HRP20050183A2 - Preparation of 1h-imidazo [4,5-c]quinolin-4-aminesvia novel 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates - Google Patents

Preparation of 1h-imidazo [4,5-c]quinolin-4-aminesvia novel 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates

Info

Publication number
HRP20050183A2
HRP20050183A2 HR20050183A HRP20050183A HRP20050183A2 HR P20050183 A2 HRP20050183 A2 HR P20050183A2 HR 20050183 A HR20050183 A HR 20050183A HR P20050183 A HRP20050183 A HR P20050183A HR P20050183 A2 HRP20050183 A2 HR P20050183A2
Authority
HR
Croatia
Prior art keywords
imidazo
quinolin
cyano
quinoline
preparation
Prior art date
Application number
HR20050183A
Other languages
English (en)
Inventor
Merli Valeriano
Mantovani Silvia
Bianchi Stefano
Original Assignee
Teva Gy�gyszergy�r R�szv�nyt�rsas�g
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Gy�gyszergy�r R�szv�nyt�rsas�g filed Critical Teva Gy�gyszergy�r R�szv�nyt�rsas�g
Publication of HRP20050183A2 publication Critical patent/HRP20050183A2/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Breeding Of Plants And Reproduction By Means Of Culturing (AREA)
HR20050183A 2002-07-26 2003-07-28 Preparation of 1h-imidazo [4,5-c]quinolin-4-aminesvia novel 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates HRP20050183A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39859202P 2002-07-26 2002-07-26
PCT/US2003/023543 WO2004011462A1 (en) 2002-07-26 2003-07-28 Preparation of 1h-imidazo [4,5-c] quinolin-4-amines via novel 1h-imidazo [4,5-c] quinolin-4-cyano and 1h-imidazo [4,5-c] quinolin-4-carboxamide intermediates

Publications (1)

Publication Number Publication Date
HRP20050183A2 true HRP20050183A2 (en) 2005-06-30

Family

ID=31188428

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20050183A HRP20050183A2 (en) 2002-07-26 2003-07-28 Preparation of 1h-imidazo [4,5-c]quinolin-4-aminesvia novel 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates

Country Status (18)

Country Link
US (3) US6841678B2 (de)
EP (1) EP1539752B1 (de)
JP (1) JP2005537287A (de)
KR (1) KR20050030958A (de)
CN (1) CN100372847C (de)
AT (1) ATE357445T1 (de)
AU (1) AU2003254221A1 (de)
CA (1) CA2493158A1 (de)
DE (1) DE60312701T8 (de)
DK (1) DK1539752T3 (de)
ES (1) ES2282691T3 (de)
HR (1) HRP20050183A2 (de)
IL (2) IL166307A0 (de)
MX (1) MXPA05000997A (de)
PL (1) PL374866A1 (de)
PT (1) PT1539752E (de)
SI (1) SI1539752T1 (de)
WO (1) WO2004011462A1 (de)

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Also Published As

Publication number Publication date
US20050101627A1 (en) 2005-05-12
CA2493158A1 (en) 2004-02-05
AU2003254221A1 (en) 2004-02-16
CN100372847C (zh) 2008-03-05
EP1539752A1 (de) 2005-06-15
DE60312701T2 (de) 2007-12-06
PT1539752E (pt) 2007-05-31
DK1539752T3 (da) 2007-07-16
MXPA05000997A (es) 2005-05-16
US7335772B2 (en) 2008-02-26
JP2005537287A (ja) 2005-12-08
IL166307A (en) 2010-04-15
US20050119294A1 (en) 2005-06-02
US7166721B2 (en) 2007-01-23
WO2004011462A1 (en) 2004-02-05
IL166307A0 (en) 2006-01-15
KR20050030958A (ko) 2005-03-31
DE60312701T8 (de) 2008-08-21
ATE357445T1 (de) 2007-04-15
SI1539752T1 (sl) 2007-08-31
US20040063743A1 (en) 2004-04-01
PL374866A1 (en) 2005-11-14
CN1684963A (zh) 2005-10-19
ES2282691T3 (es) 2007-10-16
DE60312701D1 (de) 2007-05-03
EP1539752B1 (de) 2007-03-21
US6841678B2 (en) 2005-01-11

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