HRP990023A2 - Trovafloxacin mesylate tablet - Google Patents

Trovafloxacin mesylate tablet

Info

Publication number: HRP990023A2
Authority: HR; Croatia
Prior art keywords: mixture according; tablet; trovafloxacin; tablets; mixture
Prior art date: 1998-01-21

Application number

HR60/072,013A

Other languages

English (en)

Croatian (hr)

Inventor

Christopher Michael Sinko

Original Assignee

Christopher Michael Sinko

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-01-21

Filing date

1999-01-21

Publication date

1999-08-31

1999-01-21 Application filed by Christopher Michael Sinko filed Critical Christopher Michael Sinko

1999-08-31 Publication of HRP990023A2 publication Critical patent/HRP990023A2/hr

Links

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229960005021 trovafloxacin mesylate Drugs 0.000 title claims description 20
239000000203 mixture Substances 0.000 claims description 58
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229960000497 trovafloxacin Drugs 0.000 description 20
WVPSKSLAZQPAKQ-CDMJZVDBSA-N trovafloxacin Chemical compound C([C@H]1[C@@H]([C@H]1C1)N)N1C(C(=CC=1C(=O)C(C(O)=O)=C2)F)=NC=1N2C1=CC=C(F)C=C1F WVPSKSLAZQPAKQ-CDMJZVDBSA-N 0.000 description 19
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QIQXTHQIDYTFRH-UHFFFAOYSA-N octadecanoic acid Chemical compound CCCCCCCCCCCCCCCCCC(O)=O QIQXTHQIDYTFRH-UHFFFAOYSA-N 0.000 description 1
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235000019477 peppermint oil Nutrition 0.000 description 1
230000000704 physical effect Effects 0.000 description 1
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235000013856 polydextrose Nutrition 0.000 description 1
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239000000244 polyoxyethylene sorbitan monooleate Substances 0.000 description 1
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239000011118 polyvinyl acetate Substances 0.000 description 1
239000000843 powder Substances 0.000 description 1
238000000634 powder X-ray diffraction Methods 0.000 description 1
230000002035 prolonged effect Effects 0.000 description 1
239000001327 prunus amygdalus amara l. extract Substances 0.000 description 1
238000011002 quantification Methods 0.000 description 1
238000004445 quantitative analysis Methods 0.000 description 1
239000003306 quinoline derived antiinfective agent Substances 0.000 description 1
238000004007 reversed phase HPLC Methods 0.000 description 1
230000002441 reversible effect Effects 0.000 description 1
238000005096 rolling process Methods 0.000 description 1
239000010670 sage oil Substances 0.000 description 1
150000003839 salts Chemical class 0.000 description 1
239000012898 sample dilution Substances 0.000 description 1
238000013207 serial dilution Methods 0.000 description 1
239000000741 silica gel Substances 0.000 description 1
229910002027 silica gel Inorganic materials 0.000 description 1
239000011734 sodium Substances 0.000 description 1
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235000010413 sodium alginate Nutrition 0.000 description 1
239000000661 sodium alginate Substances 0.000 description 1
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235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
229920003109 sodium starch glycolate Polymers 0.000 description 1
239000008109 sodium starch glycolate Substances 0.000 description 1
229940079832 sodium starch glycolate Drugs 0.000 description 1
239000007787 solid Substances 0.000 description 1
239000007909 solid dosage form Substances 0.000 description 1
238000000527 sonication Methods 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
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239000010935 stainless steel Substances 0.000 description 1
239000008107 starch Substances 0.000 description 1
235000019698 starch Nutrition 0.000 description 1
229940032147 starch Drugs 0.000 description 1
239000008117 stearic acid Substances 0.000 description 1
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239000000758 substrate Substances 0.000 description 1
239000000454 talc Substances 0.000 description 1
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239000001789 thuja occidentalis l. leaf oil Substances 0.000 description 1
239000010678 thyme oil Substances 0.000 description 1
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239000000196 tragacanth Substances 0.000 description 1
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239000002966 varnish Substances 0.000 description 1
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239000000811 xylitol Substances 0.000 description 1
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229960002675 xylitol Drugs 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

HR60/072,013A 1998-01-21 1999-01-21 Trovafloxacin mesylate tablet HRP990023A2 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US7201398P	1998-01-21	1998-01-21

Publications (1)

Publication Number	Publication Date
HRP990023A2 true HRP990023A2 (en)	1999-08-31

Family

ID=22105016

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HR60/072,013A HRP990023A2 (en)	1998-01-21	1999-01-21	Trovafloxacin mesylate tablet

Country Status (34)

Country	Link
US (1)	US6187341B1 (fr)
EP (1)	EP0930068A3 (fr)
JP (1)	JPH11269072A (fr)
KR (1)	KR100314977B1 (fr)
CN (1)	CN1227743A (fr)
AP (1)	AP1094A (fr)
AR (1)	AR012780A1 (fr)
AU (1)	AU758381B2 (fr)
BG (1)	BG103106A (fr)
BR (1)	BR9900116A (fr)
CA (1)	CA2259698C (fr)
CO (1)	CO4810225A1 (fr)
DZ (1)	DZ2712A1 (fr)
EA (1)	EA003247B1 (fr)
GT (1)	GT199900004A (fr)
HR (1)	HRP990023A2 (fr)
HU (1)	HUP9900154A3 (fr)
ID (1)	ID23735A (fr)
IL (1)	IL128051A0 (fr)
IS (1)	IS4947A (fr)
MA (1)	MA24747A1 (fr)
NO (1)	NO990243L (fr)
NZ (1)	NZ333838A (fr)
OA (1)	OA10958A (fr)
PA (1)	PA8466701A1 (fr)
PE (1)	PE20000169A1 (fr)
PL (1)	PL330981A1 (fr)
SG (1)	SG70666A1 (fr)
SK (1)	SK4299A3 (fr)
TN (1)	TNSN99007A1 (fr)
TR (1)	TR199900089A2 (fr)
TW (1)	TW518224B (fr)
YU (1)	YU2399A (fr)
ZA (1)	ZA99393B (fr)

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TR200101310T2 (tr) *	1998-11-10	2001-10-22	Bayer Aktiengesellschaft	Farmasötik moksifloksasin preparatı.
EP1216058A2 (fr) *	1999-09-20	2002-06-26	Alza Corporation	Procede destine a reduire la transformation polymorphique d'un medicament
ATE285821T1 (de) *	1999-10-08	2005-01-15	Affinium Pharm Inc	Fab i inhibitoren
FR2808441B1 (fr) *	2000-05-04	2004-06-18	Oreal	Utilisation de fibres dans une composition de soin ou de maquillage pour matifier la peau
DE10031043A1 (de) *	2000-06-26	2002-02-14	Bayer Ag	Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung
CA2444597A1 (fr) *	2001-04-06	2002-10-06	Affinium Pharmaceuticals, Inc.	Inhibiteurs de fab i
EP1396263A1 (fr)	2002-08-09	2004-03-10	Warner-Lambert Company	Compositions d'enrobage pour tablettes et caplets
EP1575951B1 (fr)	2002-12-06	2014-06-25	Debiopharm International SA	Composes heterocycliques, procedes de production de ceux-ci et utilisation de ceux-ci dans un traitement
CN100415284C (zh) *	2002-12-30	2008-09-03	毛友昌	六味木香片的制备方法
DE602004016831D1 (de)	2003-03-17	2008-11-13	Affinium Pharm Inc	Pharmazeutische zusammensetzungen inhibitoren von fab i und weitere antibiotika enthaltend
ES2297067T3 (es) *	2003-03-19	2008-05-01	The Jordanian Pharmaceutical Manufacturing Co. Ltd.	Composiciones farmaceuticas no higroscopicas que contienen acidos quinolinacarboxilicos de hidratados.
US8906413B2 (en) *	2003-05-12	2014-12-09	Supernus Pharmaceuticals, Inc.	Drug formulations having reduced abuse potential
WO2005009395A2 (fr) *	2003-07-23	2005-02-03	L. Perrigo Company	Composition contenant des fibres cellulosiques
EP2848614A3 (fr)	2004-06-04	2015-07-29	Debiopharm International SA	Dérivés de acrylamide et leur utilisation comme agents antibiotiques
WO2006044805A2 (fr) *	2004-10-15	2006-04-27	Supernus Pharmaceuticals, Inc.	Preparations pharmaceutiques pour lesquelles le risque d'abus est reduit
EP1973902A2 (fr) *	2005-12-05	2008-10-01	Affinium Pharmaceuticals, Inc.	Agents therapeutiques et ses procédés de fabrication et d utilisation
EP2687533B1 (fr)	2006-07-20	2017-07-19	Debiopharm International SA	Dérivés d'acrylamide en tant qu'inhibiteurs de FAB I
WO2008098374A1 (fr)	2007-02-16	2008-08-21	Affinium Pharmaceuticals, Inc.	Sels, promédicaments et polymorphes d'inhibiteurs de fab 1
SI2861608T1 (sl)	2012-06-19	2019-08-30	Debiopharm International Sa	Derivati predzdravila (E)-N-metil-N-((3-metilbenzofuran-2-IL)metil)- 3-(7-okso-5,6,7,8-tetrahidro-1 ,8-nafthiridin-3-il)akrilamid
BR122023021456A2 (pt)	2016-02-26	2024-02-20	Debiopharm International S.A.	Uso de di-hidrogeno fosfato de {6- [(e)-3-{metil[(3-metil-1-benfofuran-2- iol)metil]amino)-3- oxopro-1-en-1-il]-2-oxo-3,4-di-hidro-1,8-naftiridin-1(2h)- il}metila para tratamento de osteomielite do pé diabético e composição farmacêutica
LT3923914T (lt)	2019-02-14	2023-07-25	Debiopharm International S.A.	Afabicino kompozicija, jos gamybos būdas
CN113939306B (zh)	2019-06-14	2024-07-19	德彪药业国际股份公司	用于治疗涉及生物膜的细菌感染的药物及其用途
JP2025529185A (ja) *	2022-08-30	2025-09-04	パンネックスセラピューティクスインコーポレイテッド	パネキシン－１調節剤及びパネキシン－１が関与する疾患の治療方法

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DE3601566A1 (de) *	1986-01-21	1987-07-23	Bayer Ag	Pharmazeutische zubereitungen von ciprofloxacin
US5286754A (en)	1986-01-21	1994-02-15	Bayer Aktiengesellschaft	Pharmaceutical formulations of ciprofloxacin
US4957554A (en)	1989-08-16	1990-09-18	Minnesota Mining And Manufacturing Company	Dimensionally-controlled ceramics
DE4120646A1 (de)	1991-06-22	1992-12-24	Bayer Ag	7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate
SK23898A3 (en) *	1995-08-29	1999-05-07	Pfizer	Zwitterionic forms of trovafloxacin

1999
- 1999-01-11 PA PA19998466701A patent/PA8466701A1/es unknown
- 1999-01-13 EP EP99300258A patent/EP0930068A3/fr not_active Withdrawn
- 1999-01-14 IL IL12805199A patent/IL128051A0/xx unknown
- 1999-01-14 AP APAP/P/1999/001443A patent/AP1094A/en active
- 1999-01-14 SK SK42-99A patent/SK4299A3/sk unknown
- 1999-01-14 TR TR1999/00089A patent/TR199900089A2/xx unknown
- 1999-01-15 PE PE1999000036A patent/PE20000169A1/es not_active Application Discontinuation
- 1999-01-15 MA MA25433A patent/MA24747A1/fr unknown
- 1999-01-15 GT GT199900004A patent/GT199900004A/es unknown
- 1999-01-15 ID IDP990036D patent/ID23735A/id unknown
- 1999-01-15 OA OA9900009A patent/OA10958A/en unknown
- 1999-01-19 CA CA002259698A patent/CA2259698C/fr not_active Expired - Fee Related
- 1999-01-19 AR ARP990100191A patent/AR012780A1/es not_active Application Discontinuation
- 1999-01-19 BR BR9900116-0A patent/BR9900116A/pt not_active IP Right Cessation
- 1999-01-19 JP JP11010298A patent/JPH11269072A/ja active Pending
- 1999-01-19 IS IS4947A patent/IS4947A/is unknown
- 1999-01-20 KR KR1019990001589A patent/KR100314977B1/ko not_active Expired - Fee Related
- 1999-01-20 ZA ZA9900393A patent/ZA99393B/xx unknown
- 1999-01-20 NO NO990243A patent/NO990243L/no not_active Application Discontinuation
- 1999-01-20 NZ NZ333838A patent/NZ333838A/xx unknown
- 1999-01-20 HU HU9900154A patent/HUP9900154A3/hu unknown
- 1999-01-20 CN CN99101232A patent/CN1227743A/zh active Pending
- 1999-01-20 YU YU2399A patent/YU2399A/sh unknown
- 1999-01-20 AU AU12173/99A patent/AU758381B2/en not_active Ceased
- 1999-01-20 DZ DZ990013A patent/DZ2712A1/fr active
- 1999-01-20 PL PL99330981A patent/PL330981A1/xx unknown
- 1999-01-20 US US09/233,823 patent/US6187341B1/en not_active Expired - Fee Related
- 1999-01-20 SG SG1999000117A patent/SG70666A1/en unknown
- 1999-01-20 TN TNTNSN99007A patent/TNSN99007A1/fr unknown
- 1999-01-21 BG BG103106A patent/BG103106A/xx unknown
- 1999-01-21 HR HR60/072,013A patent/HRP990023A2/hr not_active Application Discontinuation
- 1999-01-21 CO CO99003190A patent/CO4810225A1/es unknown
- 1999-01-21 TW TW088100897A patent/TW518224B/zh not_active IP Right Cessation
- 1999-01-21 EA EA199900046A patent/EA003247B1/ru not_active IP Right Cessation

Also Published As

Publication number	Publication date
PA8466701A1 (es)	2000-09-29
DZ2712A1 (fr)	2003-09-01
AP9901443A0 (en)	1999-03-31
CN1227743A (zh)	1999-09-08
EA003247B1 (ru)	2003-02-27
AP1094A (en)	2002-08-19
IS4947A (is)	1999-07-22
HUP9900154A2 (hu)	1999-09-28
EA199900046A3 (ru)	1999-12-29
CA2259698A1 (fr)	1999-07-21
JPH11269072A (ja)	1999-10-05
NZ333838A (en)	2000-03-27
TR199900089A3 (tr)	1999-10-21
IL128051A0 (en)	1999-11-30
BR9900116A (pt)	2000-05-02
KR100314977B1 (ko)	2001-11-24
NO990243L (no)	1999-07-22
HU9900154D0 (en)	1999-03-29
TW518224B (en)	2003-01-21
PE20000169A1 (es)	2000-03-10
AU1217399A (en)	1999-08-12
NO990243D0 (no)	1999-01-20
TNSN99007A1 (fr)	2005-11-10
ID23735A (id)	2000-05-11
OA10958A (en)	2001-10-31
EA199900046A2 (ru)	1999-08-26
BG103106A (en)	1999-08-31
TR199900089A2 (xx)	1999-10-21
AR012780A1 (es)	2000-11-08
GT199900004A (es)	2000-07-08
US6187341B1 (en)	2001-02-13
YU2399A (sh)	2002-06-19
EP0930068A3 (fr)	1999-12-22
MA24747A1 (fr)	1999-10-01
EP0930068A2 (fr)	1999-07-21
SG70666A1 (en)	2000-02-22
SK4299A3 (en)	2000-06-12
AU758381B2 (en)	2003-03-20
KR19990068014A (ko)	1999-08-25
CO4810225A1 (es)	1999-06-30
PL330981A1 (en)	1999-08-02
ZA99393B (en)	2000-07-21
CA2259698C (fr)	2003-04-15
HUP9900154A3 (en)	2000-12-28

Legal Events

Date	Code	Title	Description
1999-01-21	AIPI	Request for the grant of a patent on the basis of a substantive examination of a patent application
1999-08-31	A1OB	Publication of a patent application
2003-01-08	ODRP	Renewal fee for the maintenance of a patent	Payment date: 20030108 Year of fee payment: 5
2005-09-20	ODBC	Application rejected

Publication	Publication Date	Title
HRP990023A2 (en)	1999-08-31	Trovafloxacin mesylate tablet
TWI409064B (zh)	2013-09-21	Pharmaceutical composition
RU2428178C2 (ru)	2011-09-10	Сахарные покрытия и способы их применения
KR101774676B1 (ko)	2017-09-04	히드로모르폰 및 날록손을 포함하는 제약 조성물
HU227397B1 (en)	2011-05-30	Pharmaceutical formulations containing darifenacin
CN105832687A (zh)	2016-08-10	包含氢吗啡酮和纳洛酮的药物组合物
CZ20011845A3 (cs)	2001-08-15	Farmaceutické přípravky obsahující cefuroximaxetil
EP1901719A2 (fr)	2008-03-26	Formulation de benzimidazole
KR100582350B1 (ko)	2006-05-22	탐수로신 염산염의 경구투여용 조성물 및 이의 서방성과립 제제
HU229569B1 (hu)	2014-02-28	Szelektív szerotoninújrafelvétel-gátlók szabályozott kibocsátású többrészecskés kiszerelései
HRP20040959A2 (en)	2004-12-31	Solid dispersion composition
WO2010046418A1 (fr)	2010-04-29	Composition pharmaceutique contenant du lévétiracétam
EP2435029B1 (fr)	2016-12-14	Composition pharmaceutique de tamsulosine
US20100172982A1 (en)	2010-07-08	Sustained release formulations of divalproex sodium
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JP2009513622A (ja)	2009-04-02	ロサルタンの医薬製剤
AU2005313262A1 (en)	2006-06-15	Tablets for the sustained release of indapamide and preparation method thereof
EP3501504A1 (fr)	2019-06-26	Comprimé à libération modifiée de palipéridone et son procédé de préparation
US20070020334A1 (en)	2007-01-25	Benzimidazole formulation
MXPA01009934A (es)	2002-06-21	Sistema de recubrimiento.
CZ9399A3 (cs)	2000-06-14	Tableta obsahující methansulfonát trovafloxacinu
JP2009538905A (ja)	2009-11-12	感湿性薬物を含んで成る安定性製剤及びその製造方法
CA2659179A1 (fr)	2008-02-14	Stabilisation de lorazepam sous forme de dosage a desintegration orale
HK1019558A (en)	2000-02-18	Trovafloxacin mesylate tablet
CN114652685A (zh)	2022-06-24	一种高生物利用度的伊曲康唑胶囊剂