, allergy, rheuma, pancreas functions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/545—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/549—Sugars, nucleosides, nucleotides or nucleic acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pathology (AREA)
  • Rheumatology (AREA)
  • Toxicology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
HR20040850A 2002-02-15 2003-02-14 Conjugates of biologically active compounds, methods for their preparation and use formulation and pharmaceutical applications thereof HRP20040850A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35743402P 2002-02-15 2002-02-15
PCT/US2003/004609 WO2003070174A2 (en) 2002-02-15 2003-02-14 Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof

Publications (1)

Publication Number Publication Date
HRP20040850A2 true HRP20040850A2 (en) 2005-08-31

Family

ID=27757618

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20040850A HRP20040850A2 (en) 2002-02-15 2003-02-14 Conjugates of biologically active compounds, methods for their preparation and use formulation and pharmaceutical applications thereof

Country Status (8)

Country Link
US (2) US20050171342A1 (de)
EP (1) EP1483277A4 (de)
AU (1) AU2003219770B2 (de)
CA (1) CA2476423A1 (de)
HR (1) HRP20040850A2 (de)
IL (1) IL163552A (de)
NZ (1) NZ535354A (de)
WO (1) WO2003070174A2 (de)

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Also Published As

Publication number Publication date
US20050171342A1 (en) 2005-08-04
WO2003070174A3 (en) 2003-11-13
US7579324B2 (en) 2009-08-25
EP1483277A4 (de) 2007-10-03
US20040087517A1 (en) 2004-05-06
WO2003070174A2 (en) 2003-08-28
NZ535354A (en) 2008-01-31
AU2003219770B2 (en) 2008-10-09
CA2476423A1 (en) 2003-08-28
IL163552A (en) 2010-11-30
AU2003219770A1 (en) 2003-09-09
EP1483277A2 (de) 2004-12-08

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