HU224814B1 - Use of propane-1,3-diol derivative for the preparation of a medicament useful for the topical treating of inflammatory and immune diseases - Google Patents
Use of propane-1,3-diol derivative for the preparation of a medicament useful for the topical treating of inflammatory and immune diseases Download PDFInfo
- Publication number
- HU224814B1 HU224814B1 HU9800034A HUP9800034A HU224814B1 HU 224814 B1 HU224814 B1 HU 224814B1 HU 9800034 A HU9800034 A HU 9800034A HU P9800034 A HUP9800034 A HU P9800034A HU 224814 B1 HU224814 B1 HU 224814B1
- Authority
- HU
- Hungary
- Prior art keywords
- disease
- compound
- disorder
- administered
- propane
- Prior art date
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- 208000027866 inflammatory disease Diseases 0.000 title claims 2
- 238000002360 preparation method Methods 0.000 title description 9
- 230000002757 inflammatory effect Effects 0.000 title description 4
- YPFDHNVEDLHUCE-UHFFFAOYSA-N propane-1,3-diol Chemical class OCCCO YPFDHNVEDLHUCE-UHFFFAOYSA-N 0.000 title 1
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- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Immunology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP34250395 | 1995-12-28 | ||
| PCT/JP1996/003757 WO1997024112A1 (en) | 1995-12-28 | 1996-12-24 | External preparation |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HUP9800034A2 HUP9800034A2 (hu) | 1999-05-28 |
| HUP9800034A3 HUP9800034A3 (en) | 1999-12-28 |
| HU224814B1 true HU224814B1 (en) | 2006-02-28 |
Family
ID=18354257
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU9800034A HU224814B1 (en) | 1995-12-28 | 1996-12-24 | Use of propane-1,3-diol derivative for the preparation of a medicament useful for the topical treating of inflammatory and immune diseases |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US6121329A (de) |
| EP (1) | EP0812588B1 (de) |
| AT (1) | ATE279185T1 (de) |
| AU (1) | AU705320B2 (de) |
| CA (1) | CA2213989C (de) |
| CZ (1) | CZ285953B6 (de) |
| DE (1) | DE69633613T2 (de) |
| ES (1) | ES2230571T3 (de) |
| HU (1) | HU224814B1 (de) |
| IL (1) | IL121625A (de) |
| NZ (1) | NZ324453A (de) |
| PT (1) | PT812588E (de) |
| RU (1) | RU2156127C2 (de) |
| SI (1) | SI0812588T1 (de) |
| SK (1) | SK282225B6 (de) |
| WO (1) | WO1997024112A1 (de) |
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| JP2002241272A (ja) * | 1996-07-18 | 2002-08-28 | Mitsubishi Pharma Corp | 医薬処方組成物 |
| US6476004B1 (en) | 1996-07-18 | 2002-11-05 | Mitsubishi Pharma Corporation | Pharmaceutical composition |
| JPH11209277A (ja) * | 1998-01-19 | 1999-08-03 | Yoshitomi Pharmaceut Ind Ltd | 医薬組成物 |
| GB9624038D0 (en) | 1996-11-19 | 1997-01-08 | Sandoz Ltd | Organic compounds |
| KR20000075745A (ko) | 1997-02-27 | 2000-12-26 | 가마후라 아키오 | 의약 조성물 |
| CA2326222C (en) | 1998-04-27 | 2008-09-23 | Fujisawa Pharmaceutical Co., Ltd. | Medicinal compositions |
| US20020006901A1 (en) * | 1999-02-05 | 2002-01-17 | Aldo T. Iacono | Use of aerosolized cyclosporine for prevention and treatment of pulmonary disease |
| US6541462B1 (en) * | 1999-03-25 | 2003-04-01 | Center For Molecular Medicine And Immunology | Sphingomyelin enhancement of tumor therapy |
| US7683044B2 (en) * | 1999-03-25 | 2010-03-23 | Center For Molecular Medicine And Immunology | Sphingomyelin therapy of autoimmune disease |
| EP1315735A4 (de) | 2000-08-31 | 2005-04-06 | Merck & Co Inc | Phosphat-derivate als immunoregulatorische verbindungen |
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| US20030124174A1 (en) * | 2001-10-25 | 2003-07-03 | Endo Pharmaceuticals, Inc | Method for treating non-neuropathic pain |
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| RU2220738C1 (ru) * | 2002-08-30 | 2004-01-10 | Гапонюк Петр Яковлевич | Средство для лечения ринита |
| KR20050092429A (ko) * | 2003-01-22 | 2005-09-21 | 니찌방 가부시기가이샤 | 안질환 치료용 경피 흡수형 제제, 그 사용, 및 안질환치료약의 눈의 국소 조직으로의 이행 방법 |
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| RU2233163C1 (ru) * | 2003-04-30 | 2004-07-27 | Государственное учреждение "Нижегородский научно-исследовательский кожно-венерологический институт" | Способ лечения акантолитической пузырчатки |
| EP1484057A1 (de) * | 2003-06-06 | 2004-12-08 | Aventis Pharma Deutschland GmbH | Verwendung von 2-amino-1,3-propandiolderivaten zur herstrllung eines medikaments zur behandlung von bestimmten schmerzen |
| US7524887B2 (en) | 2003-06-06 | 2009-04-28 | Sanofi-Aventis Deutschland Gmbh | 2-amino-1,3-propanediol compounds for the treatment of acute pain |
| BRPI0414193A (pt) * | 2003-09-09 | 2006-10-31 | 3M Innovative Properties Co | composição antimicrobiana, kit antimicrobiano e métodos de usar a composição e de aplicar uma composição antimicrobiana a um substrato |
| US20050058673A1 (en) | 2003-09-09 | 2005-03-17 | 3M Innovative Properties Company | Antimicrobial compositions and methods |
| GB0324210D0 (en) | 2003-10-15 | 2003-11-19 | Novartis Ag | Organic compounds |
| GB0329498D0 (en) * | 2003-12-19 | 2004-01-28 | Novartis Ag | Organic compounds |
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| NZ549162A (en) | 2004-02-24 | 2009-12-24 | Sankyo Co | Amino-pyrrol alcohol compounds |
| US20050232894A1 (en) * | 2004-04-20 | 2005-10-20 | Weiner Gregory M | Antimicrobial skin treatment composition and methods for producing and using an antimicrobial skin treatment composition |
| PL1773307T3 (pl) * | 2004-07-30 | 2015-03-31 | Novartis Ag | Preparaty 2-amino-1,3-propanodioli i ich analogów |
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| GB0504544D0 (en) * | 2005-03-04 | 2005-04-13 | Novartis Ag | Organic compounds |
| BRPI0608690B8 (pt) | 2005-03-10 | 2021-05-25 | 3M Innovative Properties Co | uso de uma composição antimicrobiana |
| WO2006099325A2 (en) | 2005-03-10 | 2006-09-21 | 3M Innovative Properties Company | Methods of treating ear infections |
| US20060229364A1 (en) * | 2005-03-10 | 2006-10-12 | 3M Innovative Properties Company | Antiviral compositions and methods of use |
| BRPI0608691A2 (pt) | 2005-03-10 | 2010-12-07 | 3M Innovative Properties Company | composição antimicrobiana, e, métodos para matar ou inativar microorganismos em tecido da mucosa de um mamìfero, para tratar uma lesão ou ferimento infectado, para descolonização de microorganismos, para proporcionar eficácia antimicrobiana residual sobre uma superfìcie e para tratar uma condição |
| US8633161B2 (en) * | 2005-03-24 | 2014-01-21 | The Ohio State University Research Foundation | Therapeutic agents for the treatment of leukemia |
| PT1905453E (pt) * | 2005-07-13 | 2012-12-04 | Santen Pharmaceutical Co Ltd | Composição conservante para utilização oftálmica |
| WO2007098139A2 (en) * | 2006-02-21 | 2007-08-30 | The Ohio State University Research Foundation | Anticancer agents |
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| US20080075793A1 (en) * | 2006-09-21 | 2008-03-27 | Dunshee Wayne K | Antiviral compositions and methods of use |
| EP3733161A1 (de) | 2007-10-12 | 2020-11-04 | Novartis AG | Zusammensetzung mit sphingosin-1-phosphat (s1p)-rezeptormodulatoren |
| RU2361604C1 (ru) * | 2007-10-29 | 2009-07-20 | Федеральное агентство по высокотехнологичной медицинской помощи Федеральное государственное учреждение "Уральский научно-исследовательский институт дерматовенерологии и иммунопатологии" (ФГУ УрНИИДВиИ Росмедтехнологий) | Способ лечения атопического дерматита |
| PL2278960T5 (pl) | 2008-03-17 | 2020-06-29 | Actelion Pharmaceuticals Ltd. | Schemat dawkowania dla selektywnego agonisty receptora sip1 |
| US8461362B2 (en) * | 2009-04-13 | 2013-06-11 | The Ohio State University Research Foundation | Protein phosphatase 2A-activating agents |
| WO2010121111A1 (en) * | 2009-04-17 | 2010-10-21 | The Ohio State University Research Foundation | Antiadhesion agents |
| WO2011009634A2 (en) * | 2009-07-24 | 2011-01-27 | Ratiopharm Gmbh | Process for producing fingolimod salts |
| CN101966145A (zh) * | 2010-09-21 | 2011-02-09 | 浙江大学 | 2-氨基-2-(2-[4-辛基苯基]乙基)-1,3-丙二醇盐酸盐制剂及其制备方法 |
| WO2012071524A1 (en) | 2010-11-24 | 2012-05-31 | Ratiopharm Gmbh | Arylsulfonate salts of fingolimod and processes for preparation thereof |
| US8309768B2 (en) | 2010-11-29 | 2012-11-13 | The Ohio State University Research Foundation | FTY720-derived anticancer agents |
| JP6111202B2 (ja) | 2011-01-07 | 2017-04-05 | ノバルティス アーゲー | 免疫抑制製剤 |
| AR085749A1 (es) | 2011-04-01 | 2013-10-23 | Novartis Ag | Formulaciones |
| RU2496486C1 (ru) | 2012-07-11 | 2013-10-27 | Александр Васильевич Иващенко | Фармацевтическая композиция с улучшенной сыпучестью, лекарственное средство, способ получения и применение |
| AU2014209141B2 (en) | 2013-01-24 | 2018-05-10 | Palvella Therapeutics, Inc. | Compositions for transdermal delivery of mTOR inhibitors |
| CN105611917A (zh) | 2013-10-11 | 2016-05-25 | 帝国制药美国公司 | 局部鞘氨醇-1-磷酸酯受体激动剂制剂及其使用方法 |
| US10675254B2 (en) | 2013-10-11 | 2020-06-09 | Teikoku Seiyaku Co., Ltd. | Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same |
| US9925138B2 (en) | 2015-01-20 | 2018-03-27 | Handa Pharmaceuticals, Llc | Stable solid fingolimod dosage forms |
| WO2016135644A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
| EP3565520B1 (de) | 2017-01-06 | 2026-02-25 | Palvella Therapeutics, Inc. | Wasserfreie zusammensetzungen von mtor-hemmern und verfahren zur verwendung |
| US10798783B2 (en) * | 2017-02-15 | 2020-10-06 | Continuous Composites Inc. | Additively manufactured composite heater |
| US11434200B2 (en) | 2017-03-09 | 2022-09-06 | Novartis Ag | Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof |
| CN115300508A (zh) * | 2017-07-05 | 2022-11-08 | 艾缇亚(上海)制药有限公司 | 包含孟鲁司特与贻贝粘附蛋白的组合的局部制剂 |
| US11000513B2 (en) | 2018-07-02 | 2021-05-11 | Palvella Therapeutics, Inc. | Anhydrous compositions of mTOR inhibitors and methods of use |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU374086A1 (ru) * | 1971-06-11 | 1973-03-20 | ЛЕКАРСТВЕННОЕ СРЕДСТВО''^ --''ОсНАЯ'•'^^^bju;r---jc^'-;^..':. :0 •--.:А |:'*''~'"~~ •' - ——«-.«aSJ^iH. | |
| SE7510988L (sv) * | 1975-10-01 | 1977-04-02 | Draco Ab | Nya farmaceutiskt aktiva foreningar |
| US4861800A (en) * | 1987-08-18 | 1989-08-29 | Buyske Donald A | Method for administering the drug deprenyl so as to minimize the danger of side effects |
| EP0356399A3 (de) * | 1988-08-26 | 1991-03-20 | Sandoz Ag | Substituierte 4-Azatricyclo (22.3.1.04.9) octacos-18-en-Derivate, Verfahren zu ihrer Herstellung und die sie enthaltenden pharmazeutischen Zusammensetzungen |
| EP0501579A1 (de) * | 1991-02-28 | 1992-09-02 | Merck Frosst Canada Inc. | Naphthalinlactone als Inhibitoren der Leukotrien-Biosynthese |
| IL102236A0 (en) * | 1991-06-27 | 1993-01-14 | Ltt Inst Co Ltd | Topical preparations containing cyclosporin |
| IT1252865B (it) * | 1991-12-31 | 1995-06-28 | Lifegroup Spa | N-acilderivati di aminoalcooli attivi come autocoidi locali ed utilizzabili nella terapia dei processi autoimmuni |
| IT1252866B (it) * | 1991-12-31 | 1995-06-28 | Lifegroup Spa | N-acilderivati di aminoalcooli con acidi policarbossilici atti alla modulazione dei mastociti nei processi infiammatori su base neuroimmunogenica |
| DE69321823T2 (de) * | 1992-10-21 | 1999-06-02 | Taito Co., Ltd., Tokio/Tokyo | 2-amino-1, 3- propandiolverbindung und immunosuppressium |
| JPH06256182A (ja) * | 1993-03-05 | 1994-09-13 | L T T Kenkyusho:Kk | 外用製剤 |
| JPH07188046A (ja) * | 1993-12-27 | 1995-07-25 | L T T Kenkyusho:Kk | シクロスポリン含有外用治療薬及びその製造方法 |
| WO1995022343A1 (en) * | 1994-02-17 | 1995-08-24 | Shiseido Company, Ltd. | Cyclosporin-containing emulsion composition |
| JPH1180026A (ja) * | 1997-09-02 | 1999-03-23 | Yoshitomi Pharmaceut Ind Ltd | 新規免疫抑制剤、その使用方法およびその同定方法 |
-
1996
- 1996-12-24 WO PCT/JP1996/003757 patent/WO1997024112A1/ja not_active Ceased
- 1996-12-24 DE DE69633613T patent/DE69633613T2/de not_active Expired - Lifetime
- 1996-12-24 ES ES96942623T patent/ES2230571T3/es not_active Expired - Lifetime
- 1996-12-24 CZ CZ972704A patent/CZ285953B6/cs not_active IP Right Cessation
- 1996-12-24 NZ NZ324453A patent/NZ324453A/xx not_active IP Right Cessation
- 1996-12-24 PT PT96942623T patent/PT812588E/pt unknown
- 1996-12-24 CA CA002213989A patent/CA2213989C/en not_active Expired - Lifetime
- 1996-12-24 US US08/894,728 patent/US6121329A/en not_active Expired - Lifetime
- 1996-12-24 RU RU97115893/14A patent/RU2156127C2/ru active
- 1996-12-24 IL IL12162596A patent/IL121625A/en not_active IP Right Cessation
- 1996-12-24 HU HU9800034A patent/HU224814B1/hu unknown
- 1996-12-24 EP EP96942623A patent/EP0812588B1/de not_active Expired - Lifetime
- 1996-12-24 AT AT96942623T patent/ATE279185T1/de active
- 1996-12-24 SK SK1157-97A patent/SK282225B6/sk not_active IP Right Cessation
- 1996-12-24 SI SI9630694T patent/SI0812588T1/xx unknown
- 1996-12-24 AU AU11729/97A patent/AU705320B2/en not_active Expired
-
2000
- 2000-06-12 US US09/592,550 patent/US6197829B1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| RU2156127C2 (ru) | 2000-09-20 |
| ATE279185T1 (de) | 2004-10-15 |
| IL121625A0 (en) | 1998-02-08 |
| EP0812588B1 (de) | 2004-10-13 |
| WO1997024112A1 (en) | 1997-07-10 |
| DE69633613D1 (de) | 2004-11-18 |
| CA2213989A1 (en) | 1997-07-10 |
| HUP9800034A3 (en) | 1999-12-28 |
| EP0812588A1 (de) | 1997-12-17 |
| DE69633613T2 (de) | 2006-02-09 |
| PT812588E (pt) | 2005-01-31 |
| CZ270497A3 (cs) | 1998-01-14 |
| SK282225B6 (sk) | 2001-12-03 |
| AU705320B2 (en) | 1999-05-20 |
| HUP9800034A2 (hu) | 1999-05-28 |
| NZ324453A (en) | 2000-03-27 |
| US6121329A (en) | 2000-09-19 |
| ES2230571T3 (es) | 2005-05-01 |
| SI0812588T1 (en) | 2005-02-28 |
| EP0812588A4 (de) | 2002-11-06 |
| IL121625A (en) | 2001-09-13 |
| CZ285953B6 (cs) | 1999-12-15 |
| US6197829B1 (en) | 2001-03-06 |
| AU1172997A (en) | 1997-07-28 |
| CA2213989C (en) | 2007-05-29 |
| SK115797A3 (en) | 1998-02-04 |
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