HUT70496A - 3-phenylureido-azepin-2-one and benzazepin-2-one derivatives, process for producing thereof, and pharmaceutical compositions conprising them - Google Patents

3-phenylureido-azepin-2-one and benzazepin-2-one derivatives, process for producing thereof, and pharmaceutical compositions conprising them Download PDF

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Publication number
HUT70496A
HUT70496A HU9402195A HU9402195A HUT70496A HU T70496 A HUT70496 A HU T70496A HU 9402195 A HU9402195 A HU 9402195A HU 9402195 A HU9402195 A HU 9402195A HU T70496 A HUT70496 A HU T70496A
Authority
HU
Hungary
Prior art keywords
phenyl
oxo
ureido
tert
butyl
Prior art date
Application number
HU9402195A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9402195D0 (en
Inventor
John A Lowe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of HU9402195D0 publication Critical patent/HU9402195D0/hu
Publication of HUT70496A publication Critical patent/HUT70496A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU9402195A 1992-01-27 1992-12-16 3-phenylureido-azepin-2-one and benzazepin-2-one derivatives, process for producing thereof, and pharmaceutical compositions conprising them HUT70496A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US82567792A 1992-01-27 1992-01-27

Publications (2)

Publication Number Publication Date
HU9402195D0 HU9402195D0 (en) 1994-09-28
HUT70496A true HUT70496A (en) 1995-10-30

Family

ID=25244657

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9402195A HUT70496A (en) 1992-01-27 1992-12-16 3-phenylureido-azepin-2-one and benzazepin-2-one derivatives, process for producing thereof, and pharmaceutical compositions conprising them

Country Status (19)

Country Link
EP (1) EP0625145A1 (de)
JP (1) JPH07503465A (de)
KR (1) KR950700257A (de)
CN (1) CN1074903A (de)
AU (1) AU3276193A (de)
BR (1) BR9207071A (de)
CA (1) CA2117367A1 (de)
CZ (1) CZ391092A3 (de)
FI (1) FI943513A0 (de)
HU (1) HUT70496A (de)
IL (1) IL104472A0 (de)
MX (1) MX9300409A (de)
NO (1) NO942775L (de)
NZ (1) NZ245759A (de)
RU (1) RU94038063A (de)
TW (1) TW213901B (de)
WO (1) WO1993015059A1 (de)
YU (1) YU4393A (de)
ZA (1) ZA93582B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2097688A1 (es) * 1993-07-14 1997-04-01 Pfizer Hexahidroazepinonas y tetrahidrobenzazepinonas sustituidas.
AU6686694A (en) * 1993-07-26 1995-02-20 Pfizer Inc. Tetrahydro-1h-benzazepinones and hexahydroazepinones as selective cholecystokinin-b receptor antagonists
DK0730581T3 (da) * 1993-11-22 2001-11-26 Merck & Co Inc 3-acylaminobezazepiner
US5453424A (en) * 1993-11-22 1995-09-26 Merck & Co., Inc. Furanodiazepines
FI971378L (fi) * 1994-10-04 1997-04-03 Pfizer Menetelmiä ja välituotteita 3-aminobentso(b)-atsepinonien valmistusta varten
JPH10511928A (ja) 1994-10-14 1998-11-17 グラクソ、ウェルカム、ソシエタ、ペル、アツィオーニ 睡眠障害の治療のためのｃｃｋ−ｂレセプター拮抗薬の使用
DE10153348A1 (de) 2001-10-29 2003-05-08 Gruenenthal Gmbh Substituierte Benzo(b)azepin-2-on-Verbindungen
KR20080031281A (ko) * 2005-06-16 2008-04-08 노파르티스 아게 락탐을 함유하는 ｈｃｖ 억제제

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0166357A3 (de) * 1984-06-26 1988-10-26 Merck & Co. Inc. Kondensierte Benzo-Laktame und deren pharmazeutische Zusammensetzungen
US4767756A (en) * 1987-07-17 1988-08-30 E. R. Squibb & Sons, Inc. 3-substituted benzazepines
EP0322779A3 (de) * 1987-12-29 1991-05-08 Yoshitomi Pharmaceutical Industries, Ltd. Benzolaktam-Verbindungen und deren pharmazeutische Verwendungen
US5206234A (en) * 1990-10-22 1993-04-27 Merck & Co., Inc. Benzolactam analogs as antagonists of cck

Also Published As

Publication number Publication date
AU3276193A (en) 1993-09-01
TW213901B (de) 1993-10-01
FI943513A7 (fi) 1994-07-26
NO942775L (no) 1994-09-20
JPH07503465A (ja) 1995-04-13
CA2117367A1 (en) 1993-08-05
EP0625145A1 (de) 1994-11-23
IL104472A0 (en) 1993-05-13
FI943513L (fi) 1994-07-26
YU4393A (sr) 1996-01-09
BR9207071A (pt) 1995-12-05
MX9300409A (es) 1993-07-01
WO1993015059A1 (en) 1993-08-05
HU9402195D0 (en) 1994-09-28
NO942775D0 (no) 1994-07-26
CN1074903A (zh) 1993-08-04
RU94038063A (ru) 1996-05-27
KR950700257A (ko) 1995-01-16
CZ391092A3 (en) 1994-01-19
NZ245759A (en) 1997-06-24
FI943513A0 (fi) 1994-07-26
ZA93582B (en) 1994-07-27

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Legal Events

Date Code Title Description
DFC4 Cancellation of temporary protection due to refusal