DK1539752T3 - Fremstilling af 1H-imidazo(4,5-c)quinolin-4-aminer via ny imidazo(4,5-c)quinolin 4-cyano og 1H-imidazo(4,5-c)quinolin-4-carboxamid mellemprodukter - Google Patents

Fremstilling af 1H-imidazo(4,5-c)quinolin-4-aminer via ny imidazo(4,5-c)quinolin 4-cyano og 1H-imidazo(4,5-c)quinolin-4-carboxamid mellemprodukter

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Publication number
DK1539752T3
DK1539752T3 DK03771977T DK03771977T DK1539752T3 DK 1539752 T3 DK1539752 T3 DK 1539752T3 DK 03771977 T DK03771977 T DK 03771977T DK 03771977 T DK03771977 T DK 03771977T DK 1539752 T3 DK1539752 T3 DK 1539752T3
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Prior art keywords
quinoline
imidazo
cyano
preparation
intermediates
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Application number
DK03771977T
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English (en)
Inventor
Valeriano Merli
Stefano Bianchi
Silvia Mantovani
Original Assignee
Teva Gyogyszergyar Zartkoeruee
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Application filed by Teva Gyogyszergyar Zartkoeruee filed Critical Teva Gyogyszergyar Zartkoeruee
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Publication of DK1539752T3 publication Critical patent/DK1539752T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Breeding Of Plants And Reproduction By Means Of Culturing (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK03771977T 2002-07-26 2003-07-28 Fremstilling af 1H-imidazo(4,5-c)quinolin-4-aminer via ny imidazo(4,5-c)quinolin 4-cyano og 1H-imidazo(4,5-c)quinolin-4-carboxamid mellemprodukter DK1539752T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39859202P 2002-07-26 2002-07-26
PCT/US2003/023543 WO2004011462A1 (en) 2002-07-26 2003-07-28 Preparation of 1h-imidazo [4,5-c] quinolin-4-amines via novel 1h-imidazo [4,5-c] quinolin-4-cyano and 1h-imidazo [4,5-c] quinolin-4-carboxamide intermediates

Publications (1)

Publication Number Publication Date
DK1539752T3 true DK1539752T3 (da) 2007-07-16

Family

ID=31188428

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03771977T DK1539752T3 (da) 2002-07-26 2003-07-28 Fremstilling af 1H-imidazo(4,5-c)quinolin-4-aminer via ny imidazo(4,5-c)quinolin 4-cyano og 1H-imidazo(4,5-c)quinolin-4-carboxamid mellemprodukter

Country Status (18)

Country Link
US (3) US6841678B2 (da)
EP (1) EP1539752B1 (da)
JP (1) JP2005537287A (da)
KR (1) KR20050030958A (da)
CN (1) CN100372847C (da)
AT (1) ATE357445T1 (da)
AU (1) AU2003254221A1 (da)
CA (1) CA2493158A1 (da)
DE (1) DE60312701T8 (da)
DK (1) DK1539752T3 (da)
ES (1) ES2282691T3 (da)
HR (1) HRP20050183A2 (da)
IL (2) IL166307A0 (da)
MX (1) MXPA05000997A (da)
PL (1) PL374866A1 (da)
PT (1) PT1539752E (da)
SI (1) SI1539752T1 (da)
WO (1) WO2004011462A1 (da)

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Also Published As

Publication number Publication date
US20050119294A1 (en) 2005-06-02
CA2493158A1 (en) 2004-02-05
EP1539752B1 (en) 2007-03-21
US20040063743A1 (en) 2004-04-01
PL374866A1 (en) 2005-11-14
PT1539752E (pt) 2007-05-31
ES2282691T3 (es) 2007-10-16
US7335772B2 (en) 2008-02-26
IL166307A0 (en) 2006-01-15
JP2005537287A (ja) 2005-12-08
EP1539752A1 (en) 2005-06-15
ATE357445T1 (de) 2007-04-15
CN1684963A (zh) 2005-10-19
AU2003254221A1 (en) 2004-02-16
DE60312701D1 (de) 2007-05-03
HRP20050183A2 (en) 2005-06-30
MXPA05000997A (es) 2005-05-16
US7166721B2 (en) 2007-01-23
DE60312701T8 (de) 2008-08-21
IL166307A (en) 2010-04-15
DE60312701T2 (de) 2007-12-06
KR20050030958A (ko) 2005-03-31
CN100372847C (zh) 2008-03-05
SI1539752T1 (sl) 2007-08-31
US6841678B2 (en) 2005-01-11
US20050101627A1 (en) 2005-05-12
WO2004011462A1 (en) 2004-02-05

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